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Found 8 of ic50 for monomerid = 18125
TargetExcitatory amino acid transporter 1(Homo sapiens (Human))
University Of Groningen

Curated by ChEMBL
LigandPNGBDBM18125((2S)-2-aminobutanedioic acid | Aspartate | CHEMBL2...)
Affinity DataIC50:  9.30E+3nMAssay Description:Inhibition of human EAAT1 expressed in HEK293 cells assessed as reduction in [3H]-D-Asp uptake incubated for 4 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExcitatory amino acid transporter 1(Homo sapiens (Human))
University Of Groningen

Curated by ChEMBL
LigandPNGBDBM18125((2S)-2-aminobutanedioic acid | Aspartate | CHEMBL2...)
Affinity DataIC50:  9.33E+3nMAssay Description:Inhibition of human EAAT1 expressed in HEK293 cells assessed as reduction in [3H]-D-Asp uptake incubated for 4 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExcitatory amino acid transporter 4(Rattus norvegicus)
University Of Groningen

Curated by ChEMBL
LigandPNGBDBM18125((2S)-2-aminobutanedioic acid | Aspartate | CHEMBL2...)
Affinity DataIC50:  1.10E+4nMAssay Description:Inhibition of rat EAAT4 expressed in tsA201 cells assessed as reduction in [3H]-D-Asp uptake incubated for 4 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExcitatory amino acid transporter 4(Rattus norvegicus)
University Of Groningen

Curated by ChEMBL
LigandPNGBDBM18125((2S)-2-aminobutanedioic acid | Aspartate | CHEMBL2...)
Affinity DataIC50:  1.10E+4nMAssay Description:Inhibition of rat EAAT4 expressed in tsA201 cells assessed as reduction in [3H]-D-Asp uptake incubated for 4 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExcitatory amino acid transporter 3(Homo sapiens (Human))
University Of Groningen

Curated by ChEMBL
LigandPNGBDBM18125((2S)-2-aminobutanedioic acid | Aspartate | CHEMBL2...)
Affinity DataIC50:  1.95E+4nMAssay Description:Inhibition of human EAAT3 expressed in HEK293 cells assessed as reduction in [3H]-D-Asp uptake incubated for 4 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetExcitatory amino acid transporter 3(Homo sapiens (Human))
University Of Groningen

Curated by ChEMBL
LigandPNGBDBM18125((2S)-2-aminobutanedioic acid | Aspartate | CHEMBL2...)
Affinity DataIC50:  2.00E+4nMAssay Description:Inhibition of human EAAT3 expressed in HEK293 cells assessed as reduction in [3H]-D-Asp uptake incubated for 4 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetExcitatory amino acid transporter 2(Homo sapiens (Human))
University Of Groningen

Curated by ChEMBL
LigandPNGBDBM18125((2S)-2-aminobutanedioic acid | Aspartate | CHEMBL2...)
Affinity DataIC50:  3.20E+4nMAssay Description:Inhibition of human EAAT2 expressed in HEK293 cells assessed as reduction in [3H]-D-Asp uptake incubated for 4 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExcitatory amino acid transporter 2(Homo sapiens (Human))
University Of Groningen

Curated by ChEMBL
LigandPNGBDBM18125((2S)-2-aminobutanedioic acid | Aspartate | CHEMBL2...)
Affinity DataIC50:  3.31E+4nMAssay Description:Inhibition of human EAAT2 expressed in HEK293 cells assessed as reduction in [3H]-D-Asp uptake incubated for 4 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed