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Compile Data Set for Download or QSAR

Found 1 hit of ic50 for monomerid = 321396   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kJ/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
BRD9 (aa 134-239)


(Homo sapiens (Human))
BDBM321396
PNG
(3-[6-[(E)-but-2-enyl]-7-oxo-1H-pyrrolo[2,3-c]pyrid...)
Show SMILES COc1ccc(cc1-c1cn(C\C=C\C)c(=O)c2[nH]ccc12)C(=O)NCCN(C)C
Show InChI InChI=1S/C23H28N4O3/c1-5-6-12-27-15-19(17-9-10-24-21(17)23(27)29)18-14-16(7-8-20(18)30-4)22(28)25-11-13-26(2)3/h5-10,14-15,24H,11-13H2,1-4H3,(H,25,28)/b6-5+
PDB

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PC cid
PC sid
UniChem
US Patent
n/an/a 23n/an/an/an/an/an/a



GENENTECH, INC.; CONSTELLATION PHARMACEUTICALS, INC.

US Patent


Assay Description
His/Flag epitope tagged BRD9134-239 was cloned, expressed, and purified to homogeneity. BRD9 binding and inhibition was assessed by monitoring the en...


US Patent US10183009 (2019)

More data for this
Ligand-Target Pair