Compile Data Set for Download or QSAR
maximum 50k data

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 8 hits in this display   

TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Innsbruck And Center For Molecular Biosciences Innsbruck-Cmbi

Curated by ChEMBL
LigandPNGBDBM50326661(CHEMBL1254018 | CHEMBL1254291)
Affinity DataKi:  0.460nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
University Of Innsbruck And Center For Molecular Biosciences Innsbruck-Cmbi

Curated by ChEMBL
LigandPNGBDBM50326661(CHEMBL1254018 | CHEMBL1254291)
Affinity DataKi:  12.2nMAssay Description:Displacement of [3H][Ile5,6]deltorphin2 from delta opioid receptor in rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Innsbruck And Center For Molecular Biosciences Innsbruck-Cmbi

Curated by ChEMBL
LigandPNGBDBM50326661(CHEMBL1254018 | CHEMBL1254291)
Affinity DataKi:  43.2nMAssay Description:Displacement of [3H]U69593 from kappa opioid receptor in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Innsbruck And Center For Molecular Biosciences Innsbruck-Cmbi

Curated by ChEMBL
LigandPNGBDBM50326661(CHEMBL1254018 | CHEMBL1254291)
Affinity DataKi:  67.2nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Innsbruck And Center For Molecular Biosciences Innsbruck-Cmbi

Curated by ChEMBL
LigandPNGBDBM50326661(CHEMBL1254018 | CHEMBL1254291)
Affinity DataKi:  328nMAssay Description:Displacement of [3H]U69593 from kappa opioid receptor in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
University Of Innsbruck And Center For Molecular Biosciences Innsbruck-Cmbi

Curated by ChEMBL
LigandPNGBDBM50326661(CHEMBL1254018 | CHEMBL1254291)
Affinity DataKi:  1.25E+3nMAssay Description:Displacement of [3H][Ile5,6]deltorphin2 from delta opioid receptor in rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Innsbruck And Center For Molecular Biosciences Innsbruck-Cmbi

Curated by ChEMBL
LigandPNGBDBM50326661(CHEMBL1254018 | CHEMBL1254291)
Affinity DataIC50:  1.27E+4nMAssay Description:Inhibition of electric eel AChE by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Innsbruck And Center For Molecular Biosciences Innsbruck-Cmbi

Curated by ChEMBL
LigandPNGBDBM50326661(CHEMBL1254018 | CHEMBL1254291)
Affinity DataIC50:  1.05E+5nMAssay Description:Inhibition of electric eel AChE by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed