TargetApoptosis regulator BAX(Homo sapiens (Human))
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
Affinity DataKi: 43nMAssay Description:Displacement of Bak BH3 domain peptide from human Bax by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
TargetApoptosis regulator BAX(Homo sapiens (Human))
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
Affinity DataKi: 800nMAssay Description:Displacement of FITC-BIM from recombinant N-terminal GST-tagged human BAX expressed in Escherichia coli after 30 mins by fluorescence polarization as...More data for this Ligand-Target Pair
TargetApoptosis regulator BAX(Homo sapiens (Human))
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
Affinity DataKi: 1.00E+3nMAssay Description:Displacement of FITC-BIM from recombinant N-terminal GST-tagged human BAX expressed in Escherichia coli after 30 mins by fluorescence polarization as...More data for this Ligand-Target Pair
TargetApoptosis regulator BAX(Homo sapiens (Human))
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
Affinity DataKi: 1.10E+3nMAssay Description:Displacement of FITC-BIM from recombinant N-terminal GST-tagged human BAX expressed in Escherichia coli after 30 mins by fluorescence polarization as...More data for this Ligand-Target Pair
TargetApoptosis regulator BAX(Homo sapiens (Human))
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
Affinity DataKi: 1.20E+3nMAssay Description:Displacement of FITC-BIM from recombinant N-terminal GST-tagged human BAX expressed in Escherichia coli after 30 mins by fluorescence polarization as...More data for this Ligand-Target Pair
TargetApoptosis regulator BAX(Homo sapiens (Human))
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
Affinity DataKi: 1.30E+3nMAssay Description:Displacement of FITC-BIM from recombinant N-terminal GST-tagged human BAX expressed in Escherichia coli after 30 mins by fluorescence polarization as...More data for this Ligand-Target Pair
TargetApoptosis regulator BAX(Homo sapiens (Human))
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
Affinity DataKi: 1.30E+3nMAssay Description:Displacement of FITC-BIM from recombinant N-terminal GST-tagged human BAX expressed in Escherichia coli after 30 mins by fluorescence polarization as...More data for this Ligand-Target Pair
TargetApoptosis regulator BAX(Homo sapiens (Human))
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
Affinity DataKi: 1.70E+3nMAssay Description:Displacement of FITC-BIM from recombinant N-terminal GST-tagged human BAX expressed in Escherichia coli after 30 mins by fluorescence polarization as...More data for this Ligand-Target Pair
TargetApoptosis regulator BAX(Homo sapiens (Human))
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
Affinity DataKi: 2.50E+3nMAssay Description:Displacement of FITC-BIM from recombinant N-terminal GST-tagged human BAX expressed in Escherichia coli after 30 mins by fluorescence polarization as...More data for this Ligand-Target Pair
TargetApoptosis regulator BAX(Homo sapiens (Human))
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
Affinity DataKi: 9.10E+3nMAssay Description:Displacement of FITC-BIM from recombinant N-terminal GST-tagged human BAX expressed in Escherichia coli after 30 mins by fluorescence polarization as...More data for this Ligand-Target Pair
TargetApoptosis regulator BAX(Homo sapiens (Human))
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
Affinity DataKi: 1.26E+4nMAssay Description:Displacement of FITC-BIM from recombinant N-terminal GST-tagged human BAX expressed in Escherichia coli after 30 mins by fluorescence polarization as...More data for this Ligand-Target Pair
TargetApoptosis regulator BAX(Homo sapiens (Human))
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
Affinity DataKi: 1.29E+4nMAssay Description:Displacement of FITC-BIM from recombinant N-terminal GST-tagged human BAX expressed in Escherichia coli after 30 mins by fluorescence polarization as...More data for this Ligand-Target Pair
TargetApoptosis regulator BAX(Homo sapiens (Human))
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
Affinity DataKi: 1.35E+4nMAssay Description:Displacement of FITC-BIM from recombinant N-terminal GST-tagged human BAX expressed in Escherichia coli after 30 mins by fluorescence polarization as...More data for this Ligand-Target Pair
TargetApoptosis regulator BAX(Homo sapiens (Human))
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
Affinity DataKi: 1.58E+4nMAssay Description:Displacement of FITC-BIM from recombinant N-terminal GST-tagged human BAX expressed in Escherichia coli after 30 mins by fluorescence polarization as...More data for this Ligand-Target Pair
TargetApoptosis regulator BAX(Homo sapiens (Human))
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
Affinity DataKi: 3.09E+4nMAssay Description:Displacement of FITC-BIM from recombinant N-terminal GST-tagged human BAX expressed in Escherichia coli after 30 mins by fluorescence polarization as...More data for this Ligand-Target Pair
TargetApoptosis regulator BAX(Homo sapiens (Human))
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
Affinity DataKi: 6.31E+4nMAssay Description:Displacement of FITC-BIM from recombinant N-terminal GST-tagged human BAX expressed in Escherichia coli after 30 mins by fluorescence polarization as...More data for this Ligand-Target Pair
TargetApoptosis regulator BAX(Homo sapiens (Human))
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
Affinity DataKi: 8.51E+4nMAssay Description:Displacement of FITC-BIM from recombinant N-terminal GST-tagged human BAX expressed in Escherichia coli after 30 mins by fluorescence polarization as...More data for this Ligand-Target Pair
TargetApoptosis regulator BAX(Homo sapiens (Human))
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
Affinity DataIC50: 43nMAssay Description:Displacement of fluorescent Bak BH3 peptide domain from human recombinant Bax by competition fluorescence polarization assayMore data for this Ligand-Target Pair
TargetApoptosis regulator BAX(Homo sapiens (Human))
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
Ligand Info
TargetApoptosis regulator BAX(Homo sapiens (Human))
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
Affinity DataIC50: 250nMAssay Description:Activation of BAX (unknown origin)More data for this Ligand-Target Pair
TargetApoptosis regulator BAX(Homo sapiens (Human))
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
Affinity DataIC50: 3.00E+3nMAssay Description:Activation of Bax in human SMMC7721 cellsMore data for this Ligand-Target Pair
TargetApoptosis regulator BAX(Homo sapiens (Human))
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
Affinity DataIC50: 3.30E+3nMAssay Description:Activation of BAX (unknown origin)More data for this Ligand-Target Pair
TargetApoptosis regulator BAX(Homo sapiens (Human))
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
Ligand Info
TargetApoptosis regulator BAX(Homo sapiens (Human))
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
Ligand Info
TargetApoptosis regulator BAX(Homo sapiens (Human))
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
Ligand Info
TargetApoptosis regulator BAX(Homo sapiens (Human))
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
Affinity DataEC50: 809nMAssay Description:Binding affinity to recombinant human full length His-tagged BAX expressed in Escherichia coli BL21 (DE3) cells preincubated for 30 min followed by F...More data for this Ligand-Target Pair
TargetApoptosis regulator BAX(Homo sapiens (Human))
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
Affinity DataEC50: 2.22E+3nMAssay Description:Binding affinity to recombinant human full length His-tagged BAX expressed in Escherichia coli BL21 (DE3) cells preincubated for 30 min followed by F...More data for this Ligand-Target Pair
TargetApoptosis regulator BAX(Homo sapiens (Human))
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
Affinity DataEC50: 725nMAssay Description:Binding affinity to recombinant human full length His-tagged BAX expressed in Escherichia coli BL21 (DE3) cells preincubated for 30 min followed by F...More data for this Ligand-Target Pair
TargetApoptosis regulator BAX(Homo sapiens (Human))
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
Affinity DataEC50: 967nMAssay Description:Binding affinity to recombinant human full length His-tagged BAX expressed in Escherichia coli BL21 (DE3) cells preincubated for 30 min followed by F...More data for this Ligand-Target Pair
TargetApoptosis regulator BAX(Homo sapiens (Human))
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
Affinity DataEC50: 925nMAssay Description:Binding affinity to recombinant human full length His-tagged BAX expressed in Escherichia coli BL21 (DE3) cells preincubated for 30 min followed by F...More data for this Ligand-Target Pair
TargetApoptosis regulator BAX(Homo sapiens (Human))
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
Affinity DataEC50: 856nMAssay Description:Binding affinity to recombinant human full length His-tagged BAX expressed in Escherichia coli BL21 (DE3) cells preincubated for 30 min followed by F...More data for this Ligand-Target Pair
TargetApoptosis regulator BAX(Homo sapiens (Human))
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
Affinity DataEC50: 532nMAssay Description:Binding affinity to recombinant human full length His-tagged BAX expressed in Escherichia coli BL21 (DE3) cells preincubated for 30 min followed by F...More data for this Ligand-Target Pair
TargetApoptosis regulator BAX(Homo sapiens (Human))
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
Affinity DataEC50: 538nMAssay Description:Binding affinity to recombinant human full length His-tagged BAX expressed in Escherichia coli BL21 (DE3) cells preincubated for 30 min followed by F...More data for this Ligand-Target Pair
TargetApoptosis regulator BAX(Homo sapiens (Human))
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
Affinity DataEC50: 992nMAssay Description:Binding affinity to recombinant human full length His-tagged BAX expressed in Escherichia coli BL21 (DE3) cells preincubated for 30 min followed by F...More data for this Ligand-Target Pair
TargetApoptosis regulator BAX(Homo sapiens (Human))
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
Affinity DataEC50: 278nMAssay Description:Binding affinity to recombinant human full length His-tagged BAX expressed in Escherichia coli BL21 (DE3) cells preincubated for 30 min followed by F...More data for this Ligand-Target Pair
TargetApoptosis regulator BAX(Homo sapiens (Human))
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
Affinity DataEC50: >1.00E+4nMAssay Description:Binding affinity to recombinant human full length His-tagged BAX expressed in Escherichia coli BL21 (DE3) cells preincubated for 30 min followed by F...More data for this Ligand-Target Pair
TargetApoptosis regulator BAX(Homo sapiens (Human))
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
Affinity DataEC50: 719nMAssay Description:Binding affinity to recombinant human full length His-tagged BAX expressed in Escherichia coli BL21 (DE3) cells preincubated for 30 min followed by F...More data for this Ligand-Target Pair
TargetApoptosis regulator BAX(Homo sapiens (Human))
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
Affinity DataEC50: 874nMAssay Description:Binding affinity to recombinant human full length His-tagged BAX expressed in Escherichia coli BL21 (DE3) cells preincubated for 30 min followed by F...More data for this Ligand-Target Pair
TargetApoptosis regulator BAX(Homo sapiens (Human))
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
Affinity DataEC50: 704nMAssay Description:Binding affinity to recombinant human full length His-tagged BAX expressed in Escherichia coli BL21 (DE3) cells preincubated for 30 min followed by F...More data for this Ligand-Target Pair
TargetApoptosis regulator BAX(Homo sapiens (Human))
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
Ligand Info
TargetApoptosis regulator BAX(Homo sapiens (Human))
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
TargetApoptosis regulator BAX(Homo sapiens (Human))
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
Affinity DataEC50: 700nMAssay Description:Activation of Bax in human HuH7 cells assessed as inhibition of mitochondrial accumulation of fluorescent probe Mitotracker Red after 12 to 72 hrs by...More data for this Ligand-Target Pair
TargetApoptosis regulator BAX(Homo sapiens (Human))
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
Affinity DataEC50: 8.20E+3nMAssay Description:Activation of Bax in human HuH7 cells assessed as inhibition of mitochondrial accumulation of fluorescent probe Mitotracker Red after 12 to 72 hrs by...More data for this Ligand-Target Pair
TargetApoptosis regulator BAX(Homo sapiens (Human))
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
Ligand Info
TargetApoptosis regulator BAX(Homo sapiens (Human))
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
TargetApoptosis regulator BAX(Homo sapiens (Human))
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
Affinity DataEC50: 1.14E+3nMAssay Description:Binding affinity to recombinant human full length His-tagged BAX expressed in Escherichia coli BL21 (DE3) cells preincubated for 30 min followed by F...More data for this Ligand-Target Pair
TargetApoptosis regulator BAX(Homo sapiens (Human))
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
Affinity DataEC50: 393nMAssay Description:Binding affinity to recombinant human full length His-tagged BAX expressed in Escherichia coli BL21 (DE3) cells preincubated for 30 min followed by F...More data for this Ligand-Target Pair