Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 9 hits in this display   

TargetKappa-type opioid receptor(Mus musculus (Mouse))
Memorial Sloan-Kettering Cancer Center

Curated by ChEMBL
LigandPNGBDBM50346952(CHEMBL1795712 | CHEMBL1795715)
Affinity DataKi:  0.0800nMAssay Description:Displacement of [125I]-BNtxA from mouse cloned KOR-1 expressed in CHO cell membrane after 90 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Memorial Sloan-Kettering Cancer Center

Curated by ChEMBL
LigandPNGBDBM50346952(CHEMBL1795712 | CHEMBL1795715)
Affinity DataKi:  0.0800nMAssay Description:Displacement of [3H]-U69593 from KOR-1 expressed in CHO cells after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Memorial Sloan-Kettering Cancer Center

Curated by ChEMBL
LigandPNGBDBM50346952(CHEMBL1795712 | CHEMBL1795715)
Affinity DataKi:  0.220nMAssay Description:Displacement of [125I]-BNtxA from mouse cloned MOR-1 expressed in CHO cell membrane after 90 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Memorial Sloan-Kettering Cancer Center

Curated by ChEMBL
LigandPNGBDBM50346952(CHEMBL1795712 | CHEMBL1795715)
Affinity DataKi:  0.700nMAssay Description:Displacement of [3H]-DAMGO from MOR-1 expressed in CHO cells after 150 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Memorial Sloan-Kettering Cancer Center

Curated by ChEMBL
LigandPNGBDBM50346952(CHEMBL1795712 | CHEMBL1795715)
Affinity DataKi:  2.55nMAssay Description:Displacement of [125I]-BNtxA from mouse cloned DOR-1 expressed in CHO cell membrane after 90 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Memorial Sloan-Kettering Cancer Center

Curated by ChEMBL
LigandPNGBDBM50346952(CHEMBL1795712 | CHEMBL1795715)
Affinity DataKi:  2.60nMAssay Description:Displacement of [3H]-DPDPE from DOR-1 expressed in CHO cells after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Memorial Sloan-Kettering Cancer Center

Curated by ChEMBL
LigandPNGBDBM50346952(CHEMBL1795712 | CHEMBL1795715)
Affinity DataKd:  0.0500nMAssay Description:Binding affinity to KOR-1 expressed in CHO cells after 90 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Memorial Sloan-Kettering Cancer Center

Curated by ChEMBL
LigandPNGBDBM50346952(CHEMBL1795712 | CHEMBL1795715)
Affinity DataKd:  2.5nMAssay Description:Binding affinity to DOR-1 expressed in CHO cells after 90 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Memorial Sloan-Kettering Cancer Center

Curated by ChEMBL
LigandPNGBDBM50346952(CHEMBL1795712 | CHEMBL1795715)
Affinity DataKd:  0.220nMAssay Description:Binding affinity to MOR-1 expressed in CHO cells after 90 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed