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Found 3519 Enz. Inhib. hit(s) with Target = 'Cholecystokinin receptor type A'
TargetCholecystokinin receptor type A(RAT)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50089269(CHEMBL276192 | N-(1-Carbamoyl-2-phenyl-ethyl)-3-{2...)
Affinity DataKi:  0.0200nMAssay Description:Inhibition of [125I]BH-CCK-8 binding to Cholecystokinin type A receptor of rat pancreatic tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50061829((R)-N-((S)-1-Carbamoyl-2-phenyl-ethyl)-3-({(S)-2-[...)
Affinity DataKi:  0.0300nMAssay Description:Binding affinity for Cholecystokinin type A receptor using [125I]BH-CCK-8 in rat pancreatic tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50061828(CHEMBL76248 | CID44356929 | N-(1-Carbamoyl-2-pheny...)
Affinity DataKi:  0.0300nMAssay Description:Binding affinity for Cholecystokinin type A receptor using [125I]BH-CCK-8 in rat pancreatic tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50061828(CHEMBL76248 | CID44356929 | N-(1-Carbamoyl-2-pheny...)
Affinity DataKi:  0.0300nMAssay Description:Inhibition of [125I]BH-CCK-8 binding to Cholecystokinin type A receptor of rat pancreatic tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50089268(CHEMBL267861 | N-(1-Carbamoyl-2-phenyl-ethyl)-3-{2...)
Affinity DataKi:  0.0500nMAssay Description:Inhibition of [125I]BH-CCK-8 binding to Cholecystokinin type A receptor of rat pancreatic tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50061832((S)-N-((S)-1-Carbamoyl-2-phenyl-ethyl)-3-{(S)-2-[(...)
Affinity DataKi:  0.0700nMAssay Description:Binding affinity for Cholecystokinin type A receptor using [125I]BH-CCK-8 in rat pancreatic tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM21147((3S)-3-[(2S)-2-[(2S)-2-{2-[(2S)-2-[(2S)-2-[(3S)-3-...)
Affinity DataKi:  0.0900nMAssay Description:Inhibition of [125I]BH-CCK-8 binding to Cholecystokinin type A receptor of rat pancreatic tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM21147((3S)-3-[(2S)-2-[(2S)-2-{2-[(2S)-2-[(2S)-2-[(3S)-3-...)
Affinity DataKi:  0.0900nMAssay Description:Binding affinity for Cholecystokinin type A receptor using [125I]BH-CCK-8 in rat pancreatic tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50449787(CHEMBL2062154 | PD-134308)
Affinity DataKi:  0.148nMAssay Description:Inhibition by displacing [3H]CCK-8S against Cholecystokinin type A receptor of rat pancreatic membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50005463((R)-1H-Indole-2-carboxylic acid (1-methyl-2-oxo-5-...)
Affinity DataKi:  0.148nMAssay Description:Inhibition by displacing [3H]CCK-8S against Cholecystokinin type A receptor of rat pancreatic membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM81962(S-L-365,260)
Affinity DataKi:  0.148nMAssay Description:Inhibition by displacing [3H]CCK-8S against Cholecystokinin type A receptor of rat pancreatic membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50016425((S)-3-{(S)-2-[(S)-2-(2-{(S)-2-[(S)-2-tert-Butoxyca...)
Affinity DataKi:  0.191nMAssay Description:Binding affinity measured by inhibiting [3H]Boc[Nle28,31]CCK27-33 specific binding to Cholecystokinin receptor in mouse brain membranes at a KD conce...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50061833((R)-N-((S)-1-Carbamoyl-2-phenyl-ethyl)-3-{(S)-2-[(...)
Affinity DataKi:  0.200nMAssay Description:Binding affinity for Cholecystokinin type A receptor using [125I]BH-CCK-8 in rat pancreatic tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Cavia porcellus)
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50016504((S)-3-(2-{[(S)-2-(2-{2-[2-tert-Butoxycarbonylamino...)
Affinity DataKi:  0.230nMAssay Description:The compound was tested for the inhibition of [3H]-Propionyl specific binding to Cholecystokinin 8 receptor of guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50369326(CHEMBL1791002)
Affinity DataKi:  0.240nMAssay Description:Binding affinity for Cholecystokinin type A receptor using [125I]BH-CCK-8 in rat pancreatic tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Cavia porcellus)
University Of Paris

Curated by ChEMBL
LigandPNGBDBM21147((3S)-3-[(2S)-2-[(2S)-2-{2-[(2S)-2-[(2S)-2-[(3S)-3-...)
Affinity DataKi:  0.280nMAssay Description:The compound was tested for the inhibition of [3H]-Propionyl specific binding to CCK-8 receptor of guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Cavia porcellus)
University Of Paris

Curated by ChEMBL
LigandPNGBDBM21147((3S)-3-[(2S)-2-[(2S)-2-{2-[(2S)-2-[(2S)-2-[(3S)-3-...)
Affinity DataKi:  0.280nMAssay Description:Displacement of 0.1 nM [3H]-pCCK-8 from guinea pig pancreatic membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Cavia porcellus)
University Of Paris

Curated by ChEMBL
LigandPNGBDBM21147((3S)-3-[(2S)-2-[(2S)-2-{2-[(2S)-2-[(2S)-2-[(3S)-3-...)
Affinity DataKi:  0.280nMAssay Description:Inhibition of [3H]pCCK-8 binding to Cholecystokinin type A receptor of Guinea pig pancreatic membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50060321(1H-Indole-2-carboxylic acid ((R)-1-methyl-2-oxo-5-...)
Affinity DataKi:  0.300nMAssay Description:Inhibition of [3H]-pCCK-8 specific binding to Cholecystokinin type A receptor of rat pancreasMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM21147((3S)-3-[(2S)-2-[(2S)-2-{2-[(2S)-2-[(2S)-2-[(3S)-3-...)
Affinity DataKi:  0.300nMAssay Description:Potency in displacing [3H]propionyl-Cholecystokinin from mouse brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Cavia porcellus)
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50016504((S)-3-(2-{[(S)-2-(2-{2-[2-tert-Butoxycarbonylamino...)
Affinity DataKi:  0.310nMAssay Description:Ability to displace 1 nM [3H]pCCK-8 from Cholecystokinin type A receptor in guinea pig pancreatic membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Homo sapiens (Human))
University Of Trieste

Curated by ChEMBL
LigandPNGBDBM50360276(CHEMBL1933104)
Affinity DataKi:  0.320nMAssay Description:Displacement of [125I]-BH-JMV-179 from wild type human CCK1 receptor expressed in COS7 cells after 60 mins by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM21147((3S)-3-[(2S)-2-[(2S)-2-{2-[(2S)-2-[(2S)-2-[(3S)-3-...)
Affinity DataKi:  0.491nMAssay Description:Binding affinity measured by inhibiting [3H]Boc[Nle28,31]CCK27-33 specific binding to Cholecystokinin receptor in mouse brain membranes at a KD conce...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM21147((3S)-3-[(2S)-2-[(2S)-2-{2-[(2S)-2-[(2S)-2-[(3S)-3-...)
Affinity DataKi:  0.520nMAssay Description:Inhibition of [3H]-pCCK-8 specific binding to Cholecystokinin type A receptor of rat pancreasMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50369325(CHEMBL1791005)
Affinity DataKi:  0.530nMAssay Description:Binding affinity for Cholecystokinin type A receptor using [125I]BH-CCK-8 in rat pancreatic tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Cavia porcellus)
University Of Paris

Curated by ChEMBL
LigandPNGBDBM21147((3S)-3-[(2S)-2-[(2S)-2-{2-[(2S)-2-[(2S)-2-[(3S)-3-...)
Affinity DataKi:  0.600nMAssay Description:Ability to displace 1 nM [3H]pCCK-8 from Cholecystokinin type A receptor in guinea pig pancreatic membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50060322(CHEMBL332261 | [(S)-1-((4aS,5S)-2-Benzyl-1,3-dioxo...)
Affinity DataKi:  0.620nMAssay Description:Inhibition of [3H]-pCCK-8 specific binding to Cholecystokinin type A receptor of rat pancreasMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Cavia porcellus)
University Of Paris

Curated by ChEMBL
LigandPNGBDBM21147((3S)-3-[(2S)-2-[(2S)-2-{2-[(2S)-2-[(2S)-2-[(3S)-3-...)
Affinity DataKi:  0.640nMAssay Description:Tested for the inhibition of [3H]-pCCK-8 binding to Cholecystokinin type A receptor in pancreatic membranes of guinea-pigMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(Cavia porcellus)
University Of Paris

Curated by ChEMBL
LigandPNGBDBM21147((3S)-3-[(2S)-2-[(2S)-2-{2-[(2S)-2-[(2S)-2-[(3S)-3-...)
Affinity DataKi:  0.640nMAssay Description:The compound was tested for the inhibition of [3H]-Propionyl specific binding to Cholecystokinin 8 receptor of guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Cavia porcellus)
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50092405((S)-N-((S)-1-Carbamoyl-2-phenyl-ethyl)-3-((S)-2-{[...)
Affinity DataKi: >0.700nMAssay Description:Affinity against Cholecystokinin type A receptor on guinea pig pancreatic membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Cavia porcellus)
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50092398((S)-3-((S)-2-{[(S)-2-tert-Butoxycarbonylamino-3-(1...)
Affinity DataKi: >0.700nMAssay Description:Affinity against Cholecystokinin type A receptor on guinea pig pancreatic membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Cavia porcellus)
University Of Paris

Curated by ChEMBL
LigandPNGBDBM21147((3S)-3-[(2S)-2-[(2S)-2-{2-[(2S)-2-[(2S)-2-[(3S)-3-...)
Affinity DataKi:  0.700nMAssay Description:Displacement of [3H]-pCCK-8 from cholecystokinin-A receptor in guinea pig pancreatic membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Cavia porcellus)
University Of Paris

Curated by ChEMBL
LigandPNGBDBM21147((3S)-3-[(2S)-2-[(2S)-2-{2-[(2S)-2-[(2S)-2-[(3S)-3-...)
Affinity DataKi:  0.700nMAssay Description:Compound was tested for binding affinity against CCK1 (cholecystokinin) receptor on guinea pig pancreatic membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50005463((R)-1H-Indole-2-carboxylic acid (1-methyl-2-oxo-5-...)
Affinity DataKi:  0.700nMAssay Description:Inhibition of [3H]-L-364,718 binding to cholecystokinin type A receptor in rat pancreas membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Cavia porcellus)
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50092405((S)-N-((S)-1-Carbamoyl-2-phenyl-ethyl)-3-((S)-2-{[...)
Affinity DataKi:  0.75nMAssay Description:Ability to displace 1 nM [3H]pCCK-8 from Cholecystokinin type A receptor in guinea pig pancreatic membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Cavia porcellus)
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50016504((S)-3-(2-{[(S)-2-(2-{2-[2-tert-Butoxycarbonylamino...)
Affinity DataKi:  0.930nMAssay Description:The compound was tested for the inhibition of [3H]-Propionyl specific binding to Cholecystokinin 8 receptor of guinea pig pancreatic membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Cavia porcellus)
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50016425((S)-3-{(S)-2-[(S)-2-(2-{(S)-2-[(S)-2-tert-Butoxyca...)
Affinity DataKi:  0.930nMAssay Description:Displacement of 0.1 nM [3H]-pCCK-8 from guinea pig pancreatic membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50089276(CHEMBL430608 | N-(1-Carbamoyl-2-phenyl-ethyl)-3-{2...)
Affinity DataKi:  0.980nMAssay Description:Inhibition of [125I]BH-CCK-8 binding to Cholecystokinin type A receptor of rat pancreatic tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50061834((R)-N-((S)-1-Carbamoyl-2-phenyl-ethyl)-3-{(S)-2-[(...)
Affinity DataKi:  0.980nMAssay Description:Binding affinity for Cholecystokinin type A receptor using [125I]BH-CCK-8 in rat pancreatic tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Cavia porcellus)
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50092388(3-(2-{[2-(3-tert-Butoxycarbonylamino-propionylamin...)
Affinity DataKi:  1.35nMAssay Description:Affinity against Cholecystokinin type A receptor on guinea pig pancreatic membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50211670(CHEMBL103750)
Affinity DataKi:  1.5nMAssay Description:Binding affinity was measured by its ability to displace [3H]CCK-8S from CCK-A receptor in rat pancreasMore data for this Ligand-Target Pair
In DepthDetails
TargetCholecystokinin receptor type A(Homo sapiens (Human))
University Of Trieste

Curated by ChEMBL
LigandPNGBDBM50321604((3S,6S,9S,12S,15R,18S,21S,24R,27S)-18-((1H-imidazo...)
Affinity DataKi:  1.60nMAssay Description:Displacement of [125I]CCK-8(SO3) from human CCK1 receptor expressed in human HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Homo sapiens (Human))
University Of Trieste

Curated by ChEMBL
LigandPNGBDBM50321604((3S,6S,9S,12S,15R,18S,21S,24R,27S)-18-((1H-imidazo...)
Affinity DataKi:  1.60nMAssay Description:Displacement of [125I]CCK-8(SO3) from human CCK1 receptor expressed in human HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Cavia porcellus)
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50016506(CHEMBL262687 | Sodium; (4-{2-(2-acetylamino-3-carb...)
Affinity DataKi:  1.70nMAssay Description:The compound was tested for the inhibition of [3H]-Propionyl specific binding to Cholecystokinin 8 receptor of guinea pig pancreatic membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50002477((S)-3-{(S)-2-[(S)-2-tert-Butoxycarbonylamino-3-(1H...)
Affinity DataKi:  1.80nMAssay Description:Displacement of [3H]pentagastrin from Cholecystokinin receptor of mouse cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50226755(CHEMBL415630)
Affinity DataKi:  2nMAssay Description:Displacement of [3H]pentagastrin from Cholecystokinin receptor of mouse cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Cavia porcellus)
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50092391(3-(2-{[2-(2-Carbamoyl-acetylamino)-3-(1H-indol-3-y...)
Affinity DataKi:  2.05nMAssay Description:Affinity against Cholecystokinin type A receptor on guinea pig pancreatic membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Homo sapiens (Human))
University Of Trieste

Curated by ChEMBL
LigandPNGBDBM50360276(CHEMBL1933104)
Affinity DataKi:  2.30nMAssay Description:Displacement of [125I]BH-(Thr,-Nle)-CCK-9 from human CCK1 receptor expressed in COS-7 cells after 60 mins by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Cavia porcellus)
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50092396(3-(2-{[2-Amino-3-(1H-indol-3-yl)-propionyl]-methyl...)
Affinity DataKi:  2.60nMAssay Description:Affinity against Cholecystokinin type A receptor on guinea pig pancreatic membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Cavia porcellus)
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50092398((S)-3-((S)-2-{[(S)-2-tert-Butoxycarbonylamino-3-(1...)
Affinity DataKi:  2.60nMAssay Description:Ability to displace 1 nM [3H]pCCK-8 from Cholecystokinin type A receptor in guinea pig pancreatic membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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