Compile Data Set for Download or QSAR
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Found 2 of ic50 for monomerid = 50080092
TargetSolute carrier family 22 member 1(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50080092((17beta)-17-hydroxyestr-4-en-3-one | 17beta-hydrox...)
Affinity DataIC50:  3.51E+4nMAssay Description:Inhibition of 4-(4-(dimethylamino)styryl)-N-methylpyridinium uptake at human OCT1 expressed in HEK293 cells by confocal microscopyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1,/2,/3,/4, mitochondrial(Homo sapiens (Human))
Novartis Institute For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50080092((17beta)-17-hydroxyestr-4-en-3-one | 17beta-hydrox...)
Affinity DataIC50:  1.20E+5nMAssay Description:In vitro inhibitory activity against pyruvate dehydrogenase kinase was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed