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Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
3
hits in this display
Target
High affinity nerve growth factor receptor
(Homo sapiens (Human))
Dongguk University
Curated by
ChEMBL
Ligand
BDBM67668
((6E)-6-[4-(4-hydroxyanilino)-1H-quinazolin-2-ylide...)
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Affinity Data
IC50: 303nM
Assay Description:
Inhibition of TrkA (unknown origin)
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
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CHEMBL
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In Depth
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Article
PubMed
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Target
ALK tyrosine kinase receptor
(Homo sapiens (Human))
Pharmadesign
Curated by
ChEMBL
Ligand
BDBM67668
((6E)-6-[4-(4-hydroxyanilino)-1H-quinazolin-2-ylide...)
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Affinity Data
IC50: 4.24E+3nM
Assay Description:
Inhibition of ALK using FL-Peptide 13, 5-FAM-KKSRGDYMTMQIG-CONH2 substrate after 60 mins by mobility shift assay
More data for this Ligand-Target Pair
Target Info
PDB
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
Purchase
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
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Target
Serine/threonine-protein kinase 33
(Homo sapiens (Human))
Broad Institute
Curated by
PubChem BioAssay
Ligand
BDBM67668
((6E)-6-[4-(4-hydroxyanilino)-1H-quinazolin-2-ylide...)
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Affinity Data
EC50: 2.43E+3nM
Assay Description:
Keywords: STK33 Kinase, Non-ATP Competitive Inhibitor Assay Overview: Purified STK33 Kinase is preincubated with potential inhibitors and allowed to ...
More data for this Ligand-Target Pair
Target Info
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
Purchase
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
PCBioAssay
Copy BDB DOI