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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
8
hits in this display
Target
Delta-type opioid receptor
(Rattus norvegicus (rat))
National Institute Of Diabetes
Curated by
ChEMBL
Ligand
BDBM50056629
(4-cyclopropylmethyl-10,17-dihydroxy-15-[1-(4-pheny...)
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Affinity Data
Ki: 47nM
Assay Description:
Binding affinity evaluated by inhibition of binding of [3H]DADLE to delta opioid receptor of rat brain
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Delta-type opioid receptor
(Homo sapiens (Human))
University Of Washington
Curated by
ChEMBL
Ligand
BDBM50056629
(4-cyclopropylmethyl-10,17-dihydroxy-15-[1-(4-pheny...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 47nM
Assay Description:
Binding affinity was determined in a crude membrane preparation from guinea pig brain by displacement of [3H]DPDPE from Opioid receptor delta 1
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Mu-type opioid receptor
(GUINEA PIG)
University Of Washington
Curated by
ChEMBL
Ligand
BDBM50056629
(4-cyclopropylmethyl-10,17-dihydroxy-15-[1-(4-pheny...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 50nM
Assay Description:
Binding affinity was determined in a crude membrane preparation from guinea pig brain by displacement of [3H]DAMGO from Opioid receptor mu 1
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Delta-type opioid receptor
(Homo sapiens (Human))
University Of Washington
Curated by
ChEMBL
Ligand
BDBM50056629
(4-cyclopropylmethyl-10,17-dihydroxy-15-[1-(4-pheny...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 75nM
Assay Description:
Binding affinity was determined in a crude membrane preparation from guinea pig brain by displacement of [3H]DPDPE from Opioid receptor delta 1
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Delta-type opioid receptor
(Rattus norvegicus (rat))
National Institute Of Diabetes
Curated by
ChEMBL
Ligand
BDBM50056629
(4-cyclopropylmethyl-10,17-dihydroxy-15-[1-(4-pheny...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 75nM
Assay Description:
Binding affinity evaluated by inhibition of binding of [3H]DADLE to delta opioid receptor of rat brain
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Kappa-type opioid receptor
(Cavia porcellus (domestic guinea pig))
University Of Washington
Curated by
ChEMBL
Ligand
BDBM50056629
(4-cyclopropylmethyl-10,17-dihydroxy-15-[1-(4-pheny...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 190nM
Assay Description:
Binding affinity was determined in a crude membrane preparation from guinea pig brain by displacement of [3H]U-69593 from Opioid receptor kappa 1
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Mu-type opioid receptor
(GUINEA PIG)
University Of Washington
Curated by
ChEMBL
Ligand
BDBM50056629
(4-cyclopropylmethyl-10,17-dihydroxy-15-[1-(4-pheny...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 210nM
Assay Description:
Binding affinity was determined in a crude membrane preparation from guinea pig brain by displacement of [3H]DAMGO from Opioid receptor mu 1
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Kappa-type opioid receptor
(Cavia porcellus (domestic guinea pig))
University Of Washington
Curated by
ChEMBL
Ligand
BDBM50056629
(4-cyclopropylmethyl-10,17-dihydroxy-15-[1-(4-pheny...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 400nM
Assay Description:
Binding affinity was determined in a crude membrane preparation from guinea pig brain by displacement of [3H]U-69593 from Opioid receptor kappa 1
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI