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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
9
hits in this display
Target
Mitogen-activated protein kinase 14
(Homo sapiens (Human))
Everbrilliant Pharma
US Patent
Ligand
BDBM50295553
(4-(4-(4-fluorophenyl)-1-(3-phenylpropyl)-5-(pyridi...)
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Affinity Data
Ki: 13nM
Assay Description:
FP signals were measured with a PHERAstar microplate reader (BMG Labtech) using black, low-binding half-area 96 well plates (Corning). Each binding d...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
Purchase
CHEMBL
PC cid
PC sid
Patents
In Depth
Details
US Patent
Copy BDB DOI
Target
Mitogen-activated protein kinase 14
(Homo sapiens (Human))
Everbrilliant Pharma
US Patent
Ligand
BDBM50295553
(4-(4-(4-fluorophenyl)-1-(3-phenylpropyl)-5-(pyridi...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 13nM
Assay Description:
FP signals were measured with a PHERAstar microplate reader (BMG Labtech) using black, low-binding half-area 96 well plates (Corning). Each binding d...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
Purchase
CHEMBL
PC cid
PC sid
Patents
In Depth
Details
US Patent
Copy BDB DOI
Target
Mitogen-activated protein kinase 14
(Homo sapiens (Human))
Everbrilliant Pharma
US Patent
Ligand
BDBM50295553
(4-(4-(4-fluorophenyl)-1-(3-phenylpropyl)-5-(pyridi...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 13nM
Assay Description:
FP signals were measured with a PHERAstar microplate reader (BMG Labtech) using black, low-binding half-area 96 well plates (Corning). Each binding d...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
Purchase
CHEMBL
PC cid
PC sid
Patents
In Depth
Details
US Patent
Copy BDB DOI
Target
Mitogen-activated protein kinase 14
(Homo sapiens (Human))
Everbrilliant Pharma
US Patent
Ligand
BDBM50295553
(4-(4-(4-fluorophenyl)-1-(3-phenylpropyl)-5-(pyridi...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 210nM
Assay Description:
FP signals were measured with a PHERAstar microplate reader (BMG Labtech) using black, low-binding half-area 96 well plates (Corning). Each binding d...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
Purchase
CHEMBL
PC cid
PC sid
Patents
In Depth
Details
US Patent
Copy BDB DOI
Target
Mitogen-activated protein kinase 14
(Homo sapiens (Human))
Everbrilliant Pharma
US Patent
Ligand
BDBM50295553
(4-(4-(4-fluorophenyl)-1-(3-phenylpropyl)-5-(pyridi...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 210nM
Assay Description:
FP signals were measured with a PHERAstar microplate reader (BMG Labtech) using black, low-binding half-area 96 well plates (Corning). Each binding d...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
Purchase
CHEMBL
PC cid
PC sid
Patents
In Depth
Details
US Patent
Copy BDB DOI
Target
Mitogen-activated protein kinase 14
(Homo sapiens (Human))
Everbrilliant Pharma
US Patent
Ligand
BDBM50295553
(4-(4-(4-fluorophenyl)-1-(3-phenylpropyl)-5-(pyridi...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 210nM
Assay Description:
FP signals were measured with a PHERAstar microplate reader (BMG Labtech) using black, low-binding half-area 96 well plates (Corning). Each binding d...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
Purchase
CHEMBL
PC cid
PC sid
Patents
In Depth
Details
US Patent
Copy BDB DOI
Target
Mitogen-activated protein kinase 14
(Homo sapiens (Human))
Everbrilliant Pharma
US Patent
Ligand
BDBM50295553
(4-(4-(4-fluorophenyl)-1-(3-phenylpropyl)-5-(pyridi...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 30nM
Assay Description:
FP signals were measured with a PHERAstar microplate reader (BMG Labtech) using black, low-binding half-area 96 well plates (Corning). Each binding d...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
Purchase
CHEMBL
PC cid
PC sid
Patents
In Depth
Details
US Patent
Copy BDB DOI
Target
Mitogen-activated protein kinase
(Toxoplasma gondii)
Tulane University School Of Medicine
Curated by
ChEMBL
Ligand
BDBM50295553
(4-(4-(4-fluorophenyl)-1-(3-phenylpropyl)-5-(pyridi...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 200nM
Assay Description:
Inhibition of Toxoplasma gondii recombinant MAPK1 expressed in Escherichia coli
More data for this Ligand-Target Pair
Target Info
UniProtKB/TrEMBL
GoogleScholar
Ligand Info
Purchase
CHEMBL
PC cid
PC sid
Patents
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Mitogen-activated protein kinase 14
(Homo sapiens (Human))
Everbrilliant Pharma
US Patent
Ligand
BDBM50295553
(4-(4-(4-fluorophenyl)-1-(3-phenylpropyl)-5-(pyridi...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 1.00E+3nM
Assay Description:
Inhibition of human recombinant p38alpha assessed as [gamma33P]ATP utilization by microplate scintillation counting
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
Purchase
CHEMBL
PC cid
PC sid
Patents
In Depth
Details
Article
PubMed
Copy BDB DOI