Compile Data Set for Download or QSAR
maximum 50k data
Found 6 of ec50 for monomerid = 50316375
TargetGlutamate receptor 2(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50316375(CHEMBL1097939 | LY-404187 | N-[2-(4'-cyanobiphenyl...)
Affinity DataEC50:  150nMAssay Description:Activity at human recombinant GluA2 receptor flip isoform expressed in HEK293 cells assessed as effect on glutamate-induced calcium flux by Fluo-4/AM...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 2(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50316375(CHEMBL1097939 | LY-404187 | N-[2-(4'-cyanobiphenyl...)
Affinity DataEC50:  1.44E+3nMAssay Description:Activity at human recombinant GluA2 flop isoform expressed in HEK203 cells assessed as blocked of receptor desensitizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 2(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50316375(CHEMBL1097939 | LY-404187 | N-[2-(4'-cyanobiphenyl...)
Affinity DataEC50:  1.44E+3nMAssay Description:Activity at human recombinant GluA2 receptor flop isoform expressed in HEK293 cells assessed as effect on glutamate-induced calcium flux by Fluo-4/AM...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 3(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50316375(CHEMBL1097939 | LY-404187 | N-[2-(4'-cyanobiphenyl...)
Affinity DataEC50:  1.66E+3nMAssay Description:Activity at human recombinant GluA3 receptor flip isoform expressed in HEK293 cells assessed as effect on glutamate-induced calcium flux by Fluo-4/AM...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 1(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50316375(CHEMBL1097939 | LY-404187 | N-[2-(4'-cyanobiphenyl...)
Affinity DataEC50:  5.65E+3nMAssay Description:Activity at human recombinant GluA1 receptor flip isoform expressed in HEK293 cells assessed as effect on glutamate-induced calcium flux by Fluo-4/AM...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 2(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50316375(CHEMBL1097939 | LY-404187 | N-[2-(4'-cyanobiphenyl...)
Affinity DataEC50:  1.50E+4nMAssay Description:Activity at human recombinant GluA2 flip isoform expressed in HEK203 cells assessed as blocked of receptor desensitizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed