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Found 98 Enz. Inhib. hit(s) with Target = 'rRNA adenine N-6-methyltransferase'
TargetrRNA adenine N-6-methyltransferase(Streptococcus pneumoniae)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50081297(1-[4-Amino-6-(indan-2-ylamino)-[1,3,5]triazin-2-yl...)
Affinity DataKi:  2.00E+3nMAssay Description:Inhibitory activity against ErmAM methylaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetrRNA adenine N-6-methyltransferase(Streptococcus pneumoniae)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50081299(CHEMBL125249 | N-(5-Fluoro-indan-2-yl)-6-piperidin...)
Affinity DataKi:  3.00E+3nMAssay Description:Inhibitory activity against ErmAM methylaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetrRNA adenine N-6-methyltransferase(Streptococcus pneumoniae)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50081279(6-(3-Amino-phenyl)-N-indan-2-yl-[1,3,5]triazine-2,...)
Affinity DataKi:  4.00E+3nMAssay Description:Inhibitory activity against ErmAM methylaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetrRNA adenine N-6-methyltransferase(Streptococcus pneumoniae)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50081285(CHEMBL124572 | N-(5-Methoxy-indan-2-yl)-6-piperidi...)
Affinity DataKi:  6.00E+3nMAssay Description:Inhibitory activity against ErmAM methylaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetrRNA adenine N-6-methyltransferase(Streptococcus pneumoniae)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50081300(2-(3-{4-[2-Amino-6-(indan-2-ylamino)-pyrimidin-4-y...)
Affinity DataKi:  7.50E+3nMAssay Description:Inhibitory activity against ErmAM methylaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetrRNA adenine N-6-methyltransferase(Streptococcus pneumoniae)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50081283(CHEMBL331440 | N-Indan-2-yl-6-piperidin-1-yl-[1,3,...)
Affinity DataKi:  8.00E+3nMAssay Description:Inhibitory activity against ErmAM methylaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetrRNA adenine N-6-methyltransferase(Streptococcus pneumoniae)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50081278(CHEMBL333812 | {1-[4-Amino-6-(indan-2-ylamino)-[1,...)
Affinity DataKi:  9.00E+3nMAssay Description:Inhibitory activity against ErmAM methylaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetrRNA adenine N-6-methyltransferase(Bacillus subtilis)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50081279(6-(3-Amino-phenyl)-N-indan-2-yl-[1,3,5]triazine-2,...)
Affinity DataKi:  1.00E+4nMAssay Description:Inhibitory activity against ErmC methylaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetrRNA adenine N-6-methyltransferase(Streptococcus pneumoniae)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50081275(2-{3-[4-Amino-6-(indan-2-ylamino)-[1,3,5]triazin-2...)
Affinity DataKi:  1.00E+4nMAssay Description:Inhibitory activity against ErmAM methylaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetrRNA adenine N-6-methyltransferase(Streptococcus pneumoniae)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50081292(CHEMBL338033 | N-Indan-2-yl-6-methylsulfanyl-[1,3,...)
Affinity DataKi:  1.00E+4nMAssay Description:Inhibitory activity against ErmAM methylaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetrRNA adenine N-6-methyltransferase(Bacillus subtilis)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50081300(2-(3-{4-[2-Amino-6-(indan-2-ylamino)-pyrimidin-4-y...)
Affinity DataKi:  1.25E+4nMAssay Description:Inhibitory activity against ErmC methylaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetrRNA adenine N-6-methyltransferase(Streptococcus pneumoniae)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50081276(CHEMBL330769 | {1-[4-Amino-6-(indan-2-ylamino)-[1,...)
Affinity DataKi:  1.25E+4nMAssay Description:Inhibitory activity against ErmAM methylaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetrRNA adenine N-6-methyltransferase(Bacillus subtilis)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50081297(1-[4-Amino-6-(indan-2-ylamino)-[1,3,5]triazin-2-yl...)
Affinity DataKi:  2.00E+4nMAssay Description:Inhibitory activity against ErmC methylaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetrRNA adenine N-6-methyltransferase(Streptococcus pneumoniae)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50081298(6-Cyclohexyl-N-indan-2-yl-[1,3,5]triazine-2,4-diam...)
Affinity DataKi:  2.50E+4nMAssay Description:Inhibitory activity against ErmAM methylaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetrRNA adenine N-6-methyltransferase(Streptococcus pneumoniae)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50081277(6-(4-Amino-phenyl)-N-indan-2-yl-[1,3,5]triazine-2,...)
Affinity DataKi:  3.50E+4nMAssay Description:Inhibitory activity against ErmAM methylaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetrRNA adenine N-6-methyltransferase(Bacillus subtilis)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50081299(CHEMBL125249 | N-(5-Fluoro-indan-2-yl)-6-piperidin...)
Affinity DataKi:  3.70E+4nMAssay Description:Inhibitory activity against ErmC methylaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetrRNA adenine N-6-methyltransferase(Streptococcus pneumoniae)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50009672(AdoHcy | CHEMBL418052 | S-(5'-adenosyl)-L-homocyst...)
Affinity DataKi:  4.00E+4nMAssay Description:Inhibitory activity against ErmAM methylaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetrRNA adenine N-6-methyltransferase(Streptococcus pneumoniae)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50009672(AdoHcy | CHEMBL418052 | S-(5'-adenosyl)-L-homocyst...)
Affinity DataKi:  4.00E+4nMAssay Description:Inhibition of ErmAM methylaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetrRNA adenine N-6-methyltransferase(Bacillus subtilis)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50081277(6-(4-Amino-phenyl)-N-indan-2-yl-[1,3,5]triazine-2,...)
Affinity DataKi: >5.00E+4nMAssay Description:Inhibitory activity against ErmC methylaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetrRNA adenine N-6-methyltransferase(Bacillus subtilis)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50081278(CHEMBL333812 | {1-[4-Amino-6-(indan-2-ylamino)-[1,...)
Affinity DataKi:  7.50E+4nMAssay Description:Inhibitory activity against ErmC methylaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetrRNA adenine N-6-methyltransferase(Bacillus subtilis)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50081285(CHEMBL124572 | N-(5-Methoxy-indan-2-yl)-6-piperidi...)
Affinity DataKi:  7.50E+4nMAssay Description:Inhibitory activity against ErmC methylaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetrRNA adenine N-6-methyltransferase(Streptococcus pneumoniae)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50081281(CHEMBL124520 | Indan-2-yl-(4-piperidin-1-yl-[1,3,5...)
Affinity DataKi: >7.50E+4nMAssay Description:Inhibitory activity against ErmAM methylaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetrRNA adenine N-6-methyltransferase(Bacillus subtilis)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50081283(CHEMBL331440 | N-Indan-2-yl-6-piperidin-1-yl-[1,3,...)
Affinity DataKi:  7.50E+4nMAssay Description:Inhibitory activity against ErmC methylaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetrRNA adenine N-6-methyltransferase(Streptococcus pneumoniae)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50081287(6-(4-Amino-phenyl)-N*4*-indan-2-yl-pyrimidine-2,4-...)
Affinity DataKi:  7.50E+4nMAssay Description:Inhibitory activity against ErmAM methylaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetrRNA adenine N-6-methyltransferase(Streptococcus pneumoniae)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50081286(CHEMBL124981 | N-Indan-1-yl-6-piperidin-1-yl-[1,3,...)
Affinity DataKi:  7.50E+4nMAssay Description:Inhibitory activity against ErmAM methylaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetrRNA adenine N-6-methyltransferase(Streptococcus pneumoniae)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50081294(CHEMBL125250 | N-Cyclohexyl-6-piperidin-1-yl-[1,3,...)
Affinity DataKi:  7.50E+4nMAssay Description:Inhibitory activity against ErmAM methylaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetrRNA adenine N-6-methyltransferase(Bacillus subtilis)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50081276(CHEMBL330769 | {1-[4-Amino-6-(indan-2-ylamino)-[1,...)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibitory activity against ErmC methylaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetrRNA adenine N-6-methyltransferase(Bacillus subtilis)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50081281(CHEMBL124520 | Indan-2-yl-(4-piperidin-1-yl-[1,3,5...)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibitory activity against ErmC methylaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetrRNA adenine N-6-methyltransferase(Bacillus subtilis)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50081282(CHEMBL419433 | N-Cyclohexyl-N'-indan-2-yl-[1,3,5]t...)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibitory activity against ErmC methylaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetrRNA adenine N-6-methyltransferase(Bacillus subtilis)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50081284(4,6-Di-piperidin-1-yl-[1,3,5]triazin-2-ylamine | C...)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibitory activity against ErmC methylaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetrRNA adenine N-6-methyltransferase(Bacillus subtilis)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50081287(6-(4-Amino-phenyl)-N*4*-indan-2-yl-pyrimidine-2,4-...)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibitory activity against ErmC methylaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetrRNA adenine N-6-methyltransferase(Bacillus subtilis)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50081275(2-{3-[4-Amino-6-(indan-2-ylamino)-[1,3,5]triazin-2...)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibitory activity against ErmC methylaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetrRNA adenine N-6-methyltransferase(Streptococcus pneumoniae)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50081289(CHEMBL124519 | N-Phenyl-6-piperidin-1-yl-[1,3,5]tr...)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibitory activity against ErmAM methylaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetrRNA adenine N-6-methyltransferase(Bacillus subtilis)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50081290(4-(Indan-2-ylamino)-6-piperidin-1-yl-[1,3,5]triazi...)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibitory activity against ErmC methylaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetrRNA adenine N-6-methyltransferase(Bacillus subtilis)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50081292(CHEMBL338033 | N-Indan-2-yl-6-methylsulfanyl-[1,3,...)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibitory activity against ErmC methylaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetrRNA adenine N-6-methyltransferase(Bacillus subtilis)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50081286(CHEMBL124981 | N-Indan-1-yl-6-piperidin-1-yl-[1,3,...)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibitory activity against ErmC methylaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetrRNA adenine N-6-methyltransferase(Bacillus subtilis)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50081291(CHEMBL123502 | N-((R)-1-Phenyl-ethyl)-6-piperidin-...)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibitory activity against ErmC methylaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetrRNA adenine N-6-methyltransferase(Streptococcus pneumoniae)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50081295(CHEMBL333773 | N-Cyclohexyl-N-methyl-6-piperidin-1...)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibitory activity against ErmAM methylaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetrRNA adenine N-6-methyltransferase(Bacillus subtilis)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50081294(CHEMBL125250 | N-Cyclohexyl-6-piperidin-1-yl-[1,3,...)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibitory activity against ErmC methylaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetrRNA adenine N-6-methyltransferase(Bacillus subtilis)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50081289(CHEMBL124519 | N-Phenyl-6-piperidin-1-yl-[1,3,5]tr...)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibitory activity against ErmC methylaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetrRNA adenine N-6-methyltransferase(Bacillus subtilis)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50081296(1-[4-Amino-6-(indan-2-ylamino)-[1,3,5]triazin-2-yl...)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibitory activity against ErmC methylaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetrRNA adenine N-6-methyltransferase(Streptococcus pneumoniae)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50081290(4-(Indan-2-ylamino)-6-piperidin-1-yl-[1,3,5]triazi...)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibitory activity against ErmAM methylaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetrRNA adenine N-6-methyltransferase(Streptococcus pneumoniae)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50081291(CHEMBL123502 | N-((R)-1-Phenyl-ethyl)-6-piperidin-...)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibitory activity against ErmAM methylaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetrRNA adenine N-6-methyltransferase(Bacillus subtilis)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50081295(CHEMBL333773 | N-Cyclohexyl-N-methyl-6-piperidin-1...)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibitory activity against ErmC methylaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetrRNA adenine N-6-methyltransferase(Streptococcus pneumoniae)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50081296(1-[4-Amino-6-(indan-2-ylamino)-[1,3,5]triazin-2-yl...)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibitory activity against ErmAM methylaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetrRNA adenine N-6-methyltransferase(Streptococcus pneumoniae)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50081282(CHEMBL419433 | N-Cyclohexyl-N'-indan-2-yl-[1,3,5]t...)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibitory activity against ErmAM methylaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetrRNA adenine N-6-methyltransferase(Streptococcus pneumoniae)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50081284(4,6-Di-piperidin-1-yl-[1,3,5]triazin-2-ylamine | C...)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibitory activity against ErmAM methylaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetrRNA adenine N-6-methyltransferase(Bacillus subtilis)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50081298(6-Cyclohexyl-N-indan-2-yl-[1,3,5]triazine-2,4-diam...)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibitory activity against ErmC methylaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetrRNA adenine N-6-methyltransferase(Streptococcus pneumoniae)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50086577((3R,4S,5S)-2-[4-Amino-6-(indan-2-ylamino)-[1,3,5]t...)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of ErmAM methylaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetrRNA adenine N-6-methyltransferase(Streptococcus pneumoniae)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50086578((1R,2S,3R,5S)-5-[4-Amino-6-(indan-2-ylamino)-[1,3,...)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of ErmAM methylaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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