Compile Data Set for Download or QSAR
maximum 50k data
Found 13 Enz. Inhib. hit(s) with Target = 'Lysophosphatidic acid receptor 4'
TargetLysophosphatidic acid receptor 4(Mus musculus)
The University Of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50148348((R)-Octadec-9-enoic acid 2-hydroxy-3-phosphonooxy-...)
Affinity DataEC50:  260nMAssay Description:Agonist activity at mouse LPA4 expressed in CHO cells by Fura-2AM dye based Ca2+ mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysophosphatidic acid receptor 4(Homo sapiens (Human))
The University Of Utah

Curated by ChEMBL
LigandPNGBDBM50430006(CHEMBL2335048)
Affinity DataEC50:  3.80nMAssay Description:Agonist activity at human LPA4 receptor transfected in HEK293 cells after 1 hr by TGFalpha shedding assay in presence of Ki16425More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysophosphatidic acid receptor 4(Homo sapiens (Human))
The University Of Utah

Curated by ChEMBL
LigandPNGBDBM50381022(CHEMBL2017139)
Affinity DataEC50:  3.30nMAssay Description:Agonist activity at human LPA4 receptor transfected in HEK293 cells after 1 hr by TGFalpha shedding assay in presence of Ki16425More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysophosphatidic acid receptor 4(Homo sapiens (Human))
The University Of Utah

Curated by ChEMBL
LigandPNGBDBM50430007(CHEMBL2335051)
Affinity DataEC50:  2.40nMAssay Description:Agonist activity at human LPA4 receptor transfected in HEK293 cells after 1 hr by TGFalpha shedding assay in presence of Ki16425More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysophosphatidic acid receptor 4(Homo sapiens (Human))
The University Of Utah

Curated by ChEMBL
LigandPNGBDBM50430008(CHEMBL2335050)
Affinity DataEC50:  4.5nMAssay Description:Agonist activity at human LPA4 receptor transfected in HEK293 cells after 1 hr by TGFalpha shedding assay in presence of Ki16425More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysophosphatidic acid receptor 4(Homo sapiens (Human))
The University Of Utah

Curated by ChEMBL
LigandPNGBDBM50430009(CHEMBL2335049)
Affinity DataEC50:  3.80nMAssay Description:Agonist activity at human LPA4 receptor transfected in HEK293 cells after 1 hr by TGFalpha shedding assay in presence of Ki16425More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysophosphatidic acid receptor 4(Homo sapiens (Human))
The University Of Utah

Curated by ChEMBL
LigandPNGBDBM50233165(CHEMBL1222042)
Affinity DataEC50:  570nMAssay Description:Agonist activity at LPA4 receptor (unknown origin) expressed in CHO cells assessed as increase in intracellular calcium level measured every 3.42 sec...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysophosphatidic acid receptor 4(Homo sapiens (Human))
The University Of Utah

Curated by ChEMBL
LigandPNGBDBM50430010(CHEMBL2335047)
Affinity DataEC50:  3.5nMAssay Description:Agonist activity at human LPA4 receptor transfected in HEK293 cells after 1 hr by TGFalpha shedding assay in presence of Ki16425More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysophosphatidic acid receptor 4(Homo sapiens (Human))
The University Of Utah

Curated by ChEMBL
LigandPNGBDBM50430011(CHEMBL153043)
Affinity DataEC50:  4.90nMAssay Description:Agonist activity at human LPA4 receptor transfected in HEK293 cells after 1 hr by TGFalpha shedding assay in presence of Ki16425More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysophosphatidic acid receptor 4(Homo sapiens (Human))
The University Of Utah

Curated by ChEMBL
LigandPNGBDBM50430012(CHEMBL357053)
Affinity DataEC50:  2.70nMAssay Description:Agonist activity at human LPA4 receptor transfected in HEK293 cells after 1 hr by TGFalpha shedding assay in presence of Ki16425More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysophosphatidic acid receptor 4(Homo sapiens (Human))
The University Of Utah

Curated by ChEMBL
LigandPNGBDBM50430013(CHEMBL364797)
Affinity DataEC50:  84nMAssay Description:Agonist activity at human LPA4 receptor transfected in HEK293 cells after 1 hr by TGFalpha shedding assay in presence of Ki16425More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysophosphatidic acid receptor 4(Homo sapiens (Human))
The University Of Utah

Curated by ChEMBL
LigandPNGBDBM50148348((R)-Octadec-9-enoic acid 2-hydroxy-3-phosphonooxy-...)
Affinity DataEC50:  8.10nMAssay Description:Agonist activity at human LPA4 receptor transfected in HEK293 cells after 1 hr by TGFalpha shedding assay in presence of Ki16425More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysophosphatidic acid receptor 4(Homo sapiens (Human))
The University Of Utah

Curated by ChEMBL
LigandPNGBDBM50430006(CHEMBL2335048)
Affinity DataEC50:  4.90nMAssay Description:Agonist activity at human LPA4 receptor transfected in HEK293 cells after 1 hr by TGFalpha shedding assay in presence of Ki16425More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed