Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 7 hits in this display   

TargetAdenosine receptor A1(BOVINE)
Universit£

Curated by ChEMBL
LigandPNGBDBM50090711(2-Phenyl-[1,8]naphthyridin-4-ol | 2-phenyl-1,8-nap...)
Affinity DataKi:  16nMAssay Description:Ability to displace the specific binding of [3H]CHA to adenosine A1 receptor from bovine brain cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Universit£

Curated by ChEMBL
LigandPNGBDBM50090711(2-Phenyl-[1,8]naphthyridin-4-ol | 2-phenyl-1,8-nap...)
Affinity DataKi:  16nMAssay Description:Binding affinity against adenosine A1 receptor in bovine cortical membranes using [3H]-CHA as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50090711(2-Phenyl-[1,8]naphthyridin-4-ol | 2-phenyl-1,8-nap...)
Affinity DataKi:  1.30E+3nMAssay Description:Binding affinity against adenosine A1 receptor in human cortical membranes using [3H]-CHA as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50090711(2-Phenyl-[1,8]naphthyridin-4-ol | 2-phenyl-1,8-nap...)
Affinity DataKi:  2.00E+3nMAssay Description:Binding affinity against adenosine A2 receptor in human striatal membranes using [3H]-CGS-21,680 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Rattus norvegicus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50090711(2-Phenyl-[1,8]naphthyridin-4-ol | 2-phenyl-1,8-nap...)
Affinity DataKi:  3.00E+3nMAssay Description:Ability to displace the specific binding of [3H](R)-PIA to adenosine A3 receptor from rat testis membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50090711(2-Phenyl-[1,8]naphthyridin-4-ol | 2-phenyl-1,8-nap...)
Affinity DataKi: >1.00E+4nMAssay Description:Ability to displace the specific binding of [3H]-CGS- to adenosine A2A receptor form bovine brain striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50090711(2-Phenyl-[1,8]naphthyridin-4-ol | 2-phenyl-1,8-nap...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity against adenosine A2 receptor in bovine striatal membranes using [3H]-CGS-21,680 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed