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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
8
hits in this display
Target
Mu-type opioid receptor
(Rattus norvegicus (rat))
University Of Innsbruck And Center For Molecular Biosciences Innsbruck-Cmbi
Curated by
ChEMBL
Ligand
BDBM50326661
(CHEMBL1254018 | CHEMBL1254291)
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Affinity Data
Ki: 0.460nM
Assay Description:
Displacement of [3H]DAMGO from mu opioid receptor in rat brain membrane
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
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Target
Delta-type opioid receptor
(Rattus norvegicus (rat))
University Of Innsbruck And Center For Molecular Biosciences Innsbruck-Cmbi
Curated by
ChEMBL
Ligand
BDBM50326661
(CHEMBL1254018 | CHEMBL1254291)
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Copy InChI
Affinity Data
Ki: 12.2nM
Assay Description:
Displacement of [3H][Ile5,6]deltorphin2 from delta opioid receptor in rat brain membrane
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
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Target
Kappa-type opioid receptor
(Cavia porcellus (domestic guinea pig))
University Of Innsbruck And Center For Molecular Biosciences Innsbruck-Cmbi
Curated by
ChEMBL
Ligand
BDBM50326661
(CHEMBL1254018 | CHEMBL1254291)
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Affinity Data
Ki: 43.2nM
Assay Description:
Displacement of [3H]U69593 from kappa opioid receptor in guinea pig brain membrane
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Mu-type opioid receptor
(Rattus norvegicus (rat))
University Of Innsbruck And Center For Molecular Biosciences Innsbruck-Cmbi
Curated by
ChEMBL
Ligand
BDBM50326661
(CHEMBL1254018 | CHEMBL1254291)
Copy SMILES
Copy InChI
Affinity Data
Ki: 67.2nM
Assay Description:
Displacement of [3H]DAMGO from mu opioid receptor in rat brain membrane
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Kappa-type opioid receptor
(Cavia porcellus (domestic guinea pig))
University Of Innsbruck And Center For Molecular Biosciences Innsbruck-Cmbi
Curated by
ChEMBL
Ligand
BDBM50326661
(CHEMBL1254018 | CHEMBL1254291)
Copy SMILES
Copy InChI
Affinity Data
Ki: 328nM
Assay Description:
Displacement of [3H]U69593 from kappa opioid receptor in guinea pig brain membrane
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Delta-type opioid receptor
(Rattus norvegicus (rat))
University Of Innsbruck And Center For Molecular Biosciences Innsbruck-Cmbi
Curated by
ChEMBL
Ligand
BDBM50326661
(CHEMBL1254018 | CHEMBL1254291)
Copy SMILES
Copy InChI
Affinity Data
Ki: 1.25E+3nM
Assay Description:
Displacement of [3H][Ile5,6]deltorphin2 from delta opioid receptor in rat brain membrane
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Acetylcholinesterase
(Electrophorus electricus (Electric eel))
University Of Innsbruck And Center For Molecular Biosciences Innsbruck-Cmbi
Curated by
ChEMBL
Ligand
BDBM50326661
(CHEMBL1254018 | CHEMBL1254291)
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Affinity Data
IC50: 1.27E+4nM
Assay Description:
Inhibition of electric eel AChE by Ellman's method
More data for this Ligand-Target Pair
Target Info
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Acetylcholinesterase
(Electrophorus electricus (Electric eel))
University Of Innsbruck And Center For Molecular Biosciences Innsbruck-Cmbi
Curated by
ChEMBL
Ligand
BDBM50326661
(CHEMBL1254018 | CHEMBL1254291)
Copy SMILES
Copy InChI
Affinity Data
IC50: 1.05E+5nM
Assay Description:
Inhibition of electric eel AChE by Ellman's method
More data for this Ligand-Target Pair
Target Info
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI