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Found 214 Enz. Inhib. hit(s) with Target = 'Pyroglutamylated RF-amide peptide receptor'
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50347819(CHEMBL1802414 | P550)
Affinity DataKi:  2nMAssay Description:Displacement of [125I]-43RFa from human QRFP receptor expressed in CHO cells by TopCount scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50347819(CHEMBL1802414 | P550)
In DepthDetails ArticlePubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50347818(CHEMBL1802413 | P518)
In DepthDetails ArticlePubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM86228(P517)
Affinity DataKi:  235nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM86226(P52)
Affinity DataKi:  245nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM86224(P513)
Affinity DataKi:  258nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM86227(P552)
Affinity DataKi:  607nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM86225(P51)
Affinity DataKi:  1.50E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50583766(CHEMBL5074999)
Affinity DataKi: >5.00E+3nMAssay Description:Displacement of [125I]-43RFa from human QRFP receptor expressed in CHO cells by TopCount scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50565194(CHEMBL4793841)
Affinity DataKi: >5.00E+3nMAssay Description:Displacement of [125I]-43RFa from human QRFP receptor expressed in CHO cell membrane by TopCount scintillation counter methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50191288(CHEMBL3982697)
Affinity DataKi: >5.00E+3nMAssay Description:Displacement of [125I]-43RFa from human QRFP receptor expressed in CHO cell membrane by TopCount scintillation counter methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM86229(YGGFMRF-amide)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50583777(CHEMBL5085324)
Affinity DataKi: >5.00E+4nMAssay Description:Displacement of [125I]-43RFa from human QRFP receptor expressed in CHO cells by TopCount scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50583773(CHEMBL5091013)
Affinity DataKi: >5.00E+4nMAssay Description:Displacement of [125I]-43RFa from human QRFP receptor expressed in CHO cells by TopCount scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50347818(CHEMBL1802413 | P518)
Affinity DataIC50:  1.30nMAssay Description:Displacement of [125I]26RFa from human GPR103 expressed in HEK293 cells incubated for 1 h by gamma counter based methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50020015(CHEMBL3287814)
Affinity DataIC50:  13nMAssay Description:Antagonist activity at human GPR103 receptor assessed as inhibition of inositol-1-phosphate production by cell-based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50020011(CHEMBL3287810)
Affinity DataIC50:  20nMAssay Description:Antagonist activity at human GPR103 receptor assessed as inhibition of inositol-1-phosphate production by cell-based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50020014(CHEMBL3287813)
Affinity DataIC50:  20nMAssay Description:Antagonist activity at human GPR103 receptor assessed as inhibition of inositol-1-phosphate production by cell-based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50020011(CHEMBL3287810)
Affinity DataIC50:  25nMAssay Description:Displacement of [125I]-QRFP43 from human GPR103 receptor overexpressed in HEK membranes after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50020015(CHEMBL3287814)
Affinity DataIC50:  40nMAssay Description:Displacement of [125I]-QRFP43 from human GPR103 receptor overexpressed in HEK membranes after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50045830(CHEMBL3314362)
Affinity DataIC50:  40nMAssay Description:Displacement of [125I]QRFP43 from human GPR103 receptor expressed in HEK cells after 90 mins incubation by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50019982(CHEMBL3287584)
Affinity DataIC50:  50nMAssay Description:Antagonist activity at human GPR103 receptor assessed as inhibition of inositol-1-phosphate production by cell-based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50020012(CHEMBL3287811)
Affinity DataIC50:  63nMAssay Description:Antagonist activity at human GPR103 receptor assessed as inhibition of inositol-1-phosphate production by cell-based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50045833(CHEMBL3314349)
Affinity DataIC50:  70nMAssay Description:Displacement of [125I]QRFP43 from human GPR103 receptor expressed in HEK cells after 90 mins incubation by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50045833(CHEMBL3314349)
Affinity DataIC50:  70nMAssay Description:Inhibition of human GPR103 receptor expressed in CHOK1 cells by IP-1 assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50019983(CHEMBL3287585)
Affinity DataIC50:  79nMAssay Description:Antagonist activity at human GPR103 receptor assessed as inhibition of inositol-1-phosphate production by cell-based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50019983(CHEMBL3287585)
Affinity DataIC50:  79nMAssay Description:Displacement of [125I]-QRFP43 from human GPR103 receptor overexpressed in HEK membranes after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50020012(CHEMBL3287811)
Affinity DataIC50:  100nMAssay Description:Displacement of [125I]-QRFP43 from human GPR103 receptor overexpressed in HEK membranes after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50020010(CHEMBL3287586)
Affinity DataIC50:  100nMAssay Description:Antagonist activity at human GPR103 receptor assessed as inhibition of inositol-1-phosphate production by cell-based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50045838(CHEMBL3314358)
Affinity DataIC50:  110nMAssay Description:Inhibition of human GPR103 receptor expressed in CHOK1 cells by IP-1 assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50020014(CHEMBL3287813)
Affinity DataIC50:  126nMAssay Description:Displacement of [125I]-QRFP43 from human GPR103 receptor overexpressed in HEK membranes after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50020010(CHEMBL3287586)
Affinity DataIC50:  126nMAssay Description:Displacement of [125I]-QRFP43 from human GPR103 receptor overexpressed in HEK membranes after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50045842(CHEMBL3314354)
Affinity DataIC50:  130nMAssay Description:Inhibition of human GPR103 receptor expressed in CHOK1 cells by IP-1 assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50020013(CHEMBL3287812)
Affinity DataIC50:  158nMAssay Description:Antagonist activity at human GPR103 receptor assessed as inhibition of inositol-1-phosphate production by cell-based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50019982(CHEMBL3287584)
Affinity DataIC50:  158nMAssay Description:Displacement of [125I]-QRFP43 from human GPR103 receptor overexpressed in HEK membranes after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50019979(CHEMBL3287833)
Affinity DataIC50:  200nMAssay Description:Displacement of [125I]-QRFP43 from human GPR103 receptor overexpressed in HEK membranes after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50045831(CHEMBL3314352)
Affinity DataIC50:  240nMAssay Description:Inhibition of human GPR103 receptor expressed in CHOK1 cells by IP-1 assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50020020(CHEMBL3287819)
Affinity DataIC50:  251nMAssay Description:Antagonist activity at human GPR103 receptor assessed as inhibition of inositol-1-phosphate production by cell-based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50020022(CHEMBL3287821)
Affinity DataIC50:  251nMAssay Description:Antagonist activity at human GPR103 receptor assessed as inhibition of inositol-1-phosphate production by cell-based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50045831(CHEMBL3314352)
Affinity DataIC50:  280nMAssay Description:Displacement of [125I]QRFP43 from human GPR103 receptor expressed in HEK cells after 90 mins incubation by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50019979(CHEMBL3287833)
Affinity DataIC50:  316nMAssay Description:Antagonist activity at human GPR103 receptor assessed as inhibition of inositol-1-phosphate production by cell-based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50045834(CHEMBL3314361)
Affinity DataIC50:  460nMAssay Description:Inhibition of human GPR103 receptor expressed in CHOK1 cells by IP-1 assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50045837(CHEMBL3314359)
Affinity DataIC50:  500nMAssay Description:Inhibition of human GPR103 receptor expressed in CHOK1 cells by IP-1 assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50019976(CHEMBL3287827)
Affinity DataIC50:  501nMAssay Description:Antagonist activity at human GPR103 receptor assessed as inhibition of inositol-1-phosphate production by cell-based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50020020(CHEMBL3287819)
Affinity DataIC50:  501nMAssay Description:Displacement of [125I]-QRFP43 from human GPR103 receptor overexpressed in HEK membranes after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50045846(CHEMBL3314350)
Affinity DataIC50:  570nMAssay Description:Inhibition of human GPR103 receptor expressed in CHOK1 cells by IP-1 assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50469449(CHEMBL4277047)
Affinity DataIC50:  579nMAssay Description:Antagonist activity at human QRFPR expressed in CHO cells co-expressing Galpha16 assessed as inhibition of 26RFa-induced Ca2+ mobilization preincubat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50020022(CHEMBL3287821)
Affinity DataIC50:  631nMAssay Description:Displacement of [125I]-QRFP43 from human GPR103 receptor overexpressed in HEK membranes after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50045836(CHEMBL3314360)
Affinity DataIC50:  710nMAssay Description:Inhibition of human GPR103 receptor expressed in CHOK1 cells by IP-1 assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50019974(CHEMBL3287825)
Affinity DataIC50:  794nMAssay Description:Antagonist activity at human GPR103 receptor assessed as inhibition of inositol-1-phosphate production by cell-based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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