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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 1 hits in this display   

TargetAromatase(Homo sapiens (Human))
Cardiff University

LigandPNGBDBM10014(2-[(4-Nitrophenyl)-[1,2,4]triazol-1-ylmethyl]benzo...)
Affinity DataIC50:  60nMpH: 7.4 T: 2°CAssay Description:The enzyme activity was assayed by measuring the 3H-labeled H2O formed from [1,2,6,7-3H ]androstenedione / androstenedione during aromatization. Afte...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed