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Found 11 of ic50 for monomerid = 12183
TargetDipeptidyl peptidase 8(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM12183((2S)-1-[(2S)-2-amino-4-{4-[bis(4-fluorophenyl)meth...)
Affinity DataIC50:  14nMAssay Description:Inhibition of human recombinant His-tagged DPP8 expressed in insect cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 8(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM12183((2S)-1-[(2S)-2-amino-4-{4-[bis(4-fluorophenyl)meth...)
Affinity DataIC50:  16nMpH: 8.0 T: 2°CAssay Description:The enzyme activity resulted in the liberation of free pNA at 405 nm. Reaction progress was monitored using a Molecular Devices SpectraMax Plus micro...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 8(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM12183((2S)-1-[(2S)-2-amino-4-{4-[bis(4-fluorophenyl)meth...)
Affinity DataIC50:  16nMAssay Description:Inhibitory concentration against Dipeptidyl-peptidase 8More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 9(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM12183((2S)-1-[(2S)-2-amino-4-{4-[bis(4-fluorophenyl)meth...)
Affinity DataIC50:  53nMAssay Description:Inhibition of human recombinant His-tagged DPP9 expressed in insect cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM12183((2S)-1-[(2S)-2-amino-4-{4-[bis(4-fluorophenyl)meth...)
Affinity DataIC50:  227nMAssay Description:Inhibitory concentration against Dipeptidyl-peptidase IV [DPP-IV]More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM12183((2S)-1-[(2S)-2-amino-4-{4-[bis(4-fluorophenyl)meth...)
Affinity DataIC50:  274nMAssay Description:The enzyme activity resulted in the liberation of free pNA at 405 nm. Reaction progress was monitored using a Molecular Devices SpectraMax Plus micro...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM12183((2S)-1-[(2S)-2-amino-4-{4-[bis(4-fluorophenyl)meth...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human recombinant His-tagged DPP4 expressed in insect cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM12183((2S)-1-[(2S)-2-amino-4-{4-[bis(4-fluorophenyl)meth...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human recombinant His-tagged DPP2 expressed in insect cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase FAP(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM12183((2S)-1-[(2S)-2-amino-4-{4-[bis(4-fluorophenyl)meth...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human recombinant FAP expressed in Hi5 insect cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM12183((2S)-1-[(2S)-2-amino-4-{4-[bis(4-fluorophenyl)meth...)
Affinity DataIC50: >1.00E+5nMAssay Description:The enzyme activity resulted in the liberation of free pNA at 405 nm. Reaction progress was monitored using a Molecular Devices SpectraMax Plus micro...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM12183((2S)-1-[(2S)-2-amino-4-{4-[bis(4-fluorophenyl)meth...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibitory concentration against DPP-II [Quiescent cell proline dipeptidase] or DPP-VIIMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed