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Found 13 Enz. Inhib. hit(s) with Target = 'Potassium voltage-gated channel subfamily KQT member 5'
TargetPotassium voltage-gated channel subfamily KQT member 5(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50426567(BMS-204352 | FLINDOKALNER | MaxiPost)
Affinity DataEC50:  2.40E+3nMAssay Description:Positive modulatory activity at voltage-gated K channel 7.5 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily KQT member 5(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50521286(CHEMBL4450214)
Affinity DataEC50:  2.43E+3nMAssay Description:Agonist activity at human KCNQ5 expressed in CHOK1 cells by whole cell patch clamp assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily KQT member 5(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50521289(CHEMBL4588394)
Affinity DataEC50:  1.68E+3nMAssay Description:Agonist activity at human KCNQ5 expressed in CHOK1 cells by whole cell patch clamp assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily KQT member 5(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50143558(CHEMBL41355 | EZOGABINE | N-(2-amino-4-(4-fluorobe...)
Affinity DataEC50:  3.45E+3nMAssay Description:Agonist activity at human KCNQ5 expressed in CHOK1 cells by whole cell patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetPotassium voltage-gated channel subfamily KQT member 5(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50521288(CHEMBL4438770)
Affinity DataEC50:  1.37E+3nMAssay Description:Agonist activity at human KCNQ5 expressed in CHOK1 cells by whole cell patch clamp assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily KQT member 5(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50526876(CHEMBL4457044)
Affinity DataEC50:  350nMAssay Description:Activation of human Kv7.5 expressed in CHO cells assessed as increase in channel current amplitude by whole cell patch clamp electrophysiology assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily KQT member 5(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50594442(CHEMBL5178988)
Affinity DataEC50:  4.50E+3nMAssay Description:Agonist activity at human KCNQ5 channel expressed in CHO cells assessed as increase in outward current by patch clamp electrophysiology methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPotassium voltage-gated channel subfamily KQT member 5(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50143558(CHEMBL41355 | EZOGABINE | N-(2-amino-4-(4-fluorobe...)
Affinity DataEC50:  800nMAssay Description:Activation of human Kv7.5 expressed in CHO cells assessed as increase in channel current amplitude by whole cell patch clamp electrophysiology assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetPotassium voltage-gated channel subfamily KQT member 5(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50592355(CHEMBL5200636)
Affinity DataEC50:  3.78E+3nMAssay Description:Agonist activity at Kv7.5 (unknown origin) expressed in CHO cells co-expressing GFPMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPotassium voltage-gated channel subfamily KQT member 5(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50592356(CHEMBL4458793)
Affinity DataEC50:  3.78E+3nMAssay Description:Agonist activity at Kv7.5 (unknown origin) expressed in CHO cells co-expressing GFPMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPotassium voltage-gated channel subfamily KQT member 5(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50592357(CHEMBL5185685)
Affinity DataEC50:  1.06E+3nMAssay Description:Agonist activity at Kv7.5 (unknown origin) expressed in CHO cells co-expressing GFPMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPotassium voltage-gated channel subfamily KQT member 5(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50592360(CHEMBL4549229)
Affinity DataEC50:  540nMAssay Description:Agonist activity at Kv7.5 (unknown origin) expressed in CHO cells co-expressing GFPMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPotassium voltage-gated channel subfamily KQT member 5(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50526877(CHEMBL4545892)
Affinity DataEC50:  1.07E+3nMAssay Description:Activation of human Kv7.5 expressed in CHO cells assessed as increase in channel current amplitude by whole cell patch clamp electrophysiology assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed