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Found 3 Enz. Inhib. hit(s) with Target = 'Mitogen-activated protein kinase kinase kinase 21'
TargetMitogen-activated protein kinase kinase kinase 21(Homo sapiens)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM2579((2S,3R,4R,6R)-3-methoxy-2-methyl-4-(methylamino)-2...)
Affinity DataIC50:  765nMAssay Description:Inhibition of human MLK4 using MEK1 as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 21(Homo sapiens)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM2579((2S,3R,4R,6R)-3-methoxy-2-methyl-4-(methylamino)-2...)
Affinity DataIC50:  1.47E+3nMAssay Description:Inhibition of human MLK4 using MEK1 as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 21(Homo sapiens)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50242512(CHEMBL4098682)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of MLK4 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed