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Found 3 of ec50 for monomerid = 7377
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM7377(4-{7-butyl-5H-pyrrolo[2,3-b]pyrazin-6-yl}phenol | ...)
Affinity DataEC50:  111nMAssay Description:Activity at human wild type CFTR expressed in F508del-CF1 cells assessed as forskolin stimulated iodide fluxChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM7377(4-{7-butyl-5H-pyrrolo[2,3-b]pyrazin-6-yl}phenol | ...)
Affinity DataEC50:  140nMAssay Description:Activity at human wild type CFTR expressed in Calu3 cells assessed as forskolin stimulated iodide fluxChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM7377(4-{7-butyl-5H-pyrrolo[2,3-b]pyrazin-6-yl}phenol | ...)
Affinity DataEC50:  150nMAssay Description:Activity at human wild type CFTR expressed in CHO cells assessed as forskolin stimulated iodide fluxChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed