Affinity DataIC50: 2.21E+4nMAssay Description:Antagonist activity at human recombinant GABAc rho-2 receptor expressed in Xenopus laevis oocytes assessed as inhibition of GABA-induced current by t...More data for this Ligand-Target Pair
Affinity DataIC50: 5.13E+4nMAssay Description:Antagonist activity at human recombinant GABAc rho-2 receptor expressed in Xenopus laevis oocytes assessed as inhibition of GABA-induced current by t...More data for this Ligand-Target Pair
Affinity DataIC50: 5.71E+4nMAssay Description:Antagonist activity at human recombinant GABAc rho-2 receptor expressed in Xenopus laevis oocytes assessed as inhibition of GABA-induced current by t...More data for this Ligand-Target Pair
Affinity DataKd: 1.40E+3nMAssay Description:Partial agonist activity against human rho-2 subunit GABA-C receptor expressed in Xenopus oocytesMore data for this Ligand-Target Pair
Affinity DataEC50: 7.00E+4nMAssay Description:Partial agonist activity againast human rho-2 subunit GABA-C receptor expressed in Xenopus oocytesMore data for this Ligand-Target Pair
Affinity DataEC50: 400nMAssay Description:Partial agonist activity against homomeric rho-2 subunit GABA-C receptor expressed in Xenopus oocytesMore data for this Ligand-Target Pair
Affinity DataEC50: 1.01E+5nMAssay Description:Activation of human rho2 GABA-C receptor at 34% of maximal GABA-induced responseMore data for this Ligand-Target Pair
Affinity DataEC50: 3.00E+3nMAssay Description:Partial agonist activity against human rho-2 subunit GABA-C receptor expressed in Xenopus oocytesMore data for this Ligand-Target Pair
Affinity DataEC50: 1.75E+4nMAssay Description:Partial agonist activity with low efficacy against rho-2 subunit GABA-C receptor expressed in Xenopus oocytesMore data for this Ligand-Target Pair
Affinity DataEC50: 3.45E+4nMAssay Description:Full agonist activity against human rho-2 subunit GABA-C receptor expressed in Xenopus oocytesMore data for this Ligand-Target Pair