Compile Data Set for Download or QSAR
maximum 50k data
Found 42 of ic50 for UniProtKB: Q8R493
TargetNeuronal acetylcholine receptor subunit beta-2/beta-4(Mus musculus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50270397(CHEMBL4070098)
Affinity DataIC50:  220nMAssay Description:Antagonist activity at mouse alpha4beta2 nAChR expressed in HEK293 cells assessed as inhibition of (S)-nicotine-induced current response measured up ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit beta-2/beta-4(Mus musculus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50270370(CHEMBL4101688)
Affinity DataIC50:  520nMAssay Description:Antagonist activity at mouse alpha4beta2 nAChR expressed in HEK293 cells assessed as inhibition of (S)-nicotine-induced current response measured up ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit beta-2/beta-4(Mus musculus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50270396(CHEMBL4073773)
Affinity DataIC50:  600nMAssay Description:Antagonist activity at mouse alpha4beta2 nAChR expressed in HEK293 cells assessed as inhibition of (S)-nicotine-induced current response measured up ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit beta-2/beta-4(Mus musculus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50270401(CHEMBL4064521)
Affinity DataIC50:  1.20E+3nMAssay Description:Antagonist activity at mouse alpha4beta2 nAChR expressed in HEK293 cells assessed as inhibition of (S)-nicotine-induced current response measured up ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit beta-2/beta-4(Mus musculus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50270364(CHEMBL4064684)
Affinity DataIC50:  1.30E+3nMAssay Description:Antagonist activity at mouse alpha4beta2 nAChR expressed in HEK293 cells assessed as inhibition of (S)-nicotine-induced current response measured up ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit beta-2/beta-4(Mus musculus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50270402(CHEMBL4097677)
Affinity DataIC50:  1.40E+3nMAssay Description:Antagonist activity at mouse alpha4beta2 nAChR expressed in HEK293 cells assessed as inhibition of (S)-nicotine-induced current response measured up ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit beta-2/beta-4(Mus musculus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50270368(CHEMBL4082570)
Affinity DataIC50:  1.80E+3nMAssay Description:Antagonist activity at mouse alpha4beta2 nAChR expressed in HEK293 cells assessed as inhibition of (S)-nicotine-induced current response measured up ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit beta-2/beta-4(Mus musculus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50006634(CHEMBL3235510)
Affinity DataIC50:  2.30E+3nMAssay Description:Antagonist activity at mouse alpha4beta2 nAChR expressed in HEK293 cells assessed as inhibition of (S)-nicotine-induced current response measured up ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit beta-2/beta-4(Mus musculus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50006638(CHEMBL2140445)
Affinity DataIC50:  2.60E+3nMAssay Description:Antagonist activity at mouse alpha4beta2 nAChR expressed in HEK293 cells assessed as inhibition of (S)-nicotine-induced current response measured up ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit beta-2/beta-4(Mus musculus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50270372(CHEMBL4104998)
Affinity DataIC50:  3.10E+3nMAssay Description:Antagonist activity at mouse alpha4beta2 nAChR expressed in HEK293 cells assessed as inhibition of (S)-nicotine-induced current response measured up ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit beta-2/beta-4(Mus musculus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50006640(CHEMBL593001)
Affinity DataIC50:  4.40E+3nMAssay Description:Antagonist activity at mouse alpha4beta2 nAChR expressed in HEK293 cells assessed as inhibition of (S)-nicotine-induced current response measured up ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit beta-2/beta-4(Mus musculus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50270371(CHEMBL4087153)
Affinity DataIC50:  5.70E+3nMAssay Description:Antagonist activity at mouse alpha4beta2 nAChR expressed in HEK293 cells assessed as inhibition of (S)-nicotine-induced current response measured up ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit beta-2/beta-4(Mus musculus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50270375(CHEMBL4075463)
Affinity DataIC50:  6.20E+3nMAssay Description:Antagonist activity at mouse alpha4beta2 nAChR expressed in HEK293 cells assessed as inhibition of (S)-nicotine-induced current response measured up ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit beta-2/beta-4(Mus musculus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50270382(CHEMBL4082090)
Affinity DataIC50:  7.20E+3nMAssay Description:Antagonist activity at mouse alpha4beta2 nAChR expressed in HEK293 cells assessed as inhibition of (S)-nicotine-induced current response measured up ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit beta-2/beta-4(Mus musculus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50270388(CHEMBL4083525)
Affinity DataIC50:  7.20E+3nMAssay Description:Antagonist activity at mouse alpha4beta2 nAChR expressed in HEK293 cells assessed as inhibition of (S)-nicotine-induced current response measured up ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit beta-2/beta-4(Mus musculus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50270405(CHEMBL4102579)
Affinity DataIC50:  9.10E+3nMAssay Description:Antagonist activity at mouse alpha4beta2 nAChR expressed in HEK293 cells assessed as inhibition of (S)-nicotine-induced current response measured up ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit beta-2/beta-4(Mus musculus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50270395(CHEMBL4092845)
Affinity DataIC50:  1.10E+4nMAssay Description:Antagonist activity at mouse alpha4beta2 nAChR expressed in HEK293 cells assessed as inhibition of (S)-nicotine-induced current response measured up ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit beta-2/beta-4(Mus musculus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50270407(CHEMBL1570477)
Affinity DataIC50:  1.10E+4nMAssay Description:Antagonist activity at mouse alpha4beta2 nAChR expressed in HEK293 cells assessed as inhibition of (S)-nicotine-induced current response measured up ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit beta-2/beta-4(Mus musculus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50270399(CHEMBL4073109)
Affinity DataIC50:  1.20E+4nMAssay Description:Antagonist activity at mouse alpha4beta2 nAChR expressed in HEK293 cells assessed as inhibition of (S)-nicotine-induced current response measured up ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit beta-2/beta-4(Mus musculus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50014648(6,7-Dimethoxy-2-methyl-1,2,3,4-tetrahydro-isoquino...)
Affinity DataIC50:  1.20E+4nMAssay Description:Antagonist activity at mouse alpha4beta2 nAChR expressed in HEK293 cells assessed as inhibition of (S)-nicotine-induced current response measured up ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit beta-2/beta-4(Mus musculus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50270373(CHEMBL4073899)
Affinity DataIC50:  1.50E+4nMAssay Description:Antagonist activity at mouse alpha4beta2 nAChR expressed in HEK293 cells assessed as inhibition of (S)-nicotine-induced current response measured up ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit beta-2/beta-4(Mus musculus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50270362(CHEMBL4077320)
Affinity DataIC50:  1.60E+4nMAssay Description:Antagonist activity at mouse alpha4beta2 nAChR expressed in HEK293 cells assessed as inhibition of (S)-nicotine-induced current response measured up ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit beta-2/beta-4(Mus musculus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50270389(CHEMBL4061335)
Affinity DataIC50:  2.30E+4nMAssay Description:Antagonist activity at mouse alpha4beta2 nAChR expressed in HEK293 cells assessed as inhibition of (S)-nicotine-induced current response measured up ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit beta-2/beta-4(Mus musculus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50270390(CHEMBL4062419)
Affinity DataIC50:  2.40E+4nMAssay Description:Antagonist activity at mouse alpha4beta2 nAChR expressed in HEK293 cells assessed as inhibition of (S)-nicotine-induced current response measured up ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit beta-2/beta-4(Mus musculus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50270403(CHEMBL4080088)
Affinity DataIC50:  3.00E+4nMAssay Description:Antagonist activity at mouse alpha4beta2 nAChR expressed in HEK293 cells assessed as inhibition of (S)-nicotine-induced current response measured up ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit beta-2/beta-4(Mus musculus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50270393(CHEMBL4071054)
Affinity DataIC50:  3.00E+4nMAssay Description:Antagonist activity at mouse alpha4beta2 nAChR expressed in HEK293 cells assessed as inhibition of (S)-nicotine-induced current response measured up ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit beta-2/beta-4(Mus musculus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50270394(CHEMBL4061094)
Affinity DataIC50:  3.00E+4nMAssay Description:Antagonist activity at mouse alpha4beta2 nAChR expressed in HEK293 cells assessed as inhibition of (S)-nicotine-induced current response measured up ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit beta-2/beta-4(Mus musculus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50270369(CHEMBL4083684)
Affinity DataIC50:  3.00E+4nMAssay Description:Antagonist activity at mouse alpha4beta2 nAChR expressed in HEK293 cells assessed as inhibition of (S)-nicotine-induced current response measured up ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit beta-2/beta-4(Mus musculus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50006633(CHEMBL3235509)
Affinity DataIC50:  3.00E+4nMAssay Description:Antagonist activity at mouse alpha4beta2 nAChR expressed in HEK293 cells assessed as inhibition of (S)-nicotine-induced current response measured up ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit beta-2/beta-4(Mus musculus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50270365(CHEMBL4078302)
Affinity DataIC50:  3.00E+4nMAssay Description:Antagonist activity at mouse alpha4beta2 nAChR expressed in HEK293 cells assessed as inhibition of (S)-nicotine-induced current response measured up ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit beta-2/beta-4(Mus musculus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50270367(CHEMBL4067385)
Affinity DataIC50:  3.00E+4nMAssay Description:Antagonist activity at mouse alpha4beta2 nAChR expressed in HEK293 cells assessed as inhibition of (S)-nicotine-induced current response measured up ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit beta-2/beta-4(Mus musculus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50270406(CHEMBL4084130)
Affinity DataIC50:  3.00E+4nMAssay Description:Antagonist activity at mouse alpha4beta2 nAChR expressed in HEK293 cells assessed as inhibition of (S)-nicotine-induced current response measured up ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit beta-2/beta-4(Mus musculus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50270374(CHEMBL4099972)
Affinity DataIC50:  3.00E+4nMAssay Description:Antagonist activity at mouse alpha4beta2 nAChR expressed in HEK293 cells assessed as inhibition of (S)-nicotine-induced current response measured up ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit beta-2/beta-4(Mus musculus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50006628(CHEMBL3235504)
Affinity DataIC50:  3.10E+4nMAssay Description:Antagonist activity at mouse alpha4/beta2 nAChR expressed in HEK293 cells assessed as inhibition of (S)-nicotine-induced activity by FLIPR membrane p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit beta-2/beta-4(Mus musculus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50270398(CHEMBL4067398)
Affinity DataIC50:  5.00E+4nMAssay Description:Antagonist activity at mouse alpha4beta2 nAChR expressed in HEK293 cells assessed as inhibition of (S)-nicotine-induced current response measured up ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit beta-2/beta-4(Mus musculus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50270366(CHEMBL4087050)
Affinity DataIC50:  5.00E+4nMAssay Description:Antagonist activity at mouse alpha4beta2 nAChR expressed in HEK293 cells assessed as inhibition of (S)-nicotine-induced current response measured up ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit beta-2/beta-4(Mus musculus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50270363(CHEMBL4086188)
Affinity DataIC50: >1.00E+5nMAssay Description:Antagonist activity at mouse alpha4beta2 nAChR expressed in HEK293 cells assessed as inhibition of (S)-nicotine-induced current response measured up ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit beta-2/beta-4(Mus musculus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50270376(Laudanosine)
Affinity DataIC50: >1.00E+5nMAssay Description:Antagonist activity at mouse alpha4beta2 nAChR expressed in HEK293 cells assessed as inhibition of (S)-nicotine-induced current response measured up ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit beta-2/beta-4(Mus musculus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50270404(CHEMBL4097292)
Affinity DataIC50:  1.00E+5nMAssay Description:Antagonist activity at mouse alpha4beta2 nAChR expressed in HEK293 cells assessed as inhibition of (S)-nicotine-induced current response measured up ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit beta-2/beta-4(Mus musculus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50270400(CHEMBL363360)
Affinity DataIC50: >1.00E+5nMAssay Description:Antagonist activity at mouse alpha4beta2 nAChR expressed in HEK293 cells assessed as inhibition of (S)-nicotine-induced current response measured up ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit beta-2/beta-4(Mus musculus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50270361(CHEMBL4077524)
Affinity DataIC50: >1.00E+5nMAssay Description:Antagonist activity at mouse alpha4beta2 nAChR expressed in HEK293 cells assessed as inhibition of (S)-nicotine-induced current response measured up ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit beta-2/beta-4(Mus musculus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50270377(CHEMBL4081330)
Affinity DataIC50: >1.00E+5nMAssay Description:Antagonist activity at mouse alpha4beta2 nAChR expressed in HEK293 cells assessed as inhibition of (S)-nicotine-induced current response measured up ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed