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Found 6 Enz. Inhib. hit(s) with Target = 'Transcription factor HES-1'
TargetTranscription factor HES-1(Mus musculus)
Chiba University

Curated by ChEMBL
LigandPNGBDBM50378454(LINDBLADIONE)
Affinity DataIC50:  4.10E+3nMAssay Description:Inhibition of Cy3-labeled mouse recombinant Hes1 (3-281) dimer formation expressed in Escherichia coli by microplate-based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTranscription factor HES-1(Mus musculus)
Chiba University

Curated by ChEMBL
LigandPNGBDBM50378456(LYCOGALIC ACID A | LYCOGARIC ACID A)
Affinity DataIC50:  6.00E+3nMAssay Description:Inhibition of Cy3-labeled mouse recombinant Hes1 (3-281) dimer formation expressed in Escherichia coli by microplate-based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscription factor HES-1(Mus musculus)
Chiba University

Curated by ChEMBL
LigandPNGBDBM50378457(CHEMBL572017)
Affinity DataIC50:  7.80E+3nMAssay Description:Inhibition of Cy3-labeled mouse recombinant Hes1 (3-281) dimer formation expressed in Escherichia coli by microplate-based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscription factor HES-1(Mus musculus)
Chiba University

Curated by ChEMBL
LigandPNGBDBM50378459(NUDIPOSIDE)
Affinity DataIC50:  9.60E+3nMAssay Description:Inhibition of Cy3-labeled mouse recombinant Hes1 (3-281) dimer formation expressed in Escherichia coli by microplate-based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscription factor HES-1(Mus musculus)
Chiba University

Curated by ChEMBL
LigandPNGBDBM50378455(LYCOGARUBIN B)
Affinity DataIC50:  1.65E+4nMAssay Description:Inhibition of Cy3-labeled mouse recombinant Hes1 (3-281) dimer formation expressed in Escherichia coli by microplate-based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscription factor HES-1(Mus musculus)
Chiba University

Curated by ChEMBL
LigandPNGBDBM50378458(LYONISIDE)
Affinity DataIC50:  4.81E+4nMAssay Description:Inhibition of Cy3-labeled mouse recombinant Hes1 (3-281) dimer formation expressed in Escherichia coli by microplate-based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed