Compile Data Set for Download or QSAR
maximum 50k data
Found 26 Enz. Inhib. hit(s) with Target = 'CAAX prenyl protease 2'
TargetCAAX prenyl protease 2(Homo sapiens (Human))
New York University Abu Dhabi

Curated by ChEMBL
LigandPNGBDBM50500099(CHEMBL3741765)
Affinity DataIC50:  3.80E+3nMAssay Description:Inhibition of human Rce1-mediated CaaX protease activity using ABZ-KSKTKC(farnesyl)QIIM and ABZ-KSKTKC(farnesyl)VIQI as substrate assessed as residua...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCAAX prenyl protease 2(Homo sapiens (Human))
New York University Abu Dhabi

Curated by ChEMBL
LigandPNGBDBM50500092(CHEMBL3741937)
Affinity DataIC50:  3.90E+3nMAssay Description:Inhibition of human Rce1-mediated CaaX protease activity using ABZ-KSKTKC(farnesyl)QIIM and ABZ-KSKTKC(farnesyl)VIQI as substrate assessed as residua...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCAAX prenyl protease 2(Homo sapiens (Human))
New York University Abu Dhabi

Curated by ChEMBL
LigandPNGBDBM50500097(CHEMBL3740962)
Affinity DataIC50:  4.20E+3nMAssay Description:Inhibition of human Rce1-mediated CaaX protease activity using ABZ-KSKTKC(farnesyl)QIIM and ABZ-KSKTKC(farnesyl)VIQI as substrate assessed as residua...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCAAX prenyl protease 2(Homo sapiens (Human))
New York University Abu Dhabi

Curated by ChEMBL
LigandPNGBDBM50500105(CHEMBL3740249)
Affinity DataIC50:  4.90E+3nMAssay Description:Inhibition of human Rce1-mediated CaaX protease activity using ABZ-KSKTKC(farnesyl)QIIM and ABZ-KSKTKC(farnesyl)VIQI as substrate assessed as residua...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCAAX prenyl protease 2(Homo sapiens (Human))
New York University Abu Dhabi

Curated by ChEMBL
LigandPNGBDBM50500103(CHEMBL3742211)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of human Rce1-mediated CaaX protease activity using ABZ-KSKTKC(farnesyl)QIIM and ABZ-KSKTKC(farnesyl)VIQI as substrate assessed as residua...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCAAX prenyl protease 2(Homo sapiens (Human))
New York University Abu Dhabi

Curated by ChEMBL
LigandPNGBDBM50500098(CHEMBL3741101)
Affinity DataIC50:  5.30E+3nMAssay Description:Inhibition of human Rce1-mediated CaaX protease activity using ABZ-KSKTKC(farnesyl)QIIM and ABZ-KSKTKC(farnesyl)VIQI as substrate assessed as residua...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCAAX prenyl protease 2(Homo sapiens (Human))
New York University Abu Dhabi

Curated by ChEMBL
LigandPNGBDBM50500106(CHEMBL3741673)
Affinity DataIC50:  5.40E+3nMAssay Description:Inhibition of human Rce1-mediated CaaX protease activity using ABZ-KSKTKC(farnesyl)QIIM and ABZ-KSKTKC(farnesyl)VIQI as substrate assessed as residua...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCAAX prenyl protease 2(Homo sapiens (Human))
New York University Abu Dhabi

Curated by ChEMBL
LigandPNGBDBM50500094(CHEMBL3740203)
Affinity DataIC50:  6.70E+3nMAssay Description:Inhibition of human Rce1-mediated CaaX protease activity using ABZ-KSKTKC(farnesyl)QIIM and ABZ-KSKTKC(farnesyl)VIQI as substrate assessed as residua...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCAAX prenyl protease 2(Homo sapiens (Human))
New York University Abu Dhabi

Curated by ChEMBL
LigandPNGBDBM50500101(CHEMBL1979298)
Affinity DataIC50:  6.90E+3nMAssay Description:Inhibition of human Rce1-mediated CaaX protease activity using ABZ-KSKTKC(farnesyl)QIIM and ABZ-KSKTKC(farnesyl)VIQI as substrate assessed as residua...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCAAX prenyl protease 2(Homo sapiens (Human))
New York University Abu Dhabi

Curated by ChEMBL
LigandPNGBDBM50096861(CHEMBL440905 | Heptadecanoic acid {[3-(2,3-dimethy...)
Affinity DataIC50:  7.00E+3nMAssay Description:Inhibition of recombinant prenyl protein-specific protease Rce1 expressed in Sf9 cells at 10 uMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCAAX prenyl protease 2(Homo sapiens (Human))
New York University Abu Dhabi

Curated by ChEMBL
LigandPNGBDBM50096860((E)-3-Biphenyl-4-yl-N-{2-[3-(2,3-dimethyl-phenylsu...)
Affinity DataIC50:  7.00E+3nMAssay Description:Inhibition of recombinant prenyl protein-specific protease Rce1 expressed in Sf9 cells at 10 uMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCAAX prenyl protease 2(Homo sapiens (Human))
New York University Abu Dhabi

Curated by ChEMBL
LigandPNGBDBM50500091(CHEMBL3740563)
Affinity DataIC50:  7.10E+3nMAssay Description:Inhibition of human Rce1-mediated CaaX protease activity using ABZ-KSKTKC(farnesyl)QIIM and ABZ-KSKTKC(farnesyl)VIQI as substrate assessed as residua...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCAAX prenyl protease 2(Homo sapiens (Human))
New York University Abu Dhabi

Curated by ChEMBL
LigandPNGBDBM50480670(CHEMBL553161)
Affinity DataIC50:  7.30E+3nMAssay Description:Inhibition of human RCE1More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCAAX prenyl protease 2(Homo sapiens (Human))
New York University Abu Dhabi

Curated by ChEMBL
LigandPNGBDBM50500100(CHEMBL3740034)
Affinity DataIC50:  8.20E+3nMAssay Description:Inhibition of human Rce1-mediated CaaX protease activity using ABZ-KSKTKC(farnesyl)QIIM and ABZ-KSKTKC(farnesyl)VIQI as substrate assessed as residua...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCAAX prenyl protease 2(Homo sapiens (Human))
New York University Abu Dhabi

Curated by ChEMBL
LigandPNGBDBM50500095(CHEMBL2003928)
Affinity DataIC50:  8.80E+3nMAssay Description:Inhibition of human Rce1-mediated CaaX protease activity using ABZ-KSKTKC(farnesyl)QIIM and ABZ-KSKTKC(farnesyl)VIQI as substrate assessed as residua...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCAAX prenyl protease 2(Homo sapiens (Human))
New York University Abu Dhabi

Curated by ChEMBL
LigandPNGBDBM50500107(CHEMBL3741464)
Affinity DataIC50:  8.90E+3nMAssay Description:Inhibition of human Rce1-mediated CaaX protease activity using ABZ-KSKTKC(farnesyl)QIIM and ABZ-KSKTKC(farnesyl)VIQI as substrate assessed as residua...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCAAX prenyl protease 2(Homo sapiens (Human))
New York University Abu Dhabi

Curated by ChEMBL
LigandPNGBDBM50500102(CHEMBL3740606)
Affinity DataIC50:  9.40E+3nMAssay Description:Inhibition of human Rce1-mediated CaaX protease activity using ABZ-KSKTKC(farnesyl)QIIM and ABZ-KSKTKC(farnesyl)VIQI as substrate assessed as residua...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCAAX prenyl protease 2(Homo sapiens (Human))
New York University Abu Dhabi

Curated by ChEMBL
LigandPNGBDBM50500109(CHEMBL3740547)
Affinity DataIC50:  9.80E+3nMAssay Description:Inhibition of human Rce1-mediated CaaX protease activity using ABZ-KSKTKC(farnesyl)QIIM and ABZ-KSKTKC(farnesyl)VIQI as substrate assessed as residua...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCAAX prenyl protease 2(Homo sapiens (Human))
New York University Abu Dhabi

Curated by ChEMBL
LigandPNGBDBM50500093(CHEMBL2006267)
Affinity DataIC50:  1.10E+4nMAssay Description:Inhibition of human Rce1-mediated CaaX protease activity using ABZ-KSKTKC(farnesyl)QIIM and ABZ-KSKTKC(farnesyl)VIQI as substrate assessed as residua...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCAAX prenyl protease 2(Homo sapiens (Human))
New York University Abu Dhabi

Curated by ChEMBL
LigandPNGBDBM50096862((9Z,12Z)-Octadeca-9,12-dienoic acid {2-[3-(2,3-dim...)
Affinity DataIC50:  1.40E+4nMAssay Description:Inhibition of recombinant prenyl protein-specific protease Rcel expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCAAX prenyl protease 2(Homo sapiens (Human))
New York University Abu Dhabi

Curated by ChEMBL
LigandPNGBDBM50500096(CHEMBL3739720)
Affinity DataIC50:  1.40E+4nMAssay Description:Inhibition of human Rce1-mediated CaaX protease activity using ABZ-KSKTKC(farnesyl)QIIM and ABZ-KSKTKC(farnesyl)VIQI as substrate assessed as residua...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCAAX prenyl protease 2(Homo sapiens (Human))
New York University Abu Dhabi

Curated by ChEMBL
LigandPNGBDBM50500108(CHEMBL3740917)
Affinity DataIC50:  1.60E+4nMAssay Description:Inhibition of human Rce1-mediated CaaX protease activity using ABZ-KSKTKC(farnesyl)QIIM and ABZ-KSKTKC(farnesyl)VIQI as substrate assessed as residua...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCAAX prenyl protease 2(Homo sapiens (Human))
New York University Abu Dhabi

Curated by ChEMBL
LigandPNGBDBM50480671(CHEMBL555914)
Affinity DataIC50:  1.70E+4nMAssay Description:Inhibition of human RCE1More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCAAX prenyl protease 2(Homo sapiens (Human))
New York University Abu Dhabi

Curated by ChEMBL
LigandPNGBDBM50500104(CHEMBL3739592)
Affinity DataIC50:  3.80E+4nMAssay Description:Inhibition of human Rce1-mediated CaaX protease activity using ABZ-KSKTKC(farnesyl)QIIM and ABZ-KSKTKC(farnesyl)VIQI as substrate assessed as residua...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCAAX prenyl protease 2(Homo sapiens (Human))
New York University Abu Dhabi

Curated by ChEMBL
LigandPNGBDBM50480672(CHEMBL561185)
Affinity DataIC50:  7.35E+4nMAssay Description:Inhibition of human RCE1More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCAAX prenyl protease 2(Homo sapiens (Human))
New York University Abu Dhabi

Curated by ChEMBL
LigandPNGBDBM50480669(CHEMBL558514)
Affinity DataIC50: >1.98E+5nMAssay Description:Inhibition of human RCE1More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed