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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

Target6,7-dimethyl-8-ribityllumazine synthase(Mycobacterium tuberculosis)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50316577(4-(2-Oxo-1,2-dihydrobenzo[cd]indole-6-sulfonamido)...)
Affinity DataKi:  1.10E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis recombinant lumazine synthase at enzyme-substrate complex state after 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target6,7-dimethyl-8-ribityllumazine synthase(Mycobacterium tuberculosis)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50316577(4-(2-Oxo-1,2-dihydrobenzo[cd]indole-6-sulfonamido)...)
Affinity DataKi:  3.80E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis recombinant lumazine synthase at enzyme-inhibitor complex state after 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target6,7-dimethyl-8-ribityllumazine synthase(Mycobacterium tuberculosis)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50316577(4-(2-Oxo-1,2-dihydrobenzo[cd]indole-6-sulfonamido)...)
Affinity DataKi:  5.72E+5nMAssay Description:Inhibition of Mycobacterium tuberculosis recombinant lumazine synthase at enzyme-substrate-inhibitor complex state after 30 mins by fluorescence assa...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed