Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 4 hits in this display   

TargetInterstitial collagenase(Homo sapiens (Human))
Affymax Research Institute

Curated by ChEMBL
LigandPNGBDBM50064791((3R,6R)-1,6-Bis-cyclohexylmethyl-3-mercaptomethyl-...)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibition of collagenase-1 (Matrix metalloproteinase-1)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrilysin(Homo sapiens (Human))
Affymax Research Institute

Curated by ChEMBL
LigandPNGBDBM50064791((3R,6R)-1,6-Bis-cyclohexylmethyl-3-mercaptomethyl-...)
Affinity DataIC50:  4.80E+3nMAssay Description:Inhibition of matrilysin (Matrix metalloproteinase-7)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
Affymax Research Institute

Curated by ChEMBL
LigandPNGBDBM50064791((3R,6R)-1,6-Bis-cyclohexylmethyl-3-mercaptomethyl-...)
Affinity DataIC50:  1.20E+4nMAssay Description:Inhibition of gelatinase-B (Matrix metalloproteinase-9)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Affymax Research Institute

Curated by ChEMBL
LigandPNGBDBM50064791((3R,6R)-1,6-Bis-cyclohexylmethyl-3-mercaptomethyl-...)
Affinity DataIC50: >4.00E+4nMAssay Description:Inhibition of stromelysin-1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed