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Found 8 Enz. Inhib. hit(s) with Target = 'Bromodomain-containing protein 3 [1-435]'
TargetBromodomain-containing protein 3 [1-435](Homo sapiens (Human))
Beigene

US Patent
LigandPNGBDBM237471(US9393232, 2.46)
Affinity DataIC50:  5.30nMpH: 7.5Assay Description:The assay was carried out in binding mixtures of the bromodomain protein, 0-10 μM compounds and tetra-acetylated histone peptide (SGRGAC.KGGAC.K...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetBromodomain-containing protein 3 [1-435](Homo sapiens (Human))
Beigene

US Patent
LigandPNGBDBM237443(US9393232, 2.16)
Affinity DataIC50:  9.90nMpH: 7.5Assay Description:The assay was carried out in binding mixtures of the bromodomain protein, 0-10 μM compounds and tetra-acetylated histone peptide (SGRGAC.KGGAC.K...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetBromodomain-containing protein 3 [1-435](Homo sapiens (Human))
Beigene

US Patent
LigandPNGBDBM237494(US9393232, 4.1 | US9393232, 4.1a | US9393232, 4.1b)
Affinity DataIC50:  14nMpH: 7.5Assay Description:The assay was carried out in binding mixtures of the bromodomain protein, 0-10 μM compounds and tetra-acetylated histone peptide (SGRGAC.KGGAC.K...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetBromodomain-containing protein 3 [1-435](Homo sapiens (Human))
Beigene

US Patent
LigandPNGBDBM237509(US9393232, 2.10a | US9393232, 2.10b)
Affinity DataIC50:  23nMpH: 7.5Assay Description:The assay was carried out in binding mixtures of the bromodomain protein, 0-10 μM compounds and tetra-acetylated histone peptide (SGRGAC.KGGAC.K...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetBromodomain-containing protein 3 [1-435](Homo sapiens (Human))
Beigene

US Patent
LigandPNGBDBM237521(US9393232, 2.22)
Affinity DataIC50:  23nMpH: 7.5Assay Description:The assay was carried out in binding mixtures of the bromodomain protein, 0-10 μM compounds and tetra-acetylated histone peptide (SGRGAC.KGGAC.K...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetBromodomain-containing protein 3 [1-435](Homo sapiens (Human))
Beigene

US Patent
LigandPNGBDBM237422(US9393232, 1.30a | US9393232, 1.30b)
Affinity DataIC50:  25nMpH: 7.5Assay Description:The assay was carried out in binding mixtures of the bromodomain protein, 0-10 μM compounds and tetra-acetylated histone peptide (SGRGAC.KGGAC.K...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetBromodomain-containing protein 3 [1-435](Homo sapiens (Human))
Beigene

US Patent
LigandPNGBDBM237428(US9393232, 2.2 | US9393232, 2.2a | US9393232, 2.2b)
Affinity DataIC50:  35nMpH: 7.5Assay Description:The assay was carried out in binding mixtures of the bromodomain protein, 0-10 μM compounds and tetra-acetylated histone peptide (SGRGAC.KGGAC.K...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetBromodomain-containing protein 3 [1-435](Homo sapiens (Human))
Beigene

US Patent
LigandPNGBDBM237408(US9393232, 1.16)
Affinity DataIC50:  140nMpH: 7.5Assay Description:The assay was carried out in binding mixtures of the bromodomain protein, 0-10 μM compounds and tetra-acetylated histone peptide (SGRGAC.KGGAC.K...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent