Compile Data Set for Download or QSAR
maximum 50k data

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetOxysterols receptor LXR-alpha(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50298696(CHEMBL574086 | N-{4-[2-(3,4-Dihydroxyphenyl)ethyl]...)
Affinity DataIC50:  1.70E+3nMAssay Description:Antagonist activity at human LXRalpha expressed in HEK293 cells assessed as inhibition of beta-galactosidase activity by luciferase reporter gene ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-beta(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50298696(CHEMBL574086 | N-{4-[2-(3,4-Dihydroxyphenyl)ethyl]...)
Affinity DataIC50: >3.00E+3nMAssay Description:Antagonist activity at human LXRbeta expressed in HEK293 cells assessed as inhibition of beta-galactosidase activity by luciferase reporter gene assa...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed