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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

TargetStromelysin-1(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50278812(5-Hydroxy-4-thioxo-4H-pyran-2-carboxylic acid (bip...)
Affinity DataIC50:  1.33E+4nMAssay Description:Inhibition of human MMP3 catalytic domain by fluorescent substrate assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50278812(5-Hydroxy-4-thioxo-4H-pyran-2-carboxylic acid (bip...)
Affinity DataIC50:  1.44E+4nMAssay Description:Inhibition of human MMP2 catalytic domain by fluorescent substrate assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50278812(5-Hydroxy-4-thioxo-4H-pyran-2-carboxylic acid (bip...)
Affinity DataIC50:  4.40E+4nMAssay Description:Inhibition of human MMP1 catalytic domain by fluorescent substrate assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed