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Found 35 Enz. Inhib. hit(s) with Target = 'Transcription factor 7-like 2'
TargetTranscription factor 7-like 2(Homo sapiens (Human))
University Of Utah

Curated by ChEMBL
LigandPNGBDBM50014098(CHEMBL3260852)
Affinity DataKi:  1.35E+3nMAssay Description:Inhibition of beta-catenin/T cell factor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscription factor 7-like 2(Homo sapiens (Human))
University Of Utah

Curated by ChEMBL
LigandPNGBDBM50014132(CHEMBL2323032)
Affinity DataKi:  3.10E+3nMAssay Description:Inhibition of human beta-casein/Tcf4 interaction after 1 hr by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscription factor 7-like 2(Homo sapiens (Human))
University Of Utah

Curated by ChEMBL
LigandPNGBDBM32102(1,6-dimethylpyrimido[5,4-e][1,2,4]triazine-5,7(1H,...)
Affinity DataKi:  3.70E+3nMAssay Description:Inhibition of human beta-casein/Tcf4 interaction after 1 hr by alphascreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscription factor 7-like 2(Homo sapiens (Human))
University Of Utah

Curated by ChEMBL
LigandPNGBDBM50014132(CHEMBL2323032)
Affinity DataKi:  3.80E+3nMAssay Description:Inhibition of human beta-casein/Tcf4 interaction after 1 hr by alphascreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscription factor 7-like 2(Homo sapiens (Human))
University Of Utah

Curated by ChEMBL
LigandPNGBDBM32102(1,6-dimethylpyrimido[5,4-e][1,2,4]triazine-5,7(1H,...)
Affinity DataKi:  5.80E+3nMAssay Description:Inhibition of human beta-casein/Tcf4 interaction after 1 hr by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscription factor 7-like 2(Homo sapiens (Human))
University Of Utah

Curated by ChEMBL
LigandPNGBDBM50094484(CHEBI:3556 | CHEMBL2323033 | US9284299, CGP049090 ...)
Affinity DataKi:  5.90E+3nMAssay Description:Inhibition of human beta-casein/Tcf4 interaction after 1 hr by alphascreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscription factor 7-like 2(Homo sapiens (Human))
University Of Utah

Curated by ChEMBL
LigandPNGBDBM50094600(CHEMBL2323029)
Affinity DataKi:  8.80E+3nMAssay Description:Inhibition of human beta-casein/Tcf4 interaction after 1 hr by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscription factor 7-like 2(Homo sapiens (Human))
University Of Utah

Curated by ChEMBL
LigandPNGBDBM50094600(CHEMBL2323029)
Affinity DataKi:  1.30E+4nMAssay Description:Inhibition of human beta-casein/Tcf4 interaction after 1 hr by alphascreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscription factor 7-like 2(Homo sapiens (Human))
University Of Utah

Curated by ChEMBL
LigandPNGBDBM50489463(CHEMBL2323031)
Affinity DataKi:  1.60E+4nMAssay Description:Inhibition of human beta-casein/Tcf4 interaction after 1 hr by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscription factor 7-like 2(Homo sapiens (Human))
University Of Utah

Curated by ChEMBL
LigandPNGBDBM50249236((R)-1-(4,9-dihydroxy-12-((R)-2-((4-hydroxyphenoxy)...)
Affinity DataKi:  1.80E+4nMAssay Description:Inhibition of human beta-casein/Tcf4 interaction after 1 hr by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscription factor 7-like 2(Homo sapiens (Human))
University Of Utah

Curated by ChEMBL
LigandPNGBDBM50489463(CHEMBL2323031)
Affinity DataKi:  2.10E+4nMAssay Description:Inhibition of human beta-casein/Tcf4 interaction after 1 hr by alphascreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscription factor 7-like 2(Homo sapiens (Human))
University Of Utah

Curated by ChEMBL
LigandPNGBDBM50094597(CHEMBL2323028)
Affinity DataKi:  2.10E+4nMAssay Description:Inhibition of human beta-casein/Tcf4 interaction after 1 hr by alphascreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscription factor 7-like 2(Homo sapiens (Human))
University Of Utah

Curated by ChEMBL
LigandPNGBDBM50489464(CHEMBL2323030)
Affinity DataKi:  2.90E+4nMAssay Description:Inhibition of human beta-casein/Tcf4 interaction after 1 hr by alphascreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscription factor 7-like 2(Homo sapiens (Human))
University Of Utah

Curated by ChEMBL
LigandPNGBDBM50094484(CHEBI:3556 | CHEMBL2323033 | US9284299, CGP049090 ...)
Affinity DataKi:  3.60E+4nMAssay Description:Inhibition of human beta-casein/Tcf4 interaction after 1 hr by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscription factor 7-like 2(Homo sapiens (Human))
University Of Utah

Curated by ChEMBL
LigandPNGBDBM50094597(CHEMBL2323028)
Affinity DataKi:  7.70E+4nMAssay Description:Inhibition of human beta-casein/Tcf4 interaction after 1 hr by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscription factor 7-like 2(Homo sapiens (Human))
University Of Utah

Curated by ChEMBL
LigandPNGBDBM50484962(CHEMBL2018626)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of beta-casein/TCF4 pathway expressed in HCT116 cells containing delta45S mutant after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTranscription factor 7-like 2(Homo sapiens (Human))
University Of Utah

Curated by ChEMBL
LigandPNGBDBM50484965(CHEMBL2018615)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibition of beta-casein/TCF4 pathway expressed in HCT116 cells containing delta45S mutant after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTranscription factor 7-like 2(Homo sapiens (Human))
University Of Utah

Curated by ChEMBL
LigandPNGBDBM50484959(CHEMBL2018726)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibition of beta-casein/TCF4 pathway expressed in HCT116 cells containing delta45S mutant after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTranscription factor 7-like 2(Homo sapiens (Human))
University Of Utah

Curated by ChEMBL
LigandPNGBDBM50484954(CHEMBL2018623)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of beta-casein/TCF4 pathway expressed in HCT116 cells containing delta45S mutant after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTranscription factor 7-like 2(Homo sapiens (Human))
University Of Utah

Curated by ChEMBL
LigandPNGBDBM50484955(CHEMBL2018727)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of beta-casein/TCF4 pathway expressed in HCT116 cells containing delta45S mutant after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTranscription factor 7-like 2(Homo sapiens (Human))
University Of Utah

Curated by ChEMBL
LigandPNGBDBM50484951(CHEMBL2018597)
Affinity DataIC50:  2.50E+3nMAssay Description:Inhibition of beta-casein/TCF4 pathway expressed in HCT116 cells containing delta45S mutant after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTranscription factor 7-like 2(Homo sapiens (Human))
University Of Utah

Curated by ChEMBL
LigandPNGBDBM50484952(CHEMBL2018621)
Affinity DataIC50:  2.50E+3nMAssay Description:Inhibition of beta-casein/TCF4 pathway expressed in HCT116 cells containing delta45S mutant after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTranscription factor 7-like 2(Homo sapiens (Human))
University Of Utah

Curated by ChEMBL
LigandPNGBDBM50484953(CHEMBL2018622)
Affinity DataIC50:  2.50E+3nMAssay Description:Inhibition of beta-casein/TCF4 pathway expressed in HCT116 cells containing delta45S mutant after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTranscription factor 7-like 2(Homo sapiens (Human))
University Of Utah

Curated by ChEMBL
LigandPNGBDBM50484958(CHEMBL2018734)
Affinity DataIC50:  2.50E+3nMAssay Description:Inhibition of beta-casein/TCF4 pathway expressed in HCT116 cells containing delta45S mutant after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTranscription factor 7-like 2(Homo sapiens (Human))
University Of Utah

Curated by ChEMBL
LigandPNGBDBM50484949(CHEMBL2018614)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of beta-casein/TCF4 pathway expressed in HCT116 cells containing delta45S mutant after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTranscription factor 7-like 2(Homo sapiens (Human))
University Of Utah

Curated by ChEMBL
LigandPNGBDBM50484961(CHEMBL2018598)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of beta-casein/TCF4 pathway expressed in HCT116 cells containing delta45S mutant after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTranscription factor 7-like 2(Homo sapiens (Human))
University Of Utah

Curated by ChEMBL
LigandPNGBDBM50484967(CHEMBL2018733)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of beta-casein/TCF4 pathway expressed in HCT116 cells containing delta45S mutant after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTranscription factor 7-like 2(Homo sapiens (Human))
University Of Utah

Curated by ChEMBL
LigandPNGBDBM50484966(CHEMBL2018617)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of beta-casein/TCF4 pathway expressed in HCT116 cells containing delta45S mutant after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTranscription factor 7-like 2(Homo sapiens (Human))
University Of Utah

Curated by ChEMBL
LigandPNGBDBM50484957(CHEMBL2018732)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of beta-casein/TCF4 pathway expressed in HCT116 cells containing delta45S mutant after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTranscription factor 7-like 2(Homo sapiens (Human))
University Of Utah

Curated by ChEMBL
LigandPNGBDBM50484956(CHEMBL2018728)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of beta-casein/TCF4 pathway expressed in HCT116 cells containing delta45S mutant after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTranscription factor 7-like 2(Homo sapiens (Human))
University Of Utah

Curated by ChEMBL
LigandPNGBDBM50484963(CHEMBL2018729)
Affinity DataIC50:  3.50E+3nMAssay Description:Inhibition of beta-casein/TCF4 pathway expressed in HCT116 cells containing delta45S mutant after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTranscription factor 7-like 2(Homo sapiens (Human))
University Of Utah

Curated by ChEMBL
LigandPNGBDBM50484950(CHEMBL569102)
Affinity DataIC50:  3.50E+3nMAssay Description:Inhibition of beta-casein/TCF4 pathway expressed in HCT116 cells containing delta45S mutant after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTranscription factor 7-like 2(Homo sapiens (Human))
University Of Utah

Curated by ChEMBL
LigandPNGBDBM50484948(CHEMBL2018612)
Affinity DataIC50:  3.50E+3nMAssay Description:Inhibition of beta-casein/TCF4 pathway expressed in HCT116 cells containing delta45S mutant after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTranscription factor 7-like 2(Homo sapiens (Human))
University Of Utah

Curated by ChEMBL
LigandPNGBDBM50484960(CHEMBL2018618)
Affinity DataIC50: >5.00E+3nMAssay Description:Inhibition of beta-casein/TCF4 pathway expressed in HCT116 cells containing delta45S mutant after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTranscription factor 7-like 2(Homo sapiens (Human))
University Of Utah

Curated by ChEMBL
LigandPNGBDBM50484964(CHEMBL2018735)
Affinity DataIC50: >5.00E+3nMAssay Description:Inhibition of beta-casein/TCF4 pathway expressed in HCT116 cells containing delta45S mutant after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed