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Found 27 Enz. Inhib. hit(s) with Target = 'HLA class II histocompatibility antigen, DR beta 3 chain'
TargetHLA class II histocompatibility antigen, DR beta 3 chain(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287637((S)-3-{(S)-2-[(S)-2-((S)-2-Acetylamino-3-naphthale...)
Affinity DataIC50:  31nMAssay Description:Ability to compete for binding to Class II MHC using ELISA assay.More data for this Ligand-Target Pair
In DepthDetails Article
TargetHLA class II histocompatibility antigen, DR beta 3 chain(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50366440(CHEMBL1790415 | SC-67655)
Affinity DataIC50:  50nMAssay Description:Ability to compete for binding to Class II MHC using ELISA assay.More data for this Ligand-Target Pair
In DepthDetails Article
TargetHLA class II histocompatibility antigen, DR beta 3 chain(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287642((S)-3-({1-[(S)-6-Amino-2-(3-bicyclo[2.2.1]hept-2-y...)
Affinity DataIC50:  76nMAssay Description:Ability to compete for binding to Class II MHC using ELISA assay.More data for this Ligand-Target Pair
In DepthDetails Article
TargetHLA class II histocompatibility antigen, DR beta 3 chain(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50366444(CHEMBL1790402)
Affinity DataIC50:  100nMAssay Description:Ability to compete for binding to Class II MHC using ELISA assay.More data for this Ligand-Target Pair
In DepthDetails Article
TargetHLA class II histocompatibility antigen, DR beta 3 chain(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287650((S)-3-({1-[2-Cyclohexyl-2-((R)-3-cyclohexyl-butyry...)
Affinity DataIC50:  130nMAssay Description:Ability to compete for binding to Class II MHC using ELISA assay.More data for this Ligand-Target Pair
In DepthDetails Article
TargetHLA class II histocompatibility antigen, DR beta 3 chain(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287636((S)-3-({1-[(S)-6-Amino-2-((S)-3-cyclohexyl-butyryl...)
Affinity DataIC50:  162nMAssay Description:Ability to compete for binding to Class II MHC using ELISA assay.More data for this Ligand-Target Pair
In DepthDetails Article
TargetHLA class II histocompatibility antigen, DR beta 3 chain(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287628((S)-3-({1-[(S)-2-(3-Cyclohexyl-propionylamino)-3-m...)
Affinity DataIC50:  170nMAssay Description:Ability to compete for binding to Class II MHC using ELISA assay.More data for this Ligand-Target Pair
In DepthDetails Article
TargetHLA class II histocompatibility antigen, DR beta 3 chain(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50366439(CHEMBL1793835)
Affinity DataIC50:  178nMAssay Description:Ability to compete for binding to Class II MHC using ELISA assay.More data for this Ligand-Target Pair
In DepthDetails Article
TargetHLA class II histocompatibility antigen, DR beta 3 chain(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287630((S)-3-({1-[(S)-6-Amino-2-(3-cycloheptyl-propionyla...)
Affinity DataIC50:  178nMAssay Description:Ability to compete for binding to Class II MHC using ELISA assay.More data for this Ligand-Target Pair
In DepthDetails Article
TargetHLA class II histocompatibility antigen, DR beta 3 chain(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50366439(CHEMBL1793835)
Affinity DataIC50:  178nMAssay Description:Ability to compete for binding to Class II MHC using ELISA assay.More data for this Ligand-Target Pair
In DepthDetails Article
TargetHLA class II histocompatibility antigen, DR beta 3 chain(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287626((S)-2-((2S,3R)-2-{(S)-2-[(S)-2-((S)-2-{(S)-2-[(S)-...)
Affinity DataIC50:  180nMAssay Description:Ability to compete for binding to Class II MHC using ELISA assay.More data for this Ligand-Target Pair
In DepthDetails Article
TargetHLA class II histocompatibility antigen, DR beta 3 chain(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287640(1-[(S)-2-((R)-3-Cyclohexyl-butyrylamino)-3-methyl-...)
Affinity DataIC50:  293nMAssay Description:Ability to compete for binding to Class II MHC using ELISA assay.More data for this Ligand-Target Pair
In DepthDetails Article
TargetHLA class II histocompatibility antigen, DR beta 3 chain(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287649((S)-3-({1-[2-((R)-3-Cyclohexyl-butyrylamino)-2-phe...)
Affinity DataIC50:  424nMAssay Description:Ability to compete for binding to Class II MHC using ELISA assay.More data for this Ligand-Target Pair
In DepthDetails Article
TargetHLA class II histocompatibility antigen, DR beta 3 chain(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287646((S)-3-({1-[(2S,3R)-2-((R)-3-Cyclohexyl-butyrylamin...)
Affinity DataIC50:  1.30E+3nMAssay Description:Ability to compete for binding to Class II MHC using ELISA assay.More data for this Ligand-Target Pair
In DepthDetails Article
TargetHLA class II histocompatibility antigen, DR beta 3 chain(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50366443(CHEMBL1790407)
Affinity DataIC50:  1.80E+3nMAssay Description:Ability to compete for binding to Class II MHC using ELISA assay.More data for this Ligand-Target Pair
In DepthDetails Article
TargetHLA class II histocompatibility antigen, DR beta 3 chain(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50366441(CHEMBL1790416)
Affinity DataIC50:  2.50E+3nMAssay Description:Ability to compete for binding to Class II MHC using ELISA assay.More data for this Ligand-Target Pair
In DepthDetails Article
TargetHLA class II histocompatibility antigen, DR beta 3 chain(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287643((S)-3-({1-[(S)-2-(3-Cyclohexyl-propionylamino)-3-(...)
Affinity DataIC50:  3.15E+3nMAssay Description:Ability to compete for binding to Class II MHC using ELISA assay.More data for this Ligand-Target Pair
In DepthDetails Article
TargetHLA class II histocompatibility antigen, DR beta 3 chain(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287652(3-({(S)-1-[2-(3-Cyclohexyl-butyrylamino)-3-methyl-...)
Affinity DataIC50:  7.00E+3nMAssay Description:Ability to compete for binding to Class II MHC using ELISA assay.More data for this Ligand-Target Pair
In DepthDetails Article
TargetHLA class II histocompatibility antigen, DR beta 3 chain(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287633(3-({(S)-(S)-1-[2-((S)-3-Cyclohexyl-butyrylamino)-6...)
Affinity DataIC50:  1.00E+4nMAssay Description:Ability to compete for binding to Class II MHC using ELISA assay.More data for this Ligand-Target Pair
In DepthDetails Article
TargetHLA class II histocompatibility antigen, DR beta 3 chain(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50366442(CHEMBL1790414)
Affinity DataIC50:  1.60E+4nMAssay Description:Ability to compete for binding to Class II MHC using ELISA assay.More data for this Ligand-Target Pair
In DepthDetails Article
TargetHLA class II histocompatibility antigen, DR beta 3 chain(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287654((S)-4-((S)-2-Carbamoyl-pyrrolidin-1-yl)-3-({1-[(S)...)
Affinity DataIC50:  2.33E+4nMAssay Description:Ability to compete for binding to Class II MHC using ELISA assay.More data for this Ligand-Target Pair
In DepthDetails Article
TargetHLA class II histocompatibility antigen, DR beta 3 chain(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287653(1-[(S)-2-((R)-3-Cyclohexyl-butyrylamino)-3-methyl-...)
Affinity DataIC50:  4.37E+4nMAssay Description:Ability to compete for binding to Class II MHC using ELISA assay.More data for this Ligand-Target Pair
In DepthDetails Article
TargetHLA class II histocompatibility antigen, DR beta 3 chain(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287631(3-({1-[(S)-2-((R)-3-Cyclohexyl-butyrylamino)-3-met...)
Affinity DataIC50: >1.00E+5nMAssay Description:Ability to compete for binding to Class II MHC using ELISA assay.More data for this Ligand-Target Pair
In DepthDetails Article
TargetHLA class II histocompatibility antigen, DR beta 3 chain(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287629((S)-4-[(S)-2-((S)-2-Amino-1-propylcarbamoyl-ethylc...)
Affinity DataIC50: >1.00E+5nMAssay Description:Ability to compete for binding to Class II MHC using ELISA assay.More data for this Ligand-Target Pair
In DepthDetails Article
TargetHLA class II histocompatibility antigen, DR beta 3 chain(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287635(1-[(S)-2-(3-Cyclohexyl-propionylamino)-3-(3H-imida...)
Affinity DataIC50: >1.00E+5nMAssay Description:Ability to compete for binding to Class II MHC using ELISA assay.More data for this Ligand-Target Pair
In DepthDetails Article
TargetHLA class II histocompatibility antigen, DR beta 3 chain(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287639((S)-3-({1-[(S)-6-Amino-2-(4-cyclohexyl-heptanoylam...)
Affinity DataIC50: >1.00E+5nMAssay Description:Ability to compete for binding to Class II MHC using ELISA assay.More data for this Ligand-Target Pair
In DepthDetails Article
TargetHLA class II histocompatibility antigen, DR beta 3 chain(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287644(1-[(S)-2-(2-Cyclohexylamino-acetylamino)-3-methyl-...)
Affinity DataIC50: >1.00E+5nMAssay Description:Ability to compete for binding to Class II MHC using ELISA assay.More data for this Ligand-Target Pair
In DepthDetails Article