Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 4 hits in this display   

Target72 kDa type IV collagenase(Homo sapiens (Human))
Incyte

Curated by ChEMBL
LigandPNGBDBM50268953((1S,2S)-N-hydroxy-2-(4-phenylpiperazine-1-carbonyl...)
Affinity DataIC50:  180nMAssay Description:Inhibition of human MMP2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Incyte

Curated by ChEMBL
LigandPNGBDBM50268953((1S,2S)-N-hydroxy-2-(4-phenylpiperazine-1-carbonyl...)
Affinity DataIC50:  470nMAssay Description:Inhibition of HER2 extracellular domain sheddase activity in human BT474 cells after 72 hrs by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50268953((1S,2S)-N-hydroxy-2-(4-phenylpiperazine-1-carbonyl...)
Affinity DataIC50:  1.55E+3nMAssay Description:Inhibition of human recombinant ADAM10More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
Incyte

Curated by ChEMBL
LigandPNGBDBM50268953((1S,2S)-N-hydroxy-2-(4-phenylpiperazine-1-carbonyl...)
Affinity DataIC50: >5.00E+3nMAssay Description:Inhibition of human MMP1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed