Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 12 hits in this display
BDBM224012(Capzimin | US10005735, Compound 12)
BDBM224012(Capzimin | US10005735, Compound 12)
BDBM224012(Capzimin | US10005735, Compound 12)
BDBM224012(Capzimin | US10005735, Compound 12)
BDBM224012(Capzimin | US10005735, Compound 12)
IC50: 4.50E+3nMAssay Description:In brief, this Rpn11 bioassay employs a fluorescent polarization readout based on the ability of the 26S proteasome to cleave the protein substrate i...More data for this Ligand-Target Pair
BDBM224012(Capzimin | US10005735, Compound 12)
IC50: 3.00E+4nMAssay Description:In brief, this Rpn11 bioassay employs a fluorescent polarization readout based on the ability of the 26S proteasome to cleave the protein substrate i...More data for this Ligand-Target Pair
BDBM224012(Capzimin | US10005735, Compound 12)
BDBM224012(Capzimin | US10005735, Compound 12)
BDBM224012(Capzimin | US10005735, Compound 12)
BDBM224012(Capzimin | US10005735, Compound 12)
BDBM224012(Capzimin | US10005735, Compound 12)
IC50: >5.00E+4nMpH: 7.5 T: 2°CAssay Description:The assay was carried out in white NUNC 96-well plates as previously described [Puerta et al., J. Biol. Inorg. Chem., 11:131-138]. Each well containe...More data for this Ligand-Target Pair
BDBM224012(Capzimin | US10005735, Compound 12)