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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
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Found
2
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Target
Fatty-acid amide hydrolase 1 [30-579]
(Rattus norvegicus (rat))
Sapienza University Of Rome
Ligand
BDBM23018
(3-(trifluoromethyl)phenyl N-[2-(5-hydroxy-1H-indol...)
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Affinity Data
IC50: 2.20E+3nM
Assay Description:
The effect of the test compounds on the enzymatic hydrolysis of [14C]anandamide was evaluated by using membranes prepared from rat brain. [14C]Ethano...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
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Target
Transient receptor potential cation channel subfamily V member 1
(Homo sapiens (Human))
Sapienza University Of Rome
Ligand
BDBM23018
(3-(trifluoromethyl)phenyl N-[2-(5-hydroxy-1H-indol...)
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Affinity Data
IC50: >1.00E+4nM
T: 2°C
Assay Description:
The antagonistic effects of test compounds were evaluated using HEK293 cells stably overexpressing human TRPV1. Experiments were carried out by measu...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI