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Found 8 Enz. Inhib. hit(s) with Target = 'Mast cell carboxypeptidase A'
TargetMast cell carboxypeptidase A(Rattus norvegicus)
Universitat Aut£Noma De Barcelona

Curated by ChEMBL
LigandPNGBDBM50530230(CHEMBL4445882)
Affinity DataKi:  0.0170nMAssay Description:Inhibition of rat CPA3 using AAFP as substrate preincubated for 45 mins measured at 30 sec intervals for 15 mins by UV/vis-spectrophotometryMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetMast cell carboxypeptidase A(Rattus norvegicus)
Universitat Aut£Noma De Barcelona

Curated by ChEMBL
LigandPNGBDBM50530230(CHEMBL4445882)
Affinity DataKi:  0.0170nMAssay Description:Inhibition of rat CPA3 using AAFP as substrate preincubated for 45 mins measured at 30 sec intervals for 15 mins by UV/vis-spectrophotometryMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetMast cell carboxypeptidase A(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50281176((S)-2-Mercaptomethyl-3-phenyl-propionic acid | 2-T...)
Affinity DataKi:  7.80nMAssay Description:Compound was tested for inhibitory activity against carboxypeptidase AMore data for this Ligand-Target Pair
In DepthDetails Article
TargetMast cell carboxypeptidase A(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50121929((phenylmethyl)butanedioic acid | 2-benzylbutanedio...)
Affinity DataKi:  450nMAssay Description:The compound was evaluated for the inhibition of Carboxypeptidase AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMast cell carboxypeptidase A(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50121917(2-Benzyl-pentanedioic acid | CHEMBL153232)
Affinity DataKi:  5.00E+3nMAssay Description:The compound was evaluated for the inhibition of Carboxypeptidase AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMast cell carboxypeptidase A(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50058391((S)-1-[(S)-2-(4-Methoxy-benzoylamino)-3-methyl-but...)
Affinity DataKi:  1.70E+4nMAssay Description:Binding affinity of the compound for carboxypeptidase AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMast cell carboxypeptidase A(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50473781(Succinic acid monobenzyl ester)
Affinity DataKd:  447nMAssay Description:Binding affinity against Carboxypeptidase AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMast cell carboxypeptidase A(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50188513((S)-6-Amino-2-(2-amino-acetylamino)-hexanoic acid ...)
Affinity DataKd:  1.29E+5nMAssay Description:Binding affinity against Carboxypeptidase AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed