Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 9 hits in this display
BDBM50065854(22-cyclopropylmethyl-9-phenoxy-14-oxa-11,22-diazah...)
Ki: 0.610nMAssay Description:Displacement of [3H]DADLE from morphine-insensitive Opioid receptor delta 1 (presence of 50 nM morphine) of rat brain membranesMore data for this Ligand-Target Pair
BDBM50065854(22-cyclopropylmethyl-9-phenoxy-14-oxa-11,22-diazah...)
BDBM50065854(22-cyclopropylmethyl-9-phenoxy-14-oxa-11,22-diazah...)
Ki: 19nMAssay Description:Displacement of [3H]DADLE from morphine-sensitive Opioid receptor delta 1 (presence of 300 nM DELT-II) of rat brain membranesMore data for this Ligand-Target Pair
Mu-type opioid receptor(Rattus norvegicus (rat))University Of Medicine & Dentistry Of New Jersey-Robert Wood Johnson Medical School (Umdnj-Rwjms)
Curated by ChEMBL
Kappa-type opioid receptor(Cavia porcellus (domestic guinea pig))University Of Medicine & Dentistry Of New Jersey-Robert Wood Johnson Medical School (Umdnj-Rwjms)
Curated by ChEMBL
Mu-type opioid receptor(Rattus norvegicus (rat))University Of Medicine & Dentistry Of New Jersey-Robert Wood Johnson Medical School (Umdnj-Rwjms)
Curated by ChEMBL
BDBM50065854(22-cyclopropylmethyl-9-phenoxy-14-oxa-11,22-diazah...)
Kappa-type opioid receptor(Cavia porcellus (domestic guinea pig))University Of Medicine & Dentistry Of New Jersey-Robert Wood Johnson Medical School (Umdnj-Rwjms)
Curated by ChEMBL
BDBM50065854(22-cyclopropylmethyl-9-phenoxy-14-oxa-11,22-diazah...)
Ki: 34nMAssay Description:Displacement of [3H]U-69593 from Opioid receptor kappa 1 of guinea pig brain membranes (pretreated with BIT and FIT to block mu and delta sites)More data for this Ligand-Target Pair
Kappa-type opioid receptor(Cavia porcellus (domestic guinea pig))University Of Medicine & Dentistry Of New Jersey-Robert Wood Johnson Medical School (Umdnj-Rwjms)
Curated by ChEMBL
BDBM50065854(22-cyclopropylmethyl-9-phenoxy-14-oxa-11,22-diazah...)