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Found 7 of ic50 for monomerid = 12590
TargetReplicase polyprotein 1ab(2019-nCoV)
Fraunhofer Institute For Translational Medicine And Pharmacology (Itmp) And Fraunhofer Cluster Of Excellence For Immune Mediated Diseases (Cimd

LigandPNGBDBM12590((6-aminoacridin-3-yl)amine | MLS003876812 | Profla...)
Affinity DataIC50:  830nMAssay Description:Primary assay principle based on quenched FRET peptide substrate of SARS-CoV-2 3CL-Pro (lhs). Inhibiting compounds reduce fluorescence signal relativ...More data for this Ligand-Target Pair
TargetReplicase polyprotein 1ab(2019-nCoV)
Fraunhofer Institute For Translational Medicine And Pharmacology (Itmp) And Fraunhofer Cluster Of Excellence For Immune Mediated Diseases (Cimd

LigandPNGBDBM12590((6-aminoacridin-3-yl)amine | MLS003876812 | Profla...)
Affinity DataIC50:  1.46E+3nMAssay Description:Inhibition of SARS-CoV-2 papain-like protease using ISG15-AMC as substrateMore data for this Ligand-Target Pair
TargetReplicase polyprotein 1ab(2019-nCoV)
Fraunhofer Institute For Translational Medicine And Pharmacology (Itmp) And Fraunhofer Cluster Of Excellence For Immune Mediated Diseases (Cimd

LigandPNGBDBM12590((6-aminoacridin-3-yl)amine | MLS003876812 | Profla...)
Affinity DataIC50:  1.66E+3nMAssay Description:Inhibition of SARS-CoV-2 papain-like protease using RLRGG-AMC as substrateMore data for this Ligand-Target Pair
TargetPC4 and SFRS1-interacting protein(Homo sapiens (Human))
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM12590((6-aminoacridin-3-yl)amine | MLS003876812 | Profla...)
Affinity DataIC50:  4.34E+3nMAssay Description:Source (MLPCN Center Name): The Scripps Research Institute Molecular Screening Center (SRIMSC) Affiliation: Ohio State University Assay Provider: Mam...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetPC4 and SFRS1-interacting protein(Homo sapiens (Human))
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM12590((6-aminoacridin-3-yl)amine | MLS003876812 | Profla...)
Affinity DataIC50:  4.46E+3nMAssay Description:Source (MLPCN Center Name): The Scripps Research Institute Molecular Screening Center (SRIMSC) Affiliation: Ohio State University Assay Provider: Mam...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
Southern Research Institute

Curated by PubChem BioAssay
LigandPNGBDBM12590((6-aminoacridin-3-yl)amine | MLS003876812 | Profla...)
Affinity DataIC50:  8.88E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetProthrombin(Homo sapiens (Human))
Astex

LigandPNGBDBM12590((6-aminoacridin-3-yl)amine | MLS003876812 | Profla...)
Affinity DataIC50:  1.20E+4nMpH: 8.0 T: 2°CAssay Description:The cleavage of the substrate was followed by monitoring the change in fluorescence at 460 nm (excitation at 365 nm) for 25 min at room temperature o...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed