Affinity DataKi: 0.100nMAssay Description:Binding affinity against human cathepsin EMore data for this Ligand-Target Pair
Affinity DataKi: 0.5nMAssay Description:Binding affinity against human cathepsin EMore data for this Ligand-Target Pair
Affinity DataKi: 0.5nMAssay Description:Binding affinity against human cathepsin EMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Binding affinity against human cathepsin EMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Inhibition of cathepsin EMore data for this Ligand-Target Pair
Affinity DataKi: 2.20nMAssay Description:Binding affinity against human cathepsin EMore data for this Ligand-Target Pair
Affinity DataKi: 2.90nMAssay Description:Binding affinity against human cathepsin EMore data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:Compound was evaluated for aspartyl protease inhibition selectivity relative to Cathepsin EMore data for this Ligand-Target Pair
Affinity DataKi: 3.30nMAssay Description:Binding affinity against human cathepsin EMore data for this Ligand-Target Pair
Affinity DataKi: 5nMAssay Description:Binding affinity to human cathepsin EMore data for this Ligand-Target Pair
Affinity DataKi: 5nMAssay Description:Inhibition of cathepsin EMore data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Binding affinity against human cathepsin EMore data for this Ligand-Target Pair
Affinity DataKi: 15nMAssay Description:Binding affinity against human cathepsin EMore data for this Ligand-Target Pair
Affinity DataKi: 17nMAssay Description:Binding affinity against human cathepsin EMore data for this Ligand-Target Pair
Affinity DataKi: 21nMAssay Description:Binding affinity against human cathepsin EMore data for this Ligand-Target Pair
Affinity DataKi: 24nMAssay Description:Binding affinity to human cathepsin EMore data for this Ligand-Target Pair
Affinity DataKi: 24nMAssay Description:Inhibition of cathepsin EMore data for this Ligand-Target Pair
Affinity DataKi: 30nMAssay Description:Inhibition of cathepsin EMore data for this Ligand-Target Pair
Affinity DataKi: 44nMAssay Description:Binding affinity against human cathepsin EMore data for this Ligand-Target Pair
Affinity DataKi: 50nMAssay Description:Compound was evaluated for aspartyl protease inhibition selectivity relative to Cathepsin EMore data for this Ligand-Target Pair
Affinity DataKi: 86nMAssay Description:Inhibition oh cathepsin EMore data for this Ligand-Target Pair
Affinity DataKi: 90nMAssay Description:Compound was evaluated for aspartyl protease inhibition selectivity relative to Cathepsin EMore data for this Ligand-Target Pair
Affinity DataKi: 142nMAssay Description:Compound was evaluated for aspartyl protease inhibition selectivity relative to Cathepsin EMore data for this Ligand-Target Pair
Affinity DataKi: 300nMAssay Description:Binding affinity against human cathepsin EMore data for this Ligand-Target Pair
Affinity DataKi: 440nMAssay Description:Inhibition of human cathepsin E assessed as inhibition constant using ACC-GKPILFFRILK-(DNP)-(dR)-NH2 as substrate by spectrophotometric analysisMore data for this Ligand-Target Pair
Affinity DataKi: 850nMAssay Description:Binding affinity against human cathepsin EMore data for this Ligand-Target Pair
Affinity DataKi: 1.10E+3nMAssay Description:Inhibition of CathE (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity against human cathepsin EMore data for this Ligand-Target Pair
Affinity DataKi: >3.06E+4nMAssay Description:Inhibition of human cathepsin EMore data for this Ligand-Target Pair
Affinity DataIC50: 0.0800nMAssay Description:Inhibition of human recombinant cathepsin E using Mca-Gly-Lys-Pro-Ile-Leu-Phe-Phe-Arg-Leu-Lys-(Dnp)-D-Arg-NH2 as substrate preincubated for 15 mins f...More data for this Ligand-Target Pair
Affinity DataIC50: 0.100nMAssay Description:Inhibition of secreted cathepsin E in human MDA-MB-231 cells using Mca-Gly-Lys-Pro-Ile-Leu-PhePhe-Arg-Leu-Lys-(Dnp)-D-Arg-NH2 as substrate pretreated...More data for this Ligand-Target Pair
Affinity DataIC50: 0.181nMAssay Description:Inhibition of cathepsin EMore data for this Ligand-Target Pair
Affinity DataIC50: 0.300nMAssay Description:Inhibition of recombinant human C-terminal His10-tagged cathepsin E (Gln18 to Pro396 residues) using Mca-Gly-Lys-Pro-Ile-Leu-PhePhe-Arg-Leu-Lys-(Dnp)...More data for this Ligand-Target Pair
Affinity DataIC50: 0.300nMAssay Description:Inhibition of cathepsin EMore data for this Ligand-Target Pair
Affinity DataIC50: 0.354nMAssay Description:Inhibition of cathepsin EMore data for this Ligand-Target Pair
Affinity DataIC50: 0.400nMAssay Description:Inhibition of recombinant human C-terminal His10-tagged cathepsin E (Gln18 to Pro396 residues) using Mca-Gly-Lys-Pro-Ile-Leu-PhePhe-Arg-Leu-Lys-(Dnp)...More data for this Ligand-Target Pair
Affinity DataIC50: 0.400nMAssay Description:Inhibition of cathepsin EMore data for this Ligand-Target Pair
Affinity DataIC50: 0.446nMAssay Description:Inhibition of cathepsin E by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.446nMAssay Description:Inhibition of Cathepsin E (unknown origin) using Mca-Gly-Lys-Pro-Ile-Leu-Phe-Phe-Arg-Leu-Lys-(Dnp)-D-Arg-NH2 as substrate incubated for 120 mins by f...More data for this Ligand-Target Pair
Affinity DataIC50: 0.5nMAssay Description:Inhibition of recombinant human C-terminal His10-tagged cathepsin E (Gln18 to Pro396 residues) using Mca-Gly-Lys-Pro-Ile-Leu-PhePhe-Arg-Leu-Lys-(Dnp)...More data for this Ligand-Target Pair
Affinity DataIC50: 0.724nMAssay Description:Inhibition of Cathepsin E (unknown origin) using Mca-Gly-Lys-Pro-Ile-Leu-Phe-Phe-Arg-Leu-Lys-(Dnp)-D-Arg-NH2 as substrate incubated for 120 mins by f...More data for this Ligand-Target Pair
Affinity DataIC50: 0.724nMAssay Description:Inhibition of cathepsin E by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.800nMAssay Description:Inhibition of cathepsin E by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.800nMAssay Description:Inhibition of cathepsin E using MCA-KPILFFRLK(Dnp)-D-R-NH2 as substrate incubated for 10 to 15 mins prior to substrate addition measured every 5 min ...More data for this Ligand-Target Pair
Affinity DataIC50: 0.886nMAssay Description:Inhibition of cathepsin EMore data for this Ligand-Target Pair
Affinity DataIC50: 0.900nMAssay Description:Inhibition of recombinant human C-terminal His10-tagged cathepsin E (Gln18 to Pro396 residues) using Mca-Gly-Lys-Pro-Ile-Leu-PhePhe-Arg-Leu-Lys-(Dnp)...More data for this Ligand-Target Pair
Affinity DataIC50: 1.90nMAssay Description:Inhibition of cathepsin E by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 4nMAssay Description:Inhibition of cathepsin EMore data for this Ligand-Target Pair
Affinity DataIC50: 4.90nMAssay Description:Inhibition of cathepsin E by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Inhibition of recombinant human C-terminal His10-tagged cathepsin E (Gln18 to Pro396 residues) using Mca-Gly-Lys-Pro-Ile-Leu-PhePhe-Arg-Leu-Lys-(Dnp)...More data for this Ligand-Target Pair