Home
About
Info
Download
WebServices
Contact
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
4
hits in this display
Target
Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Nanyang Normal University
Curated by
ChEMBL
Ligand
BDBM178001
((E)-1-(2-hydroxyphenyl)-3-(3-hydroxyphenyl)prop-2-...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 1.10E+3nM
Assay Description:
Inhibition of recombinant human MAO-B expressed in baculovirus infected BTI insect cells using kynuramine as substrate measured after 30 mins by fluo...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
Purchase
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Oligo-1,6-glucosidase IMA1
(Saccharomyces cerevisiae S288c (Baker's yeast))
Universiti Teknologi Mara
Ligand
BDBM178001
((E)-1-(2-hydroxyphenyl)-3-(3-hydroxyphenyl)prop-2-...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 4.47E+4nM
pH: 6.8
Assay Description:
The α-glucosidase inhibition assay had been carried out using baker¿s yeast a-glucosidase (EC 3.2.1.20) and p-nitrophenyl-α-D-glucopyranosi...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
Purchase
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Biofilm regulatory protein A
(Streptococcus mutans serotype c (strain ATCC 70061...)
Uab Research Foundation
US Patent
Ligand
BDBM178001
((E)-1-(2-hydroxyphenyl)-3-(3-hydroxyphenyl)prop-2-...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 6.40E+4nM
Assay Description:
A previously reported zymographic assay was utilized for the investigation of Gtf enzymatic activity, as described in Example 1. A 1:100 in fresh 5 m...
More data for this Ligand-Target Pair
Target Info
UniProtKB/SwissProt
GoogleScholar
Ligand Info
Purchase
PC cid
PC sid
Similars
In Depth
Details
US Patent
Copy BDB DOI
Target
Xanthine dehydrogenase/oxidase
(Bos taurus (Bovine))
Guangxi Medical University
Curated by
ChEMBL
Ligand
BDBM178001
((E)-1-(2-hydroxyphenyl)-3-(3-hydroxyphenyl)prop-2-...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 9.18E+4nM
Assay Description:
Inhibition of bovine milk xanthine oxidase pre-incubated for 30 mins followed by xanthine addition and measured every 30 secs for 5 mins by spectroph...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
KEGG
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
Purchase
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI