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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 8 hits in this display   

TargetDelta-type opioid receptor(Rattus norvegicus (rat))
National Institute Of Diabetes

Curated by ChEMBL
LigandPNGBDBM50056629(4-cyclopropylmethyl-10,17-dihydroxy-15-[1-(4-pheny...)
Affinity DataKi:  47nMAssay Description:Binding affinity evaluated by inhibition of binding of [3H]DADLE to delta opioid receptor of rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Washington

Curated by ChEMBL
LigandPNGBDBM50056629(4-cyclopropylmethyl-10,17-dihydroxy-15-[1-(4-pheny...)
Affinity DataKi:  47nMAssay Description:Binding affinity was determined in a crude membrane preparation from guinea pig brain by displacement of [3H]DPDPE from Opioid receptor delta 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University Of Washington

Curated by ChEMBL
LigandPNGBDBM50056629(4-cyclopropylmethyl-10,17-dihydroxy-15-[1-(4-pheny...)
Affinity DataKi:  50nMAssay Description:Binding affinity was determined in a crude membrane preparation from guinea pig brain by displacement of [3H]DAMGO from Opioid receptor mu 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Washington

Curated by ChEMBL
LigandPNGBDBM50056629(4-cyclopropylmethyl-10,17-dihydroxy-15-[1-(4-pheny...)
Affinity DataKi:  75nMAssay Description:Binding affinity was determined in a crude membrane preparation from guinea pig brain by displacement of [3H]DPDPE from Opioid receptor delta 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
National Institute Of Diabetes

Curated by ChEMBL
LigandPNGBDBM50056629(4-cyclopropylmethyl-10,17-dihydroxy-15-[1-(4-pheny...)
Affinity DataKi:  75nMAssay Description:Binding affinity evaluated by inhibition of binding of [3H]DADLE to delta opioid receptor of rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Washington

Curated by ChEMBL
LigandPNGBDBM50056629(4-cyclopropylmethyl-10,17-dihydroxy-15-[1-(4-pheny...)
Affinity DataKi:  190nMAssay Description:Binding affinity was determined in a crude membrane preparation from guinea pig brain by displacement of [3H]U-69593 from Opioid receptor kappa 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University Of Washington

Curated by ChEMBL
LigandPNGBDBM50056629(4-cyclopropylmethyl-10,17-dihydroxy-15-[1-(4-pheny...)
Affinity DataKi:  210nMAssay Description:Binding affinity was determined in a crude membrane preparation from guinea pig brain by displacement of [3H]DAMGO from Opioid receptor mu 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Washington

Curated by ChEMBL
LigandPNGBDBM50056629(4-cyclopropylmethyl-10,17-dihydroxy-15-[1-(4-pheny...)
Affinity DataKi:  400nMAssay Description:Binding affinity was determined in a crude membrane preparation from guinea pig brain by displacement of [3H]U-69593 from Opioid receptor kappa 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed