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Found 307 Enz. Inhib. hit(s) with Target = 'MAP kinase-activated protein kinase 5'
TargetMAP kinase-activated protein kinase 5(Homo sapiens (Human))
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50341519((S)-3-(4-(2-(pyrrolidin-1-ylmethyl)pyrrolidin-1-yl...)
Affinity DataKi: >1.00E+3nMAssay Description:Inhibition of PRAKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMAP kinase-activated protein kinase 5(Homo sapiens (Human))
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50224883(7-chloro-3-oxo-8-[(thiazol-5-ylmethyl)-amino]-11,1...)
Affinity DataKi: >1.53E+3nMAssay Description:Inhibition of PRAKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMAP kinase-activated protein kinase 5(Homo sapiens (Human))
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50463484(CHEMBL4248525)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of PRAK (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetMAP kinase-activated protein kinase 5(Homo sapiens (Human))
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50463479(CHEMBL4249925)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of PRAK (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetMAP kinase-activated protein kinase 5 Isoform 2(Homo sapiens (Human))
Xinthera

US Patent
LigandPNGBDBM605909(US11680056, Example 53A | US11680056, Example 53B)
Affinity DataIC50:  0.126nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMAP kinase-activated protein kinase 5 Isoform 2(Homo sapiens (Human))
Xinthera

US Patent
LigandPNGBDBM605939(US11680056, Example 68B)
Affinity DataIC50:  0.200nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMAP kinase-activated protein kinase 5 Isoform 2(Homo sapiens (Human))
Xinthera

US Patent
LigandPNGBDBM605929(US11680056, Example 63B)
Affinity DataIC50:  0.316nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMAP kinase-activated protein kinase 5 Isoform 2(Homo sapiens (Human))
Xinthera

US Patent
LigandPNGBDBM605911(US11680056, Example 54A | US11680056, Example 54B)
Affinity DataIC50:  0.631nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMAP kinase-activated protein kinase 5 Isoform 2(Homo sapiens (Human))
Xinthera

US Patent
LigandPNGBDBM605920(US11680056, Example 59A | US11680056, Example 59B)
Affinity DataIC50:  1nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMAP kinase-activated protein kinase 5 Isoform 2(Homo sapiens (Human))
Xinthera

US Patent
LigandPNGBDBM605918(US11680056, Example 58A)
Affinity DataIC50:  1.26nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMAP kinase-activated protein kinase 5 Isoform 2(Homo sapiens (Human))
Xinthera

US Patent
LigandPNGBDBM605916(US11680056, Example 57A | US11680056, Example 57B)
Affinity DataIC50:  1.26nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMAP kinase-activated protein kinase 5 Isoform 2(Homo sapiens (Human))
Xinthera

US Patent
LigandPNGBDBM605738(US11680056, Example 4 | US11680056, Example 4A | U...)
Affinity DataIC50:  1.58nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMAP kinase-activated protein kinase 5 Isoform 2(Homo sapiens (Human))
Xinthera

US Patent
LigandPNGBDBM605844(US11680056, Example 24A | US11680056, Example 24B)
Affinity DataIC50:  1.58nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMAP kinase-activated protein kinase 5 Isoform 2(Homo sapiens (Human))
Xinthera

US Patent
LigandPNGBDBM605926(US11680056, Example 62A)
Affinity DataIC50:  1.58nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMAP kinase-activated protein kinase 5 Isoform 2(Homo sapiens (Human))
Xinthera

US Patent
LigandPNGBDBM605936(US11680056, Example 67A)
Affinity DataIC50:  1.58nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMAP kinase-activated protein kinase 5 Isoform 2(Homo sapiens (Human))
Xinthera

US Patent
LigandPNGBDBM605914(US11680056, Example 56A | US11680056, Example 56B)
Affinity DataIC50:  2nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMAP kinase-activated protein kinase 5 Isoform 2(Homo sapiens (Human))
Xinthera

US Patent
LigandPNGBDBM605897(US11680056, Example 47A | US11680056, Example 47B)
Affinity DataIC50:  2nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMAP kinase-activated protein kinase 5 Isoform 2(Homo sapiens (Human))
Xinthera

US Patent
LigandPNGBDBM605930(US11680056, Example 64A | US11680056, Example 64B)
Affinity DataIC50:  2nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMAP kinase-activated protein kinase 5 Isoform 2(Homo sapiens (Human))
Xinthera

US Patent
LigandPNGBDBM605842(US11680056, Example 23A | US11680056, Example 23B)
Affinity DataIC50:  3.16nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMAP kinase-activated protein kinase 5 Isoform 2(Homo sapiens (Human))
Xinthera

US Patent
LigandPNGBDBM605838(US11680056, Example 21A | US11680056, Example 21B)
Affinity DataIC50:  3.16nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMAP kinase-activated protein kinase 5 Isoform 2(Homo sapiens (Human))
Xinthera

US Patent
LigandPNGBDBM605924(US11680056, Example 61A | US11680056, Example 61B)
Affinity DataIC50:  3.16nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMAP kinase-activated protein kinase 5 Isoform 2(Homo sapiens (Human))
Xinthera

US Patent
LigandPNGBDBM605932(US11680056, Example 65A | US11680056, Example 65B)
Affinity DataIC50:  3.98nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMAP kinase-activated protein kinase 5 Isoform 2(Homo sapiens (Human))
Xinthera

US Patent
LigandPNGBDBM605824(US11680056, Example 9A)
Affinity DataIC50:  3.98nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMAP kinase-activated protein kinase 5 Isoform 2(Homo sapiens (Human))
Xinthera

US Patent
LigandPNGBDBM605873(US11680056, Example 36A)
Affinity DataIC50:  5.01nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMAP kinase-activated protein kinase 5 Isoform 2(Homo sapiens (Human))
Xinthera

US Patent
LigandPNGBDBM605899(US11680056, Example 48A | US11680056, Example 48B)
Affinity DataIC50:  5.01nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMAP kinase-activated protein kinase 5 Isoform 2(Homo sapiens (Human))
Xinthera

US Patent
LigandPNGBDBM605817(US11680056, Example 6 | US11680056, Example 6A | U...)
Affinity DataIC50:  5.01nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMAP kinase-activated protein kinase 5 Isoform 2(Homo sapiens (Human))
Xinthera

US Patent
LigandPNGBDBM605885(US11680056, Example 41A)
Affinity DataIC50:  5.01nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMAP kinase-activated protein kinase 5 Isoform 2(Homo sapiens (Human))
Xinthera

US Patent
LigandPNGBDBM605877(US11680056, Example 37A | US11680056, Example 37B)
Affinity DataIC50:  5.01nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMAP kinase-activated protein kinase 5 Isoform 2(Homo sapiens (Human))
Xinthera

US Patent
LigandPNGBDBM605901(US11680056, Example 49A | US11680056, Example 49B)
Affinity DataIC50:  6.31nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMAP kinase-activated protein kinase 5 Isoform 2(Homo sapiens (Human))
Xinthera

US Patent
LigandPNGBDBM605874(US11680056, Example 36B)
Affinity DataIC50:  6.31nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMAP kinase-activated protein kinase 5 Isoform 2(Homo sapiens (Human))
Xinthera

US Patent
LigandPNGBDBM605935(US11680056, Example 66B)
Affinity DataIC50:  6.31nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMAP kinase-activated protein kinase 5 Isoform 2(Homo sapiens (Human))
Xinthera

US Patent
LigandPNGBDBM605854(US11680056, Example 29A | US11680056, Example 29B)
Affinity DataIC50:  7.94nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMAP kinase-activated protein kinase 5 Isoform 2(Homo sapiens (Human))
Xinthera

US Patent
LigandPNGBDBM605881(US11680056, Example 39A | US11680056, Example 39B)
Affinity DataIC50:  10nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMAP kinase-activated protein kinase 5 Isoform 2(Homo sapiens (Human))
Xinthera

US Patent
LigandPNGBDBM605732(US11680056, Example 3 | US11680056, Example 3A | U...)
Affinity DataIC50:  10nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMAP kinase-activated protein kinase 5 Isoform 2(Homo sapiens (Human))
Xinthera

US Patent
LigandPNGBDBM605916(US11680056, Example 57A | US11680056, Example 57B)
Affinity DataIC50: >10nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMAP kinase-activated protein kinase 5 Isoform 2(Homo sapiens (Human))
Xinthera

US Patent
LigandPNGBDBM605903(US11680056, Example 50A | US11680056, Example 50B)
Affinity DataIC50:  12.6nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMAP kinase-activated protein kinase 5 Isoform 2(Homo sapiens (Human))
Xinthera

US Patent
LigandPNGBDBM605848(US11680056, Example 26A | US11680056, Example 26B)
Affinity DataIC50:  12.6nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMAP kinase-activated protein kinase 5 Isoform 2(Homo sapiens (Human))
Xinthera

US Patent
LigandPNGBDBM605889(US11680056, Example 43A | US11680056, Example 43B)
Affinity DataIC50:  12.6nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMAP kinase-activated protein kinase 5 Isoform 2(Homo sapiens (Human))
Xinthera

US Patent
LigandPNGBDBM605869(US11680056, Example 35A | US11680056, Example 35B ...)
Affinity DataIC50:  15.8nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMAP kinase-activated protein kinase 5 Isoform 2(Homo sapiens (Human))
Xinthera

US Patent
LigandPNGBDBM605907(US11680056, Example 52A | US11680056, Example 52B)
Affinity DataIC50:  15.8nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMAP kinase-activated protein kinase 5 Isoform 2(Homo sapiens (Human))
Xinthera

US Patent
LigandPNGBDBM605895(US11680056, Example 46A | US11680056, Example 46B)
Affinity DataIC50:  15.8nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMAP kinase-activated protein kinase 5 Isoform 2(Homo sapiens (Human))
Xinthera

US Patent
LigandPNGBDBM605859(US11680056, Example 32A | US11680056, Example 32B ...)
Affinity DataIC50:  20nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMAP kinase-activated protein kinase 5 Isoform 2(Homo sapiens (Human))
Xinthera

US Patent
LigandPNGBDBM605865(US11680056, Example 34A)
Affinity DataIC50:  20nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMAP kinase-activated protein kinase 5 Isoform 2(Homo sapiens (Human))
Xinthera

US Patent
LigandPNGBDBM605923(US11680056, Example 60B)
Affinity DataIC50:  25.1nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMAP kinase-activated protein kinase 5 Isoform 2(Homo sapiens (Human))
Xinthera

US Patent
LigandPNGBDBM605863(US11680056, Example 33A | US11680056, Example 33B)
Affinity DataIC50:  25.1nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMAP kinase-activated protein kinase 5 Isoform 2(Homo sapiens (Human))
Xinthera

US Patent
LigandPNGBDBM605891(US11680056, Example 44A | US11680056, Example 44B)
Affinity DataIC50:  25.1nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMAP kinase-activated protein kinase 5 Isoform 2(Homo sapiens (Human))
Xinthera

US Patent
LigandPNGBDBM605869(US11680056, Example 35A | US11680056, Example 35B ...)
Affinity DataIC50:  50.1nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMAP kinase-activated protein kinase 5 Isoform 2(Homo sapiens (Human))
Xinthera

US Patent
LigandPNGBDBM605913(US11680056, Example 55)
Affinity DataIC50:  63.1nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMAP kinase-activated protein kinase 5 Isoform 2(Homo sapiens (Human))
Xinthera

US Patent
LigandPNGBDBM605905(US11680056, Example 51A)
Affinity DataIC50:  79.4nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMAP kinase-activated protein kinase 5 Isoform 2(Homo sapiens (Human))
Xinthera

US Patent
LigandPNGBDBM605937(US11680056, Example 67B)
Affinity DataIC50:  79.4nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
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