Compile Data Set for Download or QSAR
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Found 151 Enz. Inhib. hit(s) with Target = 'Dual specificity testis-specific protein kinase 1'
TargetDual specificity testis-specific protein kinase 1(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM2579((2S,3R,4R,6R)-3-methoxy-2-methyl-4-(methylamino)-2...)
Affinity DataIC50:  138nMAssay Description:Inhibition of human TESK1 using cofilin as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity testis-specific protein kinase 1(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM2579((2S,3R,4R,6R)-3-methoxy-2-methyl-4-(methylamino)-2...)
Affinity DataIC50:  261nMAssay Description:Inhibition of human TESK1 using cofilin as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity testis-specific protein kinase 1(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50390791(CHEMBL2070615)
Affinity DataIC50:  455nMAssay Description:Inhibition of TESK1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity testis-specific protein kinase 1(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50390790(CHEMBL2070614)
Affinity DataIC50:  1.13E+3nMAssay Description:Inhibition of TESK1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity testis-specific protein kinase 1(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50390789(CHEMBL2070613)
Affinity DataIC50:  2.20E+3nMAssay Description:Inhibition of TESK1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity testis-specific protein kinase 1(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50390792(CHEMBL2070616)
Affinity DataIC50:  2.27E+3nMAssay Description:Inhibition of TESK1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity testis-specific protein kinase 1(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50135286(CHEMBL3745885)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human TESK1 using cofilin as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity testis-specific protein kinase 1(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50401152(CHEMBL2205766)
Affinity DataIC50: <1.00E+4nMAssay Description:Inhibition of TESK1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity testis-specific protein kinase 1(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50390793(CHEMBL2070617)
Affinity DataIC50:  1.19E+4nMAssay Description:Inhibition of TESK1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity testis-specific protein kinase 1(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50390788(CHEMBL2070612)
Affinity DataIC50: >1.25E+4nMAssay Description:Inhibition of TESK1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity testis-specific protein kinase 1(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50390782(CHEMBL2070500)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of TESK1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity testis-specific protein kinase 1(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50390796(CHEMBL2070501)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of TESK1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity testis-specific protein kinase 1(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50390783(CHEMBL2070502)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of TESK1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity testis-specific protein kinase 1(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50390784(CHEMBL2070503)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of TESK1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity testis-specific protein kinase 1(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50390785(CHEMBL2070504)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of TESK1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity testis-specific protein kinase 1(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50390786(CHEMBL2070505)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of TESK1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity testis-specific protein kinase 1(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50390787(CHEMBL2070611)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of TESK1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity testis-specific protein kinase 1(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50390778(CHEMBL2070496)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of TESK1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity testis-specific protein kinase 1(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50390777(CHEMBL2070495)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of TESK1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity testis-specific protein kinase 1(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50390776(CHEMBL2070494)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of TESK1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity testis-specific protein kinase 1(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50390794(CHEMBL2070618)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of TESK1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity testis-specific protein kinase 1(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50390795(CHEMBL2070619)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of TESK1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity testis-specific protein kinase 1(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50390775(CHEMBL2070493)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of TESK1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity testis-specific protein kinase 1(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50390774(CHEMBL2070492)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of TESK1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity testis-specific protein kinase 1(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50390779(CHEMBL2070497)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of TESK1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity testis-specific protein kinase 1(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50390780(CHEMBL2070498)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of TESK1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity testis-specific protein kinase 1(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50390781(CHEMBL2070499)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of TESK1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity testis-specific protein kinase 1(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM31085(1-[4-[(4-ethyl-1-piperazinyl)methyl]-3-(trifluorom...)
Affinity DataKd:  2.40E+3nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetDual specificity testis-specific protein kinase 1(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM4779(CHEMBL31965 | CHEMBL545315 | CI-1033 | Canertinib ...)
Affinity DataKd:  3.20E+3nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetDual specificity testis-specific protein kinase 1(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM13216(BMS-354825 | CHEMBL1421 | DASATINIB | N-(2-Chloro-...)
Affinity DataKd:  33nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetDual specificity testis-specific protein kinase 1(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM6866(1-Acyl-1H-[1,2,4]triazole-3,5-diamine Analogue 3b ...)
Affinity DataKd:  3.10E+3nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetDual specificity testis-specific protein kinase 1(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM31096(CHEMBL290084 | Staurosporine | cid_451705)
Affinity DataKd:  320nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetDual specificity testis-specific protein kinase 1(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM13534(CHEMBL572878 | N-[4-({4-[(3-methyl-1H-pyrazol-5-yl...)
Affinity DataKd:  5.60E+3nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetDual specificity testis-specific protein kinase 1(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM21(CHEMBL24828 | N-(4-bromo-2-fluorophenyl)-6-methoxy...)
Affinity DataKd:  3.70E+3nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetDual specificity testis-specific protein kinase 1(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50308060(16-hydroxy-16-(hydroxymethyl)-15-methyl-28-oxa-4,1...)
Affinity DataKd:  290nMAssay Description:Binding affinity to TESK1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity testis-specific protein kinase 1(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50326053(CHEMBL608533 | PKC-412)
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to TESK1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity testis-specific protein kinase 1(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM2579((2S,3R,4R,6R)-3-methoxy-2-methyl-4-(methylamino)-2...)
Affinity DataKd:  320nMAssay Description:Binding constant for TESK1 kinase domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity testis-specific protein kinase 1(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50326053(CHEMBL608533 | PKC-412)
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for TESK1 kinase domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity testis-specific protein kinase 1(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50308060(16-hydroxy-16-(hydroxymethyl)-15-methyl-28-oxa-4,1...)
Affinity DataKd:  290nMAssay Description:Binding constant for TESK1 kinase domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity testis-specific protein kinase 1(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50026612(BIBF-1120 | Nintedanib | US10981896, Compound Nint...)
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for TESK1 kinase domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity testis-specific protein kinase 1(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50326053(CHEMBL608533 | PKC-412)
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for TESK1 kinase domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity testis-specific protein kinase 1(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM2579((2S,3R,4R,6R)-3-methoxy-2-methyl-4-(methylamino)-2...)
Affinity DataKd:  320nMAssay Description:Binding constant for TESK1 kinase domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity testis-specific protein kinase 1(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50300690(1-(5-Tert-Butyl-1,2-Oxazol-3-Yl)-3-(4-{7-[2-(Morph...)
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to TESK1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity testis-specific protein kinase 1(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50326054(CHEMBL1240703)
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to TESK1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity testis-specific protein kinase 1(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM13535(4-[6-methoxy-7-(3-piperidin-1-ylpropoxy)quinazolin...)
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to TESK1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity testis-specific protein kinase 1(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM16673(4-[4-({[4-chloro-3-(trifluoromethyl)phenyl]carbamo...)
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to TESK1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity testis-specific protein kinase 1(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM4814(CHEMBL535 | N-[2-(diethylamino)ethyl]-5-[(Z)-(5-fl...)
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to TESK1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity testis-specific protein kinase 1(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM5446(CHEMBL553 | ERLOTINIB HYDROCHLORIDE | Erlotinib | ...)
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for TESK1 kinase domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity testis-specific protein kinase 1(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM6568(6-(2,6-dichlorophenyl)-8-methyl-2-{[3-(methylsulfa...)
Affinity DataKd:  79nMAssay Description:Binding constant for TESK1 kinase domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity testis-specific protein kinase 1(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM26300(2-{3-[(7-{3-[ethyl(2-hydroxyethyl)amino]propoxy}qu...)
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for TESK1 kinase domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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