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Found 16 Enz. Inhib. hit(s) with Target = 'Protein phosphatase methylesterase 1'
TargetProtein phosphatase methylesterase 1(Homo sapiens (Human))
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM75707((3R)-3-cyclopentyl-4-keto-3-phenyl-diazetidine-1,2...)
Affinity DataIC50:  10nMAssay Description:Inhibition of PME1 binding to FP-rhodamine in human MDA-MB-231 cells after 30 mins by fluorescence polarization activity-based protein profiling assa...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein phosphatase methylesterase 1(Homo sapiens (Human))
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM75707((3R)-3-cyclopentyl-4-keto-3-phenyl-diazetidine-1,2...)
Affinity DataIC50:  10nMAssay Description:Source (MLPCN Center Name): The Scripps Research Institute Molecular Screening Center (SRIMSC) Center Affiliation: The Scripps Research Institute (TS...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetProtein phosphatase methylesterase 1(Homo sapiens (Human))
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50400986(CHEMBL1550905)
Affinity DataIC50:  600nMAssay Description:Inhibition of PME1 binding to FP-rhodamine in human HEK293T cells after 45 mins by fluorescence polarization activity-based protein profiling assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein phosphatase methylesterase 1(Mus musculus)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50400986(CHEMBL1550905)
Affinity DataIC50:  600nMAssay Description:Inhibition of PME1 binding to FP-rhodamine in mouse brain soluble proteome after 45 mins by fluorescence polarization activity-based protein profilin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein phosphatase methylesterase 1(Mus musculus)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50400987(CHEMBL1316687)
Affinity DataIC50:  640nMAssay Description:Inhibition of PME1 binding to FP-rhodamine in mouse brain soluble proteome after 45 mins by fluorescence polarization activity-based protein profilin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein phosphatase methylesterase 1(Mus musculus)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50400996(CHEMBL1699083)
Affinity DataIC50:  2.50E+3nMAssay Description:Inhibition of PME1 binding to FP-rhodamine in mouse brain soluble proteome after 45 mins by fluorescence polarization activity-based protein profilin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein phosphatase methylesterase 1(Mus musculus)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50400994(CHEMBL1719837)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of PME1 binding to FP-rhodamine in mouse brain soluble proteome after 45 mins by fluorescence polarization activity-based protein profilin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein phosphatase methylesterase 1(Mus musculus)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50400995(CHEMBL1706554)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of PME1 binding to FP-rhodamine in mouse brain soluble proteome after 45 mins by fluorescence polarization activity-based protein profilin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein phosphatase methylesterase 1(Mus musculus)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50400988(CHEMBL1701914)
Affinity DataIC50:  3.40E+3nMAssay Description:Inhibition of PME1 binding to FP-rhodamine in mouse brain soluble proteome after 45 mins by fluorescence polarization activity-based protein profilin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein phosphatase methylesterase 1(Homo sapiens (Human))
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50400986(CHEMBL1550905)
Affinity DataIC50:  3.50E+3nMAssay Description:Inhibition of PME1 binding to FP-rhodamine in HEK293T cells after 1 hr by fluorescence polarization activity-based protein profiling assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein phosphatase methylesterase 1(Mus musculus)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50400993(CHEMBL1729870)
Affinity DataIC50:  4.00E+3nMAssay Description:Inhibition of PME1 binding to FP-rhodamine in mouse brain soluble proteome after 45 mins by fluorescence polarization activity-based protein profilin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein phosphatase methylesterase 1(Mus musculus)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50400989(CHEMBL1718102)
Affinity DataIC50:  4.80E+3nMAssay Description:Inhibition of PME1 binding to FP-rhodamine in mouse brain soluble proteome after 45 mins by fluorescence polarization activity-based protein profilin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein phosphatase methylesterase 1(Mus musculus)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50400991(CHEMBL1711185)
Affinity DataIC50:  6.80E+3nMAssay Description:Inhibition of PME1 binding to FP-rhodamine in mouse brain soluble proteome after 45 mins by fluorescence polarization activity-based protein profilin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein phosphatase methylesterase 1(Homo sapiens (Human))
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50400997(CHEMBL1521288)
Affinity DataIC50:  1.08E+4nMAssay Description:Inhibition of PME1 binding to FP-rhodamine in human MDA-MB-231 cells after 30 mins by fluorescence polarization activity-based protein profiling assa...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein phosphatase methylesterase 1(Mus musculus)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50400990(CHEMBL1723004)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of PME1 binding to FP-rhodamine in mouse brain soluble proteome after 45 mins by fluorescence polarization activity-based protein profilin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein phosphatase methylesterase 1(Mus musculus)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50400992(CHEMBL1701983)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of PME1 binding to FP-rhodamine in mouse brain soluble proteome after 45 mins by fluorescence polarization activity-based protein profilin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed