Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 4 hits in this display   

TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
University Of Regensburg

Curated by ChEMBL
LigandPNGBDBM50090282(2-Biphenyl-4-yl-N-{1-(7-hydroxy-1,3,4,5-tetrahydro...)
Affinity DataIC50:  770nMAssay Description:Inhibition of binding of [3H]-propionyl-NPY (1 nM) to Neuropeptide Y receptor type 5 in HEC-1-B cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
University Of Regensburg

Curated by ChEMBL
LigandPNGBDBM50090282(2-Biphenyl-4-yl-N-{1-(7-hydroxy-1,3,4,5-tetrahydro...)
Affinity DataIC50:  1.19E+4nMAssay Description:NPY Y1-antagonistic activity in HEL cells by measuring the inhibition of porcine NPY (10 nM) stimulated increase in the intracellular [Ca2+] concentr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
University Of Regensburg

Curated by ChEMBL
LigandPNGBDBM50090282(2-Biphenyl-4-yl-N-{1-(7-hydroxy-1,3,4,5-tetrahydro...)
Affinity DataIC50:  2.20E+4nMAssay Description:Inhibition of binding of [3H]-propionyl-NPY (1 nM) to Neuropeptide Y receptor type 1 in SK-N-MC cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 2(Homo sapiens (Human))
University Of Regensburg

Curated by ChEMBL
LigandPNGBDBM50090282(2-Biphenyl-4-yl-N-{1-(7-hydroxy-1,3,4,5-tetrahydro...)
Affinity DataIC50:  7.80E+4nMAssay Description:Inhibition of binding of [3H]-propionyl-NPY (1 nM) to Neuropeptide Y receptor type 2 in SMS-KAN cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed