TargetCasein kinase I isoform alpha-like(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataIC50: 1.27E+3nMAssay Description:Inhibition of human CK1a1L using KRRRAL[pS]VASLPGL as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
TargetCasein kinase I isoform alpha-like(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataIC50: 2.41E+3nMAssay Description:Inhibition of human CK1a1L using KRRRAL[pS]VASLPGL as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
TargetCasein kinase I isoform alpha-like(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: 1.00E+3nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
TargetCasein kinase I isoform alpha-like(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: 1.50E+3nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
TargetCasein kinase I isoform alpha-like(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: 250nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
TargetCasein kinase I isoform alpha-like(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: 550nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
TargetCasein kinase I isoform alpha-like(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for CSNK1A1L kinase domainMore data for this Ligand-Target Pair
TargetCasein kinase I isoform alpha-like(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for CSNK1A1L kinase domainMore data for this Ligand-Target Pair
TargetCasein kinase I isoform alpha-like(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: 7.10E+3nMAssay Description:Binding constant for CSNK1A1L kinase domainMore data for this Ligand-Target Pair
TargetCasein kinase I isoform alpha-like(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: 250nMAssay Description:Binding constant for CSNK1A1L kinase domainMore data for this Ligand-Target Pair
TargetCasein kinase I isoform alpha-like(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for full-length CSNK1A1LMore data for this Ligand-Target Pair
TargetCasein kinase I isoform alpha-like(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: 250nMAssay Description:Binding constant for full-length CSNK1A1LMore data for this Ligand-Target Pair
TargetCasein kinase I isoform alpha-like(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: 2.40E+3nMAssay Description:Binding constant for CSNK1A1L kinase domainMore data for this Ligand-Target Pair
TargetCasein kinase I isoform alpha-like(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for CSNK1A1L kinase domainMore data for this Ligand-Target Pair
TargetCasein kinase I isoform alpha-like(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for CSNK1A1L kinase domainMore data for this Ligand-Target Pair
TargetCasein kinase I isoform alpha-like(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: 1.50E+3nMAssay Description:Binding constant for CSNK1A1L kinase domainMore data for this Ligand-Target Pair
TargetCasein kinase I isoform alpha-like(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for CSNK1A1L kinase domainMore data for this Ligand-Target Pair
TargetCasein kinase I isoform alpha-like(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for CSNK1A1L kinase domainMore data for this Ligand-Target Pair
TargetCasein kinase I isoform alpha-like(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for CSNK1A1L kinase domainMore data for this Ligand-Target Pair
TargetCasein kinase I isoform alpha-like(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for CSNK1A1L kinase domainMore data for this Ligand-Target Pair
TargetCasein kinase I isoform alpha-like(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for CSNK1A1L kinase domainMore data for this Ligand-Target Pair
TargetCasein kinase I isoform alpha-like(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for CSNK1A1L kinase domainMore data for this Ligand-Target Pair
TargetCasein kinase I isoform alpha-like(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for CSNK1A1L kinase domainMore data for this Ligand-Target Pair
TargetCasein kinase I isoform alpha-like(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for CSNK1A1L kinase domainMore data for this Ligand-Target Pair
TargetCasein kinase I isoform alpha-like(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for CSNK1A1L kinase domainMore data for this Ligand-Target Pair
TargetCasein kinase I isoform alpha-like(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for CSNK1A1L kinase domainMore data for this Ligand-Target Pair
TargetCasein kinase I isoform alpha-like(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for CSNK1A1L kinase domainMore data for this Ligand-Target Pair
TargetCasein kinase I isoform alpha-like(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: 2.00E+3nMAssay Description:Binding constant for CSNK1A1L kinase domainMore data for this Ligand-Target Pair
TargetCasein kinase I isoform alpha-like(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for CSNK1A1L kinase domainMore data for this Ligand-Target Pair
TargetCasein kinase I isoform alpha-like(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for CSNK1A1L kinase domainMore data for this Ligand-Target Pair
TargetCasein kinase I isoform alpha-like(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for CSNK1A1L kinase domainMore data for this Ligand-Target Pair
TargetCasein kinase I isoform alpha-like(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for CSNK1A1L kinase domainMore data for this Ligand-Target Pair
TargetCasein kinase I isoform alpha-like(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for CSNK1A1L kinase domainMore data for this Ligand-Target Pair
TargetCasein kinase I isoform alpha-like(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for CSNK1A1L kinase domainMore data for this Ligand-Target Pair
TargetCasein kinase I isoform alpha-like(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for CSNK1A1L kinase domainMore data for this Ligand-Target Pair
TargetCasein kinase I isoform alpha-like(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for CSNK1A1L kinase domainMore data for this Ligand-Target Pair
TargetCasein kinase I isoform alpha-like(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for CSNK1A1L kinase domainMore data for this Ligand-Target Pair
TargetCasein kinase I isoform alpha-like(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: 1.90E+3nMAssay Description:Binding constant for CSNK1A1L kinase domainMore data for this Ligand-Target Pair
TargetCasein kinase I isoform alpha-like(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for CSNK1A1L kinase domainMore data for this Ligand-Target Pair
TargetCasein kinase I isoform alpha-like(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for CSNK1A1L kinase domainMore data for this Ligand-Target Pair
TargetCasein kinase I isoform alpha-like(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for CSNK1A1L kinase domainMore data for this Ligand-Target Pair
TargetCasein kinase I isoform alpha-like(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for CSNK1A1L kinase domainMore data for this Ligand-Target Pair
TargetCasein kinase I isoform alpha-like(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for CSNK1A1L kinase domainMore data for this Ligand-Target Pair
TargetCasein kinase I isoform alpha-like(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for CSNK1A1L kinase domainMore data for this Ligand-Target Pair
TargetCasein kinase I isoform alpha-like(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: 5.20E+3nMAssay Description:Binding constant for CSNK1A1L kinase domainMore data for this Ligand-Target Pair
TargetCasein kinase I isoform alpha-like(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for CSNK1A1L kinase domainMore data for this Ligand-Target Pair
TargetCasein kinase I isoform alpha-like(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for CSNK1A1L kinase domainMore data for this Ligand-Target Pair
TargetCasein kinase I isoform alpha-like(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for CSNK1A1L kinase domainMore data for this Ligand-Target Pair
TargetCasein kinase I isoform alpha-like(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: 4.60E+3nMAssay Description:Binding constant for CSNK1A1L kinase domainMore data for this Ligand-Target Pair
TargetCasein kinase I isoform alpha-like(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for CSNK1A1L kinase domainMore data for this Ligand-Target Pair