Compile Data Set for Download or QSAR
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Found 5 Enz. Inhib. hit(s) with Target = 'Diamine acetyltransferase 1'
TargetDiamine acetyltransferase 1(Homo sapiens (Human))
Xavier University Of Louisiana

Curated by ChEMBL
LigandPNGBDBM45440(4-[5-(4-amidinophenoxy)pentoxy]benzamidine;2-hydro...)
Affinity DataKi:  2.00E+3nMAssay Description:Inhibition of human SSAT using spermidine as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDiamine acetyltransferase 1(Homo sapiens (Human))
Xavier University Of Louisiana

Curated by ChEMBL
LigandPNGBDBM50000999(CHEBI:81724 | DIMINAZENE)
Affinity DataKi:  2.40E+3nMAssay Description:Inhibition of human SSAT using spermidine as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDiamine acetyltransferase 1(Homo sapiens (Human))
Xavier University Of Louisiana

Curated by ChEMBL
LigandPNGBDBM50095444(CHEMBL315330 | Methyl-phosphonic acid mono-{3-[3-(...)
Affinity DataKi:  5.00E+4nMAssay Description:Inhibitory activity against human SSATMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDiamine acetyltransferase 1(Homo sapiens (Human))
Xavier University Of Louisiana

Curated by ChEMBL
LigandPNGBDBM50095431(CHEMBL86940 | N-Ethyl-N'-[3-(3-prop-2-ynylamino-pr...)
Affinity DataIC50:  4.00E+4nMAssay Description:Inhibitory activity of compound against SSAT extracted from superinduced H157 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDiamine acetyltransferase 1(Homo sapiens (Human))
Xavier University Of Louisiana

Curated by ChEMBL
LigandPNGBDBM50095437(CHEMBL33387 | N-[3-(Cyclopropylmethyl-amino)-propy...)
Affinity DataIC50:  1.00E+5nMAssay Description:Inhibitory activity of compound against SSAT extracted from superinduced H157 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed