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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 5 hits in this display   

TargetMatrix metalloproteinase-9(Homo sapiens (Human))
The Hebrew University Of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50146802(CHEMBL95068 | piperidin-1-ylcarbonylphosphonic aci...)
Affinity DataIC50:  500nMAssay Description:In vitro inhibitory activity against recombinant matrix metalloprotease-9 was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
The Hebrew University Of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50146802(CHEMBL95068 | piperidin-1-ylcarbonylphosphonic aci...)
Affinity DataIC50:  1.00E+3nMAssay Description:In vitro inhibitory activity against recombinant matrix metalloprotease-2 was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
The Hebrew University Of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50146802(CHEMBL95068 | piperidin-1-ylcarbonylphosphonic aci...)
Affinity DataIC50:  7.00E+4nMAssay Description:In vitro inhibitory activity against recombinant matrix metalloprotease-1 was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
The Hebrew University Of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50146802(CHEMBL95068 | piperidin-1-ylcarbonylphosphonic aci...)
Affinity DataIC50:  9.00E+4nMAssay Description:In vitro inhibitory activity against recombinant matrix metalloprotease-3 was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil collagenase(Homo sapiens (Human))
The Hebrew University Of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50146802(CHEMBL95068 | piperidin-1-ylcarbonylphosphonic aci...)
Affinity DataIC50: >1.00E+5nMAssay Description:In vitro inhibitory activity against recombinant matrix metalloprotease-8 was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed