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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Elan Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50345603(4-(5-(naphthalen-2-yl)-1H-tetrazol-1-yl)pyridine |...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of JNK1 by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 9(Homo sapiens (Human))
Elan Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50345603(4-(5-(naphthalen-2-yl)-1H-tetrazol-1-yl)pyridine |...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of JNK2 by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
Elan Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50345603(4-(5-(naphthalen-2-yl)-1H-tetrazol-1-yl)pyridine |...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of JNK3 by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed