Found 22 Enz. Inhib. hit(s) with Target = 'Potassium channel subfamily K member 10' 
Affinity DataIC50: 7.60E+3nMAssay Description:Inhibition of of TREK2 (unknown origin) expressed in HEK293 cells assessed as reduction in channel currentsMore data for this Ligand-Target Pair
Affinity DataIC50: 2.40E+4nMAssay Description:Inhibition of of TREK2 (unknown origin) expressed in oocytes assessed as reduction in channel currentsMore data for this Ligand-Target Pair
TargetPotassium channel subfamily K member 10(Rattus norvegicus)
Gyeongsang National University
Curated by ChEMBL
Gyeongsang National University
Curated by ChEMBL
Affinity DataIC50: 6.20E+4nMAssay Description:Inhibition of rat TREK2 channel -mediated current expressed in HEK293 at 60 mV holding potential by patch clamp methodMore data for this Ligand-Target Pair
TargetPotassium channel subfamily K member 10(Rattus norvegicus)
Gyeongsang National University
Curated by ChEMBL
Gyeongsang National University
Curated by ChEMBL
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of rat TREK2 channel -mediated current expressed in HEK293 at 60 mV holding potential by patch clamp methodMore data for this Ligand-Target Pair
TargetPotassium channel subfamily K member 10(Rattus norvegicus)
Gyeongsang National University
Curated by ChEMBL
Gyeongsang National University
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of rat TREK2 channel -mediated current expressed in HEK293 at 60 mV holding potential by patch clamp methodMore data for this Ligand-Target Pair
Affinity DataEC50: >3.00E+4nMAssay Description:Activation of human TREK2 by thallium flux mobilization assayMore data for this Ligand-Target Pair
Affinity DataEC50: 6.80E+3nMAssay Description:Activation of human TREK2 by thallium flux mobilization assayMore data for this Ligand-Target Pair
Affinity DataEC50: 5.90E+3nMAssay Description:Activation of human TREK2 by thallium flux mobilization assayMore data for this Ligand-Target Pair
Affinity DataEC50: 7.70E+3nMAssay Description:Activation of human TREK2 by thallium flux mobilization assayMore data for this Ligand-Target Pair
Affinity DataEC50: 5.50E+3nMAssay Description:Activation of human TREK2 by thallium flux mobilization assayMore data for this Ligand-Target Pair
Affinity DataEC50: 2.85E+4nMAssay Description:Activation of human TREK2 by thallium flux mobilization assayMore data for this Ligand-Target Pair
Affinity DataEC50: >3.00E+4nMAssay Description:Activation of human TREK2 by thallium flux mobilization assayMore data for this Ligand-Target Pair
Affinity DataEC50: 5.60E+3nMAssay Description:Activation of human TREK2 by thallium flux mobilization assayMore data for this Ligand-Target Pair
Affinity DataEC50: 2.65E+4nMAssay Description:Activation of human TREK2 by thallium flux mobilization assayMore data for this Ligand-Target Pair
Affinity DataEC50: >3.00E+4nMAssay Description:Activation of human TREK2 by thallium flux mobilization assayMore data for this Ligand-Target Pair
Affinity DataEC50: <3.60E+3nMAssay Description:Activation of human TREK2 by thallium flux mobilization assayMore data for this Ligand-Target Pair
Affinity DataEC50: >3.00E+4nMAssay Description:Activation of human TREK2 by thallium flux mobilization assayMore data for this Ligand-Target Pair
Affinity DataEC50: 5.00E+3nMAssay Description:Activation of human TREK2 by thallium flux mobilization assayMore data for this Ligand-Target Pair
Affinity DataEC50: 7.70E+3nMAssay Description:Activation of human TREK2 by thallium flux mobilization assayMore data for this Ligand-Target Pair
TargetPotassium channel subfamily K member 10(Rattus norvegicus)
Gyeongsang National University
Curated by ChEMBL
Gyeongsang National University
Curated by ChEMBL
Affinity DataEC50: 1.67E+5nMAssay Description:Activation of rat TREK2 channel -mediated current expressed in HEK293 at 60 mV holding potential by patch clamp methodMore data for this Ligand-Target Pair
Affinity DataEC50: 3.00E+4nMAssay Description:Activation of TREK2 (unknown origin) expressed in Xenopus oocytes assessed as increase in channel currentsMore data for this Ligand-Target Pair
Affinity DataEC50: 7.50E+3nMAssay Description:Activation of human TREK2 by thallium flux mobilization assayMore data for this Ligand-Target Pair
