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Found 874 Enz. Inhib. hit(s) with Target = 'Alpha-1,3-mannosyl-glycoprotein 2-beta-N-acetylglucosaminyltransferase'
LigandPNGBDBM308636(BDBM308807 | US9656955, Example 150 | trans-N-[2-c...)
Affinity DataKi: <1nMAssay Description:Radioligand binding assays using recombinant CHO cell membranes expressing human GlyT1: Radioligand binding to human GlyT1c transporter-expressing me...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM309106(Trans-N-(3-chlorobenzyl)-4-(4-fluorophenyl)-1-[(1-...)
Affinity DataKi: <10nMAssay Description:Radioligand binding assays using recombinant CHO cell membranes expressing human GlyT1: Radioligand binding to human GlyT1c transporter-expressing me...More data for this Ligand-Target Pair
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LigandPNGBDBM309109(Trans-N-(3,4-difluorobenzyl)-4-(4-fluorophenyl)-1-...)
Affinity DataKi: <10nMAssay Description:Radioligand binding assays using recombinant CHO cell membranes expressing human GlyT1: Radioligand binding to human GlyT1c transporter-expressing me...More data for this Ligand-Target Pair
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LigandPNGBDBM309120(Trans-N-(3-chloro-4-fluorobenzyl)-4-(4-fluoropheny...)
Affinity DataKi: <10nMAssay Description:Radioligand binding assays using recombinant CHO cell membranes expressing human GlyT1: Radioligand binding to human GlyT1c transporter-expressing me...More data for this Ligand-Target Pair
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LigandPNGBDBM309123((3R,4S)-N-[4-fluoro-3-(trifluoromethyl)phenyl]-1-[...)
Affinity DataKi: <10nMAssay Description:Radioligand binding assays using recombinant CHO cell membranes expressing human GlyT1: Radioligand binding to human GlyT1c transporter-expressing me...More data for this Ligand-Target Pair
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LigandPNGBDBM309124((3R,4S)vN-[4-fluoro-3-(trifluoromethoxy)phenyl]-1-...)
Affinity DataKi: <10nMAssay Description:Radioligand binding assays using recombinant CHO cell membranes expressing human GlyT1: Radioligand binding to human GlyT1c transporter-expressing me...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM309129((3R,4S)-4-(4-fluorophenyl)-N-[4-fluoro-3-(trifluor...)
Affinity DataKi: <10nMAssay Description:Radioligand binding assays using recombinant CHO cell membranes expressing human GlyT1: Radioligand binding to human GlyT1c transporter-expressing me...More data for this Ligand-Target Pair
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LigandPNGBDBM309129((3R,4S)-4-(4-fluorophenyl)-N-[4-fluoro-3-(trifluor...)
Affinity DataKi: <10nMAssay Description:Radioligand binding assays using recombinant CHO cell membranes expressing human GlyT1: Radioligand binding to human GlyT1c transporter-expressing me...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM309130((3R,4S)-4-(4-fluorophenyl)-N-[4-fluoro-3-(trifluor...)
Affinity DataKi: <10nMAssay Description:Radioligand binding assays using recombinant CHO cell membranes expressing human GlyT1: Radioligand binding to human GlyT1c transporter-expressing me...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM309143((3R,4S)-4-(4-fluorophenyl)-N-hexyl-1-[(1-methyl-1H...)
Affinity DataKi: <10nMAssay Description:Radioligand binding assays using recombinant CHO cell membranes expressing human GlyT1: Radioligand binding to human GlyT1c transporter-expressing me...More data for this Ligand-Target Pair
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LigandPNGBDBM309148((3R,4S)-1-[(1-methyl-1H-imidazol-4-yl)sulfonyl]-4-...)
Affinity DataKi: <10nMAssay Description:Radioligand binding assays using recombinant CHO cell membranes expressing human GlyT1: Radioligand binding to human GlyT1c transporter-expressing me...More data for this Ligand-Target Pair
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LigandPNGBDBM309159(Trans-1-[(1-methyl-1H-imidazol-4-yl)sulfonyl]-4-(t...)
Affinity DataKi: <10nMAssay Description:Radioligand binding assays using recombinant CHO cell membranes expressing human GlyT1: Radioligand binding to human GlyT1c transporter-expressing me...More data for this Ligand-Target Pair
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LigandPNGBDBM309163(BDBM309164 | Trans-1-[(1-methyl-1H-imidazol-4-yl)s...)
Affinity DataKi: <10nMAssay Description:Radioligand binding assays using recombinant CHO cell membranes expressing human GlyT1: Radioligand binding to human GlyT1c transporter-expressing me...More data for this Ligand-Target Pair
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LigandPNGBDBM309163(BDBM309164 | Trans-1-[(1-methyl-1H-imidazol-4-yl)s...)
Affinity DataKi: <10nMAssay Description:Radioligand binding assays using recombinant CHO cell membranes expressing human GlyT1: Radioligand binding to human GlyT1c transporter-expressing me...More data for this Ligand-Target Pair
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LigandPNGBDBM309199(N-{(3R,4S)-4-(4-fluorophenyl)-1-[(1-methyl-1H-imid...)
Affinity DataKi: <10nMAssay Description:Radioligand binding assays using recombinant CHO cell membranes expressing human GlyT1: Radioligand binding to human GlyT1c transporter-expressing me...More data for this Ligand-Target Pair
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LigandPNGBDBM309202(N-{(3R,4S)-4-(4-fluorophenyl)-1-[(1-methyl-1H-imid...)
Affinity DataKi: <10nMAssay Description:Radioligand binding assays using recombinant CHO cell membranes expressing human GlyT1: Radioligand binding to human GlyT1c transporter-expressing me...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM309204(6-(3-fluorophenyl)-N-{(3R,4S)-4-(4-fluorophenyl)-1...)
Affinity DataKi: <10nMAssay Description:Radioligand binding assays using recombinant CHO cell membranes expressing human GlyT1: Radioligand binding to human GlyT1c transporter-expressing me...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM309205(6-(4-fluorophenyl)-N-{(3R,4S)-4-(4-fluorophenyl)-1...)
Affinity DataKi: <10nMAssay Description:Radioligand binding assays using recombinant CHO cell membranes expressing human GlyT1: Radioligand binding to human GlyT1c transporter-expressing me...More data for this Ligand-Target Pair
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LigandPNGBDBM309206(6-(3-chlorophenyl)-N-{(3R,4S)-4-(4-fluorophenyl)-1...)
Affinity DataKi: <10nMAssay Description:Radioligand binding assays using recombinant CHO cell membranes expressing human GlyT1: Radioligand binding to human GlyT1c transporter-expressing me...More data for this Ligand-Target Pair
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LigandPNGBDBM309207(6-(4-chlorophenyl)-N-{(3R,4S)-4-(4-fluorophenyl)-1...)
Affinity DataKi: <10nMAssay Description:Radioligand binding assays using recombinant CHO cell membranes expressing human GlyT1: Radioligand binding to human GlyT1c transporter-expressing me...More data for this Ligand-Target Pair
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LigandPNGBDBM309210((3R,4S)-N-(2,2-difluorohexyl)-4-(4-fluorophenyl)-1...)
Affinity DataKi: <10nMAssay Description:Radioligand binding assays using recombinant CHO cell membranes expressing human GlyT1: Radioligand binding to human GlyT1c transporter-expressing me...More data for this Ligand-Target Pair
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LigandPNGBDBM309221((3R,4S)-4-(4-fluorophenyl)-1-[(1-methyl-1H-imidazo...)
Affinity DataKi: <10nMAssay Description:Radioligand binding assays using recombinant CHO cell membranes expressing human GlyT1: Radioligand binding to human GlyT1c transporter-expressing me...More data for this Ligand-Target Pair
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LigandPNGBDBM309222((3R,4S)-4-(4-fluorophenyl)-N-[4-fluoro-3-(pyridin-...)
Affinity DataKi: <10nMAssay Description:Radioligand binding assays using recombinant CHO cell membranes expressing human GlyT1: Radioligand binding to human GlyT1c transporter-expressing me...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM309223((3R,4S)-4-(4-fluorophenyl)-N-[4-fluoro-3-(pyridin-...)
Affinity DataKi: <10nMAssay Description:Radioligand binding assays using recombinant CHO cell membranes expressing human GlyT1: Radioligand binding to human GlyT1c transporter-expressing me...More data for this Ligand-Target Pair
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LigandPNGBDBM309224((3R,4S)-N-(4-fluoro-3-methylphenyl)-4-(4-fluorophe...)
Affinity DataKi: <10nMAssay Description:Radioligand binding assays using recombinant CHO cell membranes expressing human GlyT1: Radioligand binding to human GlyT1c transporter-expressing me...More data for this Ligand-Target Pair
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LigandPNGBDBM309225(5-fluoro-N-{(3R,4S)-4-(4-fluorophenyl)-1-[(1-methy...)
Affinity DataKi: <10nMAssay Description:Radioligand binding assays using recombinant CHO cell membranes expressing human GlyT1: Radioligand binding to human GlyT1c transporter-expressing me...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM309226((3R,4S)-4-(4-fluorophenyl)-N-[4-fluoro-3-(pyrimidi...)
Affinity DataKi: <10nMAssay Description:Radioligand binding assays using recombinant CHO cell membranes expressing human GlyT1: Radioligand binding to human GlyT1c transporter-expressing me...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM309236(4-chloro-N-{(3R,4S)-4-(4-fluorophenyl)-1-[(1-methy...)
Affinity DataKi: <10nMAssay Description:Radioligand binding assays using recombinant CHO cell membranes expressing human GlyT1: Radioligand binding to human GlyT1c transporter-expressing me...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM309253(4-(benzyloxy)-5-fluoro-N-{(3R,4S)-1-[(1-methyl-1H-...)
Affinity DataKi: <10nMAssay Description:Radioligand binding assays using recombinant CHO cell membranes expressing human GlyT1: Radioligand binding to human GlyT1c transporter-expressing me...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM309272(5-fluoro-N-{(3R,4S)-4-(4-fluorophenyl)-1-[(1-methy...)
Affinity DataKi: <10nMAssay Description:Radioligand binding assays using recombinant CHO cell membranes expressing human GlyT1: Radioligand binding to human GlyT1c transporter-expressing me...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM309277(Trans-4-(3-fluoropyridin-2-yl)-1-[(1-methyl-1H-imi...)
Affinity DataKi: <10nMAssay Description:Radioligand binding assays using recombinant CHO cell membranes expressing human GlyT1: Radioligand binding to human GlyT1c transporter-expressing me...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM309278((3R,4S)-4-(4-fluorophenyl)-1-[(1-methyl-1H-imidazo...)
Affinity DataKi: <10nMAssay Description:Radioligand binding assays using recombinant CHO cell membranes expressing human GlyT1: Radioligand binding to human GlyT1c transporter-expressing me...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM309280(5-fluoro-N-{(3R,4S)-1-[(1-methyl-1H-imidazol-4-yl)...)
Affinity DataKi: <10nMAssay Description:Radioligand binding assays using recombinant CHO cell membranes expressing human GlyT1: Radioligand binding to human GlyT1c transporter-expressing me...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM309282(5-chloro-N-{(3R,4S)-4-(4-fluorophenyl)-1-[(1-methy...)
Affinity DataKi: <10nMAssay Description:Radioligand binding assays using recombinant CHO cell membranes expressing human GlyT1: Radioligand binding to human GlyT1c transporter-expressing me...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM309283(N-{(3R,4S)-4-(4-fluorophenyl)-1-[(1-methyl-1H-imid...)
Affinity DataKi: <10nMAssay Description:Radioligand binding assays using recombinant CHO cell membranes expressing human GlyT1: Radioligand binding to human GlyT1c transporter-expressing me...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM309284(5-chloro-N-{(3R,4S)-1-[(1-methyl-1H-imidazol-4-yl)...)
Affinity DataKi: <10nMAssay Description:Radioligand binding assays using recombinant CHO cell membranes expressing human GlyT1: Radioligand binding to human GlyT1c transporter-expressing me...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM309285(N-{((3R,4S)-1-[(1-methyl-1H-imidazol-4-yl)sulfonyl...)
Affinity DataKi: <10nMAssay Description:Radioligand binding assays using recombinant CHO cell membranes expressing human GlyT1: Radioligand binding to human GlyT1c transporter-expressing me...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM309286(5-fluoro-N-{(3R,4S)-4-(4-fluorophenyl)-1-[(1-methy...)
Affinity DataKi: <10nMAssay Description:Radioligand binding assays using recombinant CHO cell membranes expressing human GlyT1: Radioligand binding to human GlyT1c transporter-expressing me...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM309291(Trans-1-[(1-methyl-1H-imidazol-4-yl)sulfonyl]-4-(t...)
Affinity DataKi: <10nMAssay Description:Radioligand binding assays using recombinant CHO cell membranes expressing human GlyT1: Radioligand binding to human GlyT1c transporter-expressing me...More data for this Ligand-Target Pair
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LigandPNGBDBM309293(Trans-N-[2-chloro-4-(trifluoromethyl)benzyl]-4-(3-...)
Affinity DataKi: <10nMAssay Description:Radioligand binding assays using recombinant CHO cell membranes expressing human GlyT1: Radioligand binding to human GlyT1c transporter-expressing me...More data for this Ligand-Target Pair
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LigandPNGBDBM309311(US9656955, Example 836 | trans-4-(4-fluorophenyl)-...)
Affinity DataKi: <10nMAssay Description:Radioligand binding assays using recombinant CHO cell membranes expressing human GlyT1: Radioligand binding to human GlyT1c transporter-expressing me...More data for this Ligand-Target Pair
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LigandPNGBDBM309312((3R,4S)-4-(4-fluorophenyl)-1-[(1-methyl-1H-1,2,3-t...)
Affinity DataKi: <10nMAssay Description:Radioligand binding assays using recombinant CHO cell membranes expressing human GlyT1: Radioligand binding to human GlyT1c transporter-expressing me...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM309313((3R,4S)-4-(4-fluorophenyl)-N-[4-fluoro-3-(trifluor...)
Affinity DataKi: <10nMAssay Description:Radioligand binding assays using recombinant CHO cell membranes expressing human GlyT1: Radioligand binding to human GlyT1c transporter-expressing me...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM309314((3R,4S)-4-(4-fluorophenyl)-1-[(1-methyl-1H-1,2,3-t...)
Affinity DataKi: <10nMAssay Description:Radioligand binding assays using recombinant CHO cell membranes expressing human GlyT1: Radioligand binding to human GlyT1c transporter-expressing me...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM309315((3R,4S)-4-(4-fluorophenyl)-N-[4-fluoro-3-(trifluor...)
Affinity DataKi: <10nMAssay Description:Radioligand binding assays using recombinant CHO cell membranes expressing human GlyT1: Radioligand binding to human GlyT1c transporter-expressing me...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM309316((3R,4S)-N-(3-chlorophenyl)-4-(4-fluorophenyl)-1-[(...)
Affinity DataKi: <10nMAssay Description:Radioligand binding assays using recombinant CHO cell membranes expressing human GlyT1: Radioligand binding to human GlyT1c transporter-expressing me...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM309317((3R,4S)-N-(3-chloro-4-fluorophenyl)-4-(4-fluorophe...)
Affinity DataKi: <10nMAssay Description:Radioligand binding assays using recombinant CHO cell membranes expressing human GlyT1: Radioligand binding to human GlyT1c transporter-expressing me...More data for this Ligand-Target Pair
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LigandPNGBDBM294227(US9586942, 1)
Affinity DataKi: <10nMAssay Description:Human GlyT1c expressing recombinant hGlyT1c_5_CHO cells were plated at 20,000 cells per well in 96 well Cytostar-T scintillation microplates (Amersha...More data for this Ligand-Target Pair
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LigandPNGBDBM294228(N-(1-((7S,8R)-7-(azetidin-1-yl)-8-benzyl-5,6,7,8-t...)
Affinity DataKi: <10nMAssay Description:Human GlyT1c expressing recombinant hGlyT1c_5_CHO cells were plated at 20,000 cells per well in 96 well Cytostar-T scintillation microplates (Amersha...More data for this Ligand-Target Pair
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LigandPNGBDBM294231(US9586942, 5*)
Affinity DataKi: <10nMAssay Description:Human GlyT1c expressing recombinant hGlyT1c_5_CHO cells were plated at 20,000 cells per well in 96 well Cytostar-T scintillation microplates (Amersha...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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