Affinity DataIC50: 0.210nMAssay Description:Antagonist activity at BLT1 receptor expressed in human HL60 cells assessed as inhibition of LTB4-stimulated calcium flux after 30 minsMore data for this Ligand-Target Pair
Affinity DataIC50: 38.5nMAssay Description:Antagonist activity at FLAG-tagged human BLT1 receptor expressed in HEK293 cells assessed as inhibition of LTB4-stimulated calcium mobilization prein...More data for this Ligand-Target Pair
Affinity DataIC50: 628nMAssay Description:Antagonist activity at FLAG-tagged human BLT2 receptor expressed in HEK293 cells assessed as inhibition of LTB4-stimulated calcium mobilization prein...More data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Roche Research Center
Curated by ChEMBL
Roche Research Center
Curated by ChEMBL
Affinity DataIC50: >3.00E+3nMAssay Description:Inhibition of human ERG expressed in CHO cells assessed as reduction of current amplitudeMore data for this Ligand-Target Pair
Affinity DataIC50: >7.50E+3nMAssay Description:Inhibition of CYP1A2 by fluorescence methodMore data for this Ligand-Target Pair
Affinity DataIC50: >7.50E+3nMAssay Description:Inhibition of CYP3A4 fluorescence methodMore data for this Ligand-Target Pair
Affinity DataIC50: >7.50E+3nMAssay Description:Inhibition of CYP2D6 flourescence methodMore data for this Ligand-Target Pair
Affinity DataIC50: >7.50E+3nMAssay Description:Inhibition of CYP2C19 flourescence methodMore data for this Ligand-Target Pair
Affinity DataIC50: >1.25E+4nMAssay Description:Inhibition of CYP2C9 by LC/MS methodMore data for this Ligand-Target Pair
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of CYP2C9 fluorescence methodMore data for this Ligand-Target Pair