TargetMast cell carboxypeptidase A(Rattus norvegicus)
Universitat Aut£Noma De Barcelona
Curated by ChEMBL
Universitat Aut£Noma De Barcelona
Curated by ChEMBL
Affinity DataKi: 0.0170nMAssay Description:Inhibition of rat CPA3 using AAFP as substrate preincubated for 45 mins measured at 30 sec intervals for 15 mins by UV/vis-spectrophotometryMore data for this Ligand-Target Pair
TargetMast cell carboxypeptidase A(Rattus norvegicus)
Universitat Aut£Noma De Barcelona
Curated by ChEMBL
Universitat Aut£Noma De Barcelona
Curated by ChEMBL
Affinity DataKi: 0.0170nMAssay Description:Inhibition of rat CPA3 using AAFP as substrate preincubated for 45 mins measured at 30 sec intervals for 15 mins by UV/vis-spectrophotometryMore data for this Ligand-Target Pair
Affinity DataKi: 7.80nMAssay Description:Compound was tested for inhibitory activity against carboxypeptidase AMore data for this Ligand-Target Pair
Affinity DataKi: 450nMAssay Description:The compound was evaluated for the inhibition of Carboxypeptidase AMore data for this Ligand-Target Pair
Affinity DataKi: 5.00E+3nMAssay Description:The compound was evaluated for the inhibition of Carboxypeptidase AMore data for this Ligand-Target Pair
Affinity DataKi: 1.70E+4nMAssay Description:Binding affinity of the compound for carboxypeptidase AMore data for this Ligand-Target Pair
Affinity DataKd: 447nMAssay Description:Binding affinity against Carboxypeptidase AMore data for this Ligand-Target Pair
Affinity DataKd: 1.29E+5nMAssay Description:Binding affinity against Carboxypeptidase AMore data for this Ligand-Target Pair